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KINOMEscan℠ Webinar Series

Accelerating kinase drug discovery

In this webinar series, we showcase how KINOMEscan, DiscoverX's premier kinase profiling solution, can address your kinase drug discovery challenges from discovery to lead optimization and beyond.  Topics covered include general technology overview as well as focused topics covering experimental set up (how to design screens) and data analysis.
 
Webinars will continue to be added to this series, please check back often.

 


Event Date ▼ Event Name PDF Link Webinar Link
December 7, 2016 Webinar: The Interplay of Kinase Broad Profiling and Phenotypic Screening - 60 min.

What will be covered?

  • Learn about the significance of kinase broad profiling and phenotypic screening on early kinase drug discovery
  • Learn how to design a kinase inhibitor broad profiling project and how the chemo-bioinformatic analysis can impact target deconvolution after phenotypic screening
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July 20, 2016 Webinar: Introduction to KINOMEscan: Broad Applications to Drive Drug Discovery - 60 min.

What will be covered?

  • Overview of the KINOMEscan assay technology
  • Application of the KINOMEscan platform for selectivity and potency optimization
  • Development of chemical probes for understudied kinases
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June 17, 2016 データまで二週間:キナーゼ・ブロモドメイン・アポトーシス阻害剤を評価 - 60 min.

What will be covered?

  • KINOMEscanアッセイ原理の詳細:結合系と機能系を比較
  • 新規キナーゼ標的:CDK10, CDK12, CDK20, MLKL and MLKL (full length), IRAK2 等
  • 40種類ものブロモドメインに対する阻害剤を評価
  • アポトーシス阻害剤の同定:BCL2scan
  • scanMAX報告書から得られる、裏データ・裏情報のご紹介
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March 16, 2016 KINOMEscan Profiling Services Webinar: Efficient Design and Interpretation of KINOMEscan Experiments: A Driver for All Stages of Drug Development - 60 min.

What will be covered?

  • Application of KINOMEscan technology for selectivity and potency optimization of your lead molecules
  • Design scanMAX, KdELECT or scanELECT experiments
  • Improved flexibility of custom panels for hit identification, hit to lead, SAR and lead optimization
  • 20 new kinase assays launched in 2016
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October 14, 2015 Introduction to KINOMEscan® - Kinase Screening and Profiling Services - 35 min.

What will be covered

  • Overview of the KINOMEscan technology
  • Analysis of the KINOMEscan study report and included data information
  • Application of the KINOMEscan platform for Selectivity and Potency optimization
  • Data visualization tool: TREEspot
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June 11, 2015 Extracting Maximum Value from KINOMEscan®: Study Report Interpretation - 60 min.

What will be covered

  • Overview of the KINOMEscan technology platform
  • Explanation of the data included in the KINOMEscan study report
  • Designing efficient strategies for KINOMEscan screening
  • Data analysis overview: frequently overlooked data provided by scanMAX® screens
  • An introduction to a useful data visualization tool: TREEspot
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November 18, 2014 Webinar: Efficient design and interpretation of KINOMEscan® inhibitor profiling experiments - 60 min.

What will be covered?

  • Overview of the KINOMEscan assay technology
  • Experimental design:  strategies for choosing a screening concentration
  • Interpretation of screening data: what to study and what to ignore
  • Predicting inhibitor affinities from single point screening data
  • Efficient strategies for designing follow-up experiments
  • Selectivity is in the eye of the beholder: data visualization using TREEspot™ and Scatter Plots
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March 26, 2014 Extracting Maximum Value from KINOMEscan: Study Report Interpretation - 60 min.

What will be covered?

  • Overview of the KINOMEscan assay technology
  • Analysis of the KINOMEscan study report and included data information
  • Refresher on efficient strategies for designing KINOMEscan experiments
  • Data analysis overview:  frequently overlooked data provided by scanMAX screens
  • Data visualization tools: TREEspot
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March 19, 2013 Beyond Potency & Selectivity: Why Are Binding Kinetics Valuable In Kinase Drug Discovery? - 60 min.

What will be covered?

• KINOMEscan Technology: Applications for selectivity & potency optimization
scanMODE: Technology overview and applications
scanKINETIC: Technology overview and applications
• Key platform benefits
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