Family ▲ | Target Gene | Common Name | Arrestin | cAMP | Calcium | Internalization |
5-Hydroxytryptamine | HTR1A | 5-hydroxytryptamine receptor 1A (5HT1A) | X | X | | |
5-Hydroxytryptamine | HTR1B | 5-hydroxytryptamine receptor 1B (5HT1B) | X | X | | |
5-Hydroxytryptamine | HTR1F | 5-hydroxytryptamine receptor 1F (5HT1F) | X | X | | |
5-Hydroxytryptamine | HTR2A | 5-hydroxytryptamine receptor 2A (5HT2A) | X | | X | |
5-Hydroxytryptamine | HTR2B | 5-hydroxytryptamine receptor 2B (5HT2B) | | | X | |
5-Hydroxytryptamine | HTR2C | 5-hydroxytryptamine receptor 2C (5HT2C) | X | | X | X |
5-Hydroxytryptamine | HTR2C(VGV) | 5-hydroxytryptamine receptor 2C - VGV isoform (5HT2C) | X | | | |
5-Hydroxytryptamine | HTR2C(VNV) | 5-hydroxytryptamine receptor 2C - VNV isoform (5HT2C) | X | | | |
5-Hydroxytryptamine | HTR2C(VSV) | 5-hydroxytryptamine receptor 2C - VSV isoform (5HT2C) | X | | | |
5-Hydroxytryptamine | HTR5A | 5-hydroxytryptamine receptor 5A (5HT5A) | X | X | | |
5-Hydroxytryptamine | HTR6 | 5-hydroxytryptamine receptor 6 (5HT6) | X | | | |
5-Hydroxytryptamine | HTR7D | 5-hydroxytryptamine receptor 7D (5HT7D) | | X | | |
5-Hydroxytryptamine | mHTR2A | 5-Hydroxytryptamine receptor 2A (m5HT2A) | X | | | |
5-Hydroxytryptamine | mHTR2C | 5-Hydroxytryptamine receptor 2C (m5HT2C) | X | | | |
5-Hydroxytryptamine | rHTR2C | 5-hydroxytryptamine receptor 2C (HTR2C) | X | | | |
5-Hydroxytryptamine | HTR1E | 5-hydroxytryptamine receptor 1E (5HT1E) | X | | | |
Acetylcholine | rCHRM4 | Cholinergic receptor, muscarinic 4 (rM4) | X | | | |
Acetylcholine | CHRM1 | Cholinergic receptor, muscarinic 1 (M1) | X | | X | X |
Acetylcholine | CHRM2 | Cholinergic receptor, muscarinic 2 (M2) | X | X | | X |
Acetylcholine | CHRM3 | Cholinergic receptor, muscarinic 3 (M3) | X | | X | X |
Acetylcholine | CHRM4 | Cholinergic receptor, muscarinic 4 (M4) | X | X | | X |
Acetylcholine | CHRM5 | Cholinergic receptor, muscarinic 5 (M5) | X | | X | X |
Adenosine | ADORA1 | Adenosine receptor A1 (A1) | X | X | | |
Adenosine | ADORA2A | Adenosine receptor A2A (A2A) | | | X | |
Adenosine | ADORA2B | Adenosine receptor A2B (A2B) | | X | | |
Adenosine | ADORA3 | Adenosine receptor A3 (A3) | X | X | | |
Adenosine | mADORA2B | Adenosine receptor A2B (mA2B) | X | | | |
Adenosine | mADORA3 | adenosine receptor A3 (mA3) | X | | | |
Adrenoceptors | ADRA1A | Adrenergic receptor alpha 1A (α1A-adrenoceptor) | | | X | |
Adrenoceptors | ADRA1B | Adrenergic receptor alpha 1B (α1B-adrenoceptor) | X | | X | |
Adrenoceptors | ADRA2A | Adrenergic receptor alpha 2A (α2A-adrenoceptor) | X | X | | |
Adrenoceptors | ADRA2B | Adrenergic receptor alpha 2B (α2B-adrenoceptor) | X | | | |
Adrenoceptors | ADRA2C | Adrenergic receptor alpha 2C (α2C-adrenoceptor) | X | X | | X |
Adrenoceptors | ADRB1 | Adrenergic receptor beta 1 (β1-adrenoreceptor) | X | X | | |
Adrenoceptors | ADRB2 | Adrenergic receptor beta 2 (β2-adrenoreceptor) | X | X | | X |
Adrenoceptors | ADRB3 | Adrenergic receptor beta 3 (β3-adrenoreceptor) | | X | | |
Adrenoceptors | ADRA1D(82-572) | Adrenergic receptor alpha 1D (α1D-adrenoceptor) | X | | | |
Angiotensin | AGTR1 | Angiotensin II receptor, type 1 (AT1) | X | | X | |
Apelin | AGTRL1 | Apelin receptor (APJ) | X | X | | X |
Apelin | mAGTRL1 | Apelin receptor (mAPJ) | X | | | |
Bile acid | GPBAR1 | G protein-coupled bile acid receptor 1 (GPBA) | X | X | | |
Bombesin | BRS3 | Bombesin receptor, subtype 3 (BB3) | X | | X | |
Bombesin | GRPR | Gastrin releasing peptide receptor (BB2) | X | | X | X |
Bombesin | NMBR | Neuromedin B Receptor (BB1) | X | | X | X |
Bradykinin | BDKRB1 | Bradykinin receptor B1 (B1) | X | | X | |
Bradykinin | BDKRB2 | Bradykinin receptor B2 (B2) | X | | X | X |
Calcitonin | CALCR | Calcitonin receptor (CT) | X | X | | |
Calcitonin | CALCRL-RAMP1 | Calcitonin receptor-like (Calcitonin receptor-like receptor) | X | X | | |
Calcitonin | CALCRL-RAMP2 | Calcitonin receptor-like (Calcitonin receptor-like receptor) | X | | | |
Calcitonin | CALCRL-RAMP3 | Calcitonin receptor-like (Calcitonin receptor-like receptor) | X | X | | |
Calcitonin | CALCR-RAMP2 | Calcitonin receptor (CT) | X | X | | |
Calcitonin | CALCR-RAMP3 | Calcitonin receptor (CT) | X | X | | |
Calcium sensing | CASR | Calcium-sensing receptor (CaS) | | | X | |
Cannabinoid | CNR1 | Cannabinoid receptor 1 (CB1) | X | X | | |
Cannabinoid | CNR2 | Cannabinoid receptor 2 (CB2) | X | X | | |
Cannabinoid | mCNR1 | Cannabinoid receptor 1 (mCB1) | X | | | |
Cannabinoid | mCNR2 | Cannabinoid receptor 2 (mCB2) | X | | | |
Cannabinoid | rCNR2 | Cannabinoid receptor 2 (CB2) | X | | | |
Chemerin | CMKLR1 | Chemokine-like receptor 1 (CMKLR1) | X | X | | X |
Chemokine | CCR1 | Chemokine (C-C motif) receptor 1 (CCR1) | X | X | | X |
Chemokine | CCR10 | Chemokine (C-C motif) receptor 10 (CCR10) | X | X | | X |
Chemokine | CCR2 | Chemokine (C-C motif) receptor 2 (CCR2) | X | | | X |
Chemokine | CCR3 | Chemokine (C-C motif) receptor 3 (CCR3) | X | | | |
Chemokine | CCR4 | Chemokine (C-C motif) receptor 4 (CCR4) | X | | | X |
Chemokine | CCR5 | Chemokine (C-C motif) receptor 5 (CCR5) | X | X | | X |
Chemokine | CCR6 | Chemokine (C-C motif) receptor 6 (CCR6) | X | X | | X |
Chemokine | CCR7 | Chemokine (C-C motif) receptor 7 (CCR7) | X | X | | X |
Chemokine | CCR8 | Chemokine (C-C motif) receptor 8 (CCR8) | X | | | |
Chemokine | CCR9 | Chemokine (C-C motif) receptor 9 (CCR9) | X | | | |
Chemokine | CCRL1 | chemokine (C-C motif) receptor-like 1 (CCRL1) | X | | | |
Chemokine | CCRL2 | Chemokine (C-C motif) receptor-like 2 (CCRL2) | X | | | |
Chemokine | CX3CR1 | Chemokine C-X3-C receptor 1 (CX3CR1) | X | | | |
Chemokine | CXCR1 | Chemokine (C-X-C motif) receptor 1 (CXCR1) | X | X | | X |
Chemokine | CXCR2 | Chemokine (C-X-C motif) receptor 2 (CXCR2) | X | X | | X |
Chemokine | CXCR3 | Chemokine (C-X-C motif) receptor 3 (CXCR3) | X | X | | X |
Chemokine | CXCR4 | Chemokine (C-X-C motif) receptor 4 (CXCR4) | X | X | | X |
Chemokine | CXCR5 | Burkitt lymphoma receptor (CXCR5) | X | X | | |
Chemokine | CXCR6 | Chemokine (C-X-C motif) receptor 6 (CXCR6) | X | | | |
Chemokine | CXCR7 | Chemokine (C-X-C motif) receptor 7 (CXCR7) | X | | | X |
Chemokine | cyno CXCR1 | Chemokine (C-X-C motif) receptor 1 (CXCR1) | X | | | |
Chemokine | cyno CXCR2 | Chemokine (C-X-C motif) receptor 2 (CXCR2) | X | | | |
Chemokine | DARC | Duffy blood group, chemokine receptor (FY) | X | | | |
Chemokine | mCX3CR1 | Chemokine (C-X3-C motif) receptor 1 (mCX3CR1) | X | | | |
Chemokine | mCXCR2 | Chemokine (C-X-C motif) receptor 2 (mCXCR2) | X | | | |
Chemokine | mCXCR3 | Chemokine (C-X-C motif) receptor 3 (mCXCR3) | X | | | |
Chemokine | mCXCR4 | Chemokine (C-X-C motif) receptor 4 (mCXCR4) | X | | | |
Chemokine | mCXCR5 | Burkitt lymphoma receptor (mCXCR5) | X | | | |
Chemokine | mCXCR6 | Chemokine (C-X-C motif) receptor 6 (mCXCR6) | X | | | |
Chemokine | mCXCR7 | Chemokine (C-X-C motif) receptor 7 (mCXCR7) | X | | | |
Chemokine | mCCR1 | Chemokine (C-C motif) receptor 1 (mCC1) | X | | | |
Chemokine | mCCR2 | Chemokine (C-C motif) receptor 2 (mCCR2) | X | | | |
Chemokine | mCCR3 | Chemokine (C-C motif) receptor 3 (mCCR3) | X | | | |
Chemokine | mCCR4 | Chemokine (C-C motif) receptor 4 (mCCR4) | X | | | |
Chemokine | mCCR5 | Chemokine (C-C motif) receptor 5 (mCCR5) | X | | | |
Chemokine | mCCR6 | Chemokine (C-C motif) receptor 6 (mCCR6) | X | | | |
Chemokine | mCCR7 | Chemokine (C-C motif) receptor 7 (mCCR7) | X | | | |
Chemokine | mCCR8 | Chemokine (C-C motif) receptor 8 (mCCR8) | X | | | |
Chemokine | mCCR9 | Chemokine (C-C motif) receptor 9 (mCCR9) | X | | | |
Chemokine | mCMKLR1 | Chemokine-Like Receptor 1 (mCMKLR1) | X | | | |
Cholecystokinin | CCKAR | Cholecystokinin A receptor (CCK1) | X | | X | X |
Cholecystokinin | CCKBR | Cholecystokinin B receptor (CCK2) | X | | X | X |
Class A Orphan | EBI2 | G protein-coupled receptor 183 (GPR183) | X | X | | X |
Class A Orphan | GPR1 | G-protein coupled receptor 1 (GPR1) | X | | | X |
Class A Orphan | GPR101 | G-protein coupled receptor 101 (GPR101) | X | | | |
Class A Orphan | GHSR1b | Growth hormone secretagogue receptor 1b (GHSR1b) | X | | | |
Class A Orphan | GPR119 | G-protein coupled receptor 119 (GPR119) | X | | | |
Class A Orphan | GPR12 | G-protein coupled receptor 12 (GPR12) | X | | | |
Class A Orphan | GPR132 | G-protein coupled receptor 132 (GPR132) | X | | | |
Class A Orphan | GPR135 | G-protein coupled receptor 135 (GPR135) | X | | | |
Class A Orphan | GPR139 | G-protein coupled receptor 139 (GPR139) | X | | | |
Class A Orphan | GPR141 | G-protein coupled receptor 141 (GPR141) | X | | | |
Class A Orphan | GPR142 | G-protein coupled receptor 142 (GPR142) | X | | | |
Class A Orphan | GPR146 | G-protein coupled receptor 146 (GPR146) | X | | | |
Class A Orphan | GPR148 | G-protein coupled receptor 148 (GPR148) | X | | | |
Class A Orphan | GPR149 | G-protein coupled receptor 149 (GPR149) | X | | | |
Class A Orphan | GPR15 | G-protein coupled receptor 15 (GPR15) | X | | | |
Class A Orphan | GPR150 | G-protein coupled receptor 150 (GPR150) | X | | | |
Class A Orphan | GPR151 | G-protein coupled receptor 151 (GPR151) | X | | | |
Class A Orphan | GPR152 | G-protein coupled receptor 152 (GPR152) | X | | | |
Class A Orphan | GPR31 | G-protein coupled receptor 31 (GPR31) | X | | | |
Class A Orphan | GPR32 | G-protein coupled receptor 32 (GPR32) | X | | | |
Class A Orphan | GPR35 | G-protein coupled receptor 35 (GPR35) | X | X | | X |
Class A Orphan | GPR37 | Endothelin B receptor-like (EDNRBL) | X | | | |
Class A Orphan | GPR37L1 | G protein-coupled receptor 37 like 1 (GPR37L1) | X | | | |
Class A Orphan | GPR39 | G-protein coupled receptor 39 (GPR39) | X | | X | |
Class A Orphan | GPR4 | G-protein coupled receptor 4 (GPR4) | X | | | |
Class A Orphan | GPR45 | G-protein coupled receptor 45 (GPR45) | X | | | |
Class A Orphan | GPR50 | G-protein coupled receptor 50 (GPR50) | X | | | |
Class A Orphan | GPR52 | G-protein coupled receptor 52 (GPR52) | X | | | |
Class A Orphan | GPR55 | G protein-coupled receptor 55 (GPR55) | X | | | |
Class A Orphan | GPR6 | G-protein coupled receptor 6 (GPR6) | X | | | |
Class A Orphan | GPR61 | G-protein coupled receptor 61 (GPR61) | X | | | |
Class A Orphan | GPR65 | G-protein coupled receptor 65 (GPR65) | X | | | |
Class A Orphan | GPR75 | G-protein coupled receptor 75 (GPR75) | X | | | |
Class A Orphan | GPR78 | G-protein coupled receptor 78 (GPR78) | X | | | |
Class A Orphan | GPR79 | G protein-coupled receptor 79 pseudogene (GPR79) | X | | | |
Class A Orphan | MRGPRD | MAS-related GPR, member D (MRGPRD) | X | | | |
Class A Orphan | MRGPRE | MAS-related GPR, member E (MRGPRE) | X | | | |
Class A Orphan | MRGPRF | MAS-related GPR, member F (MRGPRF) | X | | | |
Class A Orphan | MRGPRX1 | MAS-related GPR, member X1 (MRGPRX1) | X | | X | |
Class A Orphan | MRGPRX2 | MAS-related GPR, member X2 (MRGX2) | X | | X | |
Class A Orphan | MRGPRX4 | MAS-related GPR, member X4 (MRGPRX4) | X | | | |
Class A Orphan | OPN5 | Opsin 5 (OPN5) | X | | | |
Class A Orphan | mGPR1 | G-Protein Coupled Receptor 1 (mGPR1) | X | | | |
Class A Orphan | OXGR1 | Oxoglutarate (alpha-ketoglutarate) receptor 1 (OXGR1) | X | | X | |
Class A Orphan | mEBI2 | G-protein coupled receptor 183 (GPR183) | X | | | |
Class A Orphan | LGR4 | Leucine-rich repeat-containing G protein-coupled receptor 4 (LGR4) | X | | | |
Class A Orphan | LGR5 | Leucine-rich repeat-containing G protein-coupled receptor 5 (LGR5) | X | | | |
Class A Orphan | LGR6 | Leucine-rich repeat-containing G protein-coupled receptor 6 (LGR6) | X | | | |
Class A Orphan | GPR161 | G-protein coupled receptor 161 (GPR161) | X | | | |
Class A Orphan | GPR162 | G-protein coupled receptor 162 (GPR162) | X | | | |
Class A Orphan | GPR17 | G-protein coupled receptor 17 (GPR17) | X | | X | |
Class A Orphan | GPR171 | G-protein coupled receptor 171 (GPR171) | X | | | |
Class A Orphan | GPR173 | G-protein coupled receptor 173 (GPR173) | X | | | |
Class A Orphan | GPR176 | G-protein coupled receptor 176 (GPR176) | X | | | |
Class A Orphan | GPR18 | G-protein coupled receptor 18 (GPR18) | X | | | |
Class A Orphan | GPR182 | G-protein coupled receptor 182 (GPR182) | X | | | |
Class A Orphan | GPR20 | G-protein coupled receptor 20 (GPR20) | X | | | |
Class A Orphan | GPR23 | Lysophosphatidic acid receptor 4 (LPA4) | X | | | |
Class A Orphan | GPR25 | G-protein coupled receptor 25 (GPR25) | X | | | |
Class A Orphan | GPR26 | G-protein coupled receptor 26 (GPR26) | X | | | |
Class A Orphan | GPR27 | G-protein coupled receptor 27 (GPR27) | X | | | |
Class A Orphan | GPR3 | G-protein coupled receptor 3 (GPR3) | X | | | |
Class A Orphan | GPR83 | G-protein coupled receptor 83 (GPR83) | X | | | |
Class A Orphan | GPR84 | G-protein coupled receptor 84 (GPR84) | X | X | | |
Class A Orphan | GPR85 | G-protein coupled receptor 85 (GPR85) | X | | | |
Class A Orphan | GPR88 | G-protein coupled receptor 88 (GPR88) | X | | | |
Class A Orphan | P2RY8 | Purinergic receptor P2Y, G-protein coupled, 8 (P2RY8) | X | | | |
Class A Orphan | TAAR5 | Trace amine associated receptor 5 (TAAR5) | X | | | |
Class A Orphan | rGPR35 | G-protein coupled receptor 35 (rGPR35) | X | | | |
Class A Orphan | mGPR84 | G-protein coupled receptor 84, Mouse (GPR84) | X | | | |
Class A Orphan | GPR22 | G-protein coupled receptor 22 (GPR22) | X | | | |
Class B Orphan | GPR97 | G-protein coupled receptor 97 (GPR97) | X | | | |
Class B Orphan | GPR123 | G-protein coupled receptor 123 (GPR123) | X | | | |
Class B Orphan | GPR157 | G-protein coupled receptor 157 (GPR157) | X | | | |
Class B Orphan | BAI1 | Brain-specific angiogenesis inhibitor 1 (BAI1) | X | | | |
Class B Orphan | BAI2 | Brain-specific angiogenesis inhibitor 2 (BAI2) | X | | | |
Class B Orphan | BAI3 | Brain-specific angiogenesis inhibitor 3 (BAI3) | X | | | |
Complement peptide | C3AR1 | Complement component 3a receptor 1 (C3A) | X | | | |
Complement peptide | C5AR1 | Complement component 5a receptor 1 (C5A) | X | X | | X |
Complement peptide | C5L2 | G-Protein Coupled Receptor 77 (C5L2) | X | | | X |
Complement peptide | mC5AR1 | Complement component 5a receptor 1 (mC5AR) | X | | | |
Corticotropin-releasing factor | mCRHR1 | Corticotropin releasing hormone receptor 1 (mCRF1) | X | | | |
Corticotropin-releasing factor | CRHR1 | Corticotropin releasing hormone receptor 1 (CRF1) | X | X | | X |
Corticotropin-releasing factor | CRHR2 | Corticotropin releasing hormone receptor 2 (CRF2) | X | X | | X |
Dopamine | DRD1 | Dopamine receptor D1 (D1) | X | X | | X |
Dopamine | DRD2L | Dopamine Receptor D2 (long isoform) (D2L) | X | X | | |
Dopamine | DRD2S | Dopamine Receptor D2 (short isoform) (D2S) | X | X | | |
Dopamine | DRD3 | Dopamine Receptor D3 (D3) | X | | | |
Dopamine | DRD4 | Dopamine Receptor D4 (D4) | X | X | | |
Dopamine | DRD5 | Dopamine receptor D5 (D5) | X | X | | |
Dopamine | mDRD5 | Dopamine receptor D5 (mDRD5) | X | | | |
Dopamine | rDRD1 | Dopamine receptor D1 (rD1) | X | | | |
Dopamine | rDRD2L | Dopamine Receptor D2 (long isoform) (rD2L) | X | | | |
Dopamine | rDRD2S | Dopamine Receptor D2 (short isoform) (rD2S) | X | | | |
Endothelin | mEDNRA | Endothelin receptor type A (mETA) | X | | | |
Endothelin | mEDNRB | Endothelin receptor type B (mETB) | X | | | |
Endothelin | EDNRA | Endothelin receptor type A (ETA) | X | | X | |
Endothelin | EDNRB | Endothelin receptor type B (ETB) | X | | | X |
Estrogen (G protein coupled) receptor | GPR30 | G protein-coupled estrogen receptor 1 (GPER) | X | | | |
Formylpeptide | mFPR1 | Formylpeptide receptor 1 (mFPR1) | X | | | |
Formylpeptide | mFPR2 | Formylpeptide receptor 2 (FPR2) | X | | | |
Formylpeptide | FPR1 | Formylpeptide receptor 1 (FPR1) | X | X | | X |
Formylpeptide | FPR3 | Formyl peptide receptor 3 (FPRL2) | | X | | |
Formylpeptide | FPRL1 | Formylpeptide receptor-like 1 (FPR2/ALX) | X | X | | X |
Free fatty acid | GPR120 | G-protein coupled receptor 120, long isoform (FFA4) | X | | | X |
Free fatty acid | GPR120S | G-protein Coupled Receptor 120, short isoform (FFA4) | X | | | |
Free Fatty Acid | FFAR1 | Free fatty acid receptor 1 (FFA1) | X | | X | |
Free Fatty Acid | FFAR2 | Free fatty acid receptor 2 (GPR43) | | | X | |
Free Fatty Acid | FFAR3 | Free fatty acid receptor 3 (GPR41) | | X | | |
Free fatty acid | cyno GPR120 | G-protein coupled receptor 120 (FFA4) | X | | | |
Free Fatty Acid | mFFAR1 | Free fatty acid receptor 1 (FFA1) | X | | | |
Free Fatty Acid | rFFAR1 | Free fatty acid receptor 1 (FFA1) | X | | | |
Free fatty acid | rGPR120 | G-protein coupled receptor 120 (FFA4) | X | | | |
GABAB | GABBR1-GABBR2 | gamma-aminobutyric acid (GABA) B receptor, 1 (GABB1) | | X | | |
Galanin | GALR1 | Galanin receptor 1 (GALR1) | X | X | | X |
Galanin | GALR2 | Galanin receptor 2 (GALR2) | X | | X | |
Galanin | mGALR2 | Galanin Receptor 2 (mGALR2) | X | | | |
Ghrelin | mGHSR | Ghrelin receptor (ghrelin) | X | | | |
Ghrelin | GHSR | Ghrelin receptor (ghrelin) | X | | X | |
Glucagon | GIPR | Gastric inhibitory polypeptide receptor (GIP) | X | X | | |
Glucagon | GLP1R | Glucagon-like peptide receptor 1 (GLP-1) | X | X | | X |
Glucagon | GLP2R | Glucagon-like peptide receptor 2 (GLP-2) | X | X | | X |
Glucagon | GCGR | Glucagon receptor (glucagon) | X | X | | X |
Glucagon | GHRHR | Growth hormone releasing hormone receptor (GHRH) | | X | | |
Glucagon | mGIPR | Gastric inhibitory polypeptide receptor (mGIP) | X | | | |
Glucagon | mGLP1R | Glucagon-like peptide receptor 1 (mGLP-1) | X | | | |
Glucagon | mGCGR | Glucagon Receptor (glucagon) | X | | | |
Glucagon | SCTR | Secretin receptor (secretin) | X | X | | X |
Glycoprotein hormone receptor | TSHR(L) | Thyroid Stimulating Hormone Receptor (TSH) | X | X | | |
Glycoprotein hormone receptor | LHCGR | Choriogonadotropin receptor (LH) | X | X | | |
Glycoprotein hormone receptor | FSHR | Follicle stimulating hormone receptor (FSHR) | X | X | | |
Gonadotropin-releasing hormone | GNRHR | Gonadotropin-releasing hormone receptor (GnRH) | | | X | |
Histamine | HRH1 | Histamine receptor H1 (H1) | X | | X | |
Histamine | HRH2 | Histamine receptor H2 (H2) | X | X | X | |
Histamine | HRH3 | Histamine receptor H3 (H3) | X | X | | |
Histamine | HRH4 | Histamine receptor H4 (H4) | X | | | |
Hydroxycarboxylic acid | GPR109A | Hydroxycarboxylic acid receptor 2 (HCA2) | X | X | | |
Hydroxycarboxylic acid | GPR109B | Hydroxycarboxylic acid receptor 3 (HCA3) | X | X | | |
Hydroxycarboxylic acid | GPR81 | Hydroxycarboxylic acid receptor 1 (HCA1) | | X | | |
Kisspeptin receptor | KISS1R | KISS1-derived peptide receptor (kisspeptin) | X | | | |
Leukotriene | LTB4R | Leukotriene B4 receptor (BLT1) | X | X | X | X |
Leukotriene | mLTB4R | Leukotriene B4 receptor (mBLT1) | X | | | |
Leukotriene | OXER1 | Oxoeicosanoid (OXE) receptor 1 (OXE) | X | X | | X |
Leukotriene | CYSLTR2 | Cysteinyl leukotriene receptor 2 (CYSLT2) | | | X | |
Lysophospholipid (LPA) | EDG2 | Lysophosphatidic acid receptor 1 (LPA1) | | | X | X |
Lysophospholipid (LPA) | EDG4 | Lysophosphatidic acid receptor 2 (LPA2) | X | | X | |
Lysophospholipid (LPA) | EDG7 | Lysophosphatidic acid receptor 3 (LPA3) | X | | X | X |
Lysophospholipid (LPA) | GPR92 | Lysophosphatidic acid receptor 5 (GPR92) | X | | X | |
Lysophospholipid (S1P) | mEDG1 | Sphingosine 1-phosphate receptor 1 (mS1P1) | X | | | |
Lysophospholipid (S1P) | mEDG3 | Sphingosine 1-phosphate receptor 3 (S1P3) | X | | | |
Lysophospholipid (S1P) | mEDG5 | Sphingosine 1-phosphate receptor 2 (mS1P2) | X | | | |
Lysophospholipid (S1P) | EDG5 | Sphingosine 1-phosphate receptor 2 (S1P2) | X | | | X |
Lysophospholipid (S1P) | EDG6 | Sphingosine 1-phosphate receptor 4 (S1P4) | X | | | |
Lysophospholipid (S1P) | EDG3 | Sphingosine 1-phosphate receptor 3 (S1P3) | X | | X | X |
Lysophospholipid (S1P) | EDG1 | Sphingosine 1-phosphate receptor 1 (S1P1) | X | X | | X |
Lysophospholipid (S1P) | cEDG5 | Sphingosine 1-phosphate receptor 2 (cS1P2) | X | | | |
Lysophospholipid (S1P) | sEDG5 | Sphingosine 1-phosphate receptor 2 (sS1P2) | X | | | |
Lysophospholipid (S1P) | rEDG5 | Sphingosine 1-phosphate receptor 2 (rS1P2) | X | | | |
Melanin-concentrating hormone | MCHR1 | Melanin concentrating hormone receptor 1 (MCH1) | X | X | | X |
Melanin-concentrating hormone | MCHR2 | Melanin-concentrating hormone receptor 2 (MCH2) | X | | X | |
Melanin-concentrating hormone | mMCHR1 | Melanin concentrating hormone receptor 1 (MCH1) | X | | | |
Melanocortin | MC5R | Melanocortin receptor 5 (MC5) | X | X | | |
Melanocortin | MC1R | Melanocortin receptor 1 (MC1) | X | X | | |
Melanocortin | MC3R | Melanocortin receptor 3 (MC3) | X | X | | X |
Melanocortin | MC4R | Melanocortin receptor 4 (MC4) | X | X | | |
Melatonin | MTNR1A | Melatonin receptor 1A (MT1) | X | X | | X |
Melatonin | MTNR1B | Melatonin receptor 1B (MT2) | X | X | | X |
Metabotropic glutamate | GRM1 | Metabotropic glutamate receptor 1 (mGlu1) | | | X | |
Metabotropic glutamate | GRM2 | Metabotropic glutamate receptor 2 (mGlu2) | | X | | |
Metabotropic glutamate | GRM3 | Metabotropic glutamate receptor 3 (MGlu3) | | X | | |
Metabotropic glutamate | GRM4 | Metabotropic glutamate receptor 4 (mGlu4) | | X | | |
Metabotropic glutamate | GRM5 | Metabotropic glutamate receptor 5 (mGlu5) | | | X | |
Metabotropic glutamate | GRM6 | Metabotropic glutamate receptor 6 (mGlu6) | | X | | |
Motilin | MLNR | Motilin receptor (motilin) | X | | X | X |
Neuromedin U | NMU1R | Neuromedin U receptor 1 (NMU1) | X | | X | X |
Neuropeptide B & W | NPBWR1 | Neuropeptides B/W receptor 1 (NPBW1) | X | X | | |
Neuropeptide B & W | NPBWR2 | Neuropeptides B/W receptor 2 (NPBW2) | X | X | | |
Neuropeptide FF & AF | NPFFR1 | Neuropeptide FF receptor 1 (NPFF1) | X | X | | |
Neuropeptide S | NPSR1b | neuropeptide S receptor 1 (NPS receptor) | X | | | |
Neuropeptide Y | NPY1R | Neuropeptide Y receptor Y1 (Y1) | X | | | |
Neuropeptide Y | NPY2R | Neuropeptide Y receptor Y2 (Y2) | X | X | X | X |
Neuropeptide Y | mPPYR1 | Pancreatic polypeptide receptor 1 (Y4) | X | | | |
Neuropeptide Y | mNPY1R | Neuropeptide Y1 receptor (Y1) | X | | | |
Neuropeptide Y | mNPY2R | Neuropeptide Y2 receptor (NPY2R) | X | | | |
Neuropeptide Y | PPYR1 | Pancreatic polypeptide receptor 1 (Y4) | X | X | | |
Neurotensin | NTSR1 | Neurotensin receptor 1 (NTS1) | X | | X | X |
Opioid | OPRD1 | Opioid receptor delta (δ) | X | X | | X |
Opioid | OPRK1 | Opioid receptor kappa (κ) | X | X | | X |
Opioid | OPRL1 | Opioid receptor-like receptor (NOP) | X | X | | X |
Opioid | OPRM1 | Opioid receptor mu (μ) | X | X | | X |
Opioid | mOPRD1 | Opioid receptor delta (δ (murine)) | X | | | |
Opioid | mOPRK1 | Opioid receptor kappa (κ (murine)) | X | | | |
Opioid | mOPRM1 | Opioid receptor mu (μ (murine)) | X | | | |
Opioid | rOPRM1 | Opioid receptor mu (μ) | X | | | |
Orexin | HCRTR1 | Orexin receptor 1 (OX1) | X | | X | X |
Orexin | HCRTR2 | Orexin receptor 2 (OX2) | X | | X | X |
Other 7TM proteins | GPR107 | G-protein coupled receptor 107 (GPR107) | X | | | |
Other 7TM proteins | GPR137 | G-protein coupled receptor 137B (TM7SF1) | X | | | |
Other 7TM proteins | GPR143 | G-protein coupled receptor 143 (GPR143) | X | | | |
P2Y | mP2RY12 | P2Y Purinoceptor 12 (mP2Y12) | X | | | |
P2Y | mP2RY6 | P2Y Purinoceptor 6 (P2Y6) | X | | | |
P2Y | P2RY1 | Purinergic receptor P2Y, G-protein coupled, 1 (P2RY1) | X | | X | X |
P2Y | P2RY11 | Purinergic receptor P2Y, G-protein coupled, 11 (P2Y11) | X | | | |
P2Y | P2RY12 | Purinergic receptor P2Y, G-protein coupled, 12 (P2Y12) | X | | | X |
P2Y | P2RY2 | Purinergic receptor P2Y, G-protein coupled, 2 (P2Y2) | X | | X | X |
P2Y | P2RY4 | Pyrimidinergic receptor P2Y, G-protein coupled, 4 (P2Y4) | X | | | X |
P2Y | P2RY6 | Pyrimidinergic receptor P2Y, G-protein coupled, 6 (P2Y6) | X | | | |
Parathyroid hormone | PTHR1 | Parathyroid hormone receptor 1 (PTH1) | X | X | X | X |
Parathyroid hormone | PTHR2 | Parathyroid hormone receptor 2 (PTH2) | X | X | X | X |
Peptide P518 | GPR103 | pyroglutamylated RFamide peptide receptor (QRFPR) | X | | X | |
Platelet-activating factor | PTAFR | Platelet activating receptor (PAF) | X | | X | X |
Platelet-activating factor | mPTAFR | Platelet-activating factor receptor (mPAF) | X | | | |
Prokineticin | PROKR1 | Prokineticin receptor 1 (PKR1) | X | X | X | X |
Prokineticin | PROKR2 | Prokineticin receptor 2 (PKR2) | X | | | X |
Prokineticin | rPROKR1 | Prokineticin receptor 1 (rPROKR1) | X | | | |
Prokineticin | rPROKR2 | Prokineticin receptor 2 (rPKR2) | X | | | |
Prolactin releasing peptide receptor | PRLHR | Prolactin releasing hormone receptor (PRRP) | X | | X | X |
Prostanoid | rCRTH2 | Prostanoid DP2 receptor (rGPR44) | X | | | |
Prostanoid | rPTGER4 | Prostaglandin E receptor 4 (subtype EP4), rat (rEP4) | X | | | |
Prostanoid | TBXA2R | Thromboxane A2 receptor (TP) | X | | X | X |
Prostanoid | mPTGER4 | Prostaglandin E receptor 4 (subtype EP4) (EP4) | X | | | |
Prostanoid | PTGDR | Prostaglandin D2 receptor (DP1) | | X | | |
Prostanoid | PTGER1 | Prostaglandin E receptor 1 (subtype EP1) (EP1) | X | | X | |
Prostanoid | PTGER2 | Prostaglandin E receptor 2 (subtype EP2) (EP2) | X | X | | |
Prostanoid | PTGER3 | Prostaglandin E receptor 3 (subtype EP3) (EP3) | X | X | X | |
Prostanoid | PTGER4 | Prostaglandin E receptor 4 (subtype EP4) (EP4) | X | | | X |
Prostanoid | PTGFR | Prostaglandin F receptor (FP) (FP) | X | | X | X |
Prostanoid | PTGIR | Prostaglandin I2 (prostacyclin) receptor (IP) (IP1) | X | X | | X |
Prostanoid | mCRTH2 | Prostanoid DP2 receptor (mDP2) | X | | | |
Prostanoid | CRTH2 | prostaglandin D2 receptor 2 (PTGDR2) | X | X | | |
Protease activated | F2R | Coagulation factor II (thrombin) receptor (PAR1) | X | | | |
Protease activated | F2RL1 | Coagulation factor II (thrombin) receptor-like 1 (PAR2) (PAR2) | X | | X | X |
Protease activated | F2RL3 | Coagulation factor II (thrombin) receptor-like 3 (PAR4) (PAR4) | X | | X | X |
Relaxin | mRXFP3 | Relaxin family peptide receptor 3 (RXFP3) | X | | | |
Relaxin | mRXFP4 | Relaxin family peptide receptor 4 (RXFP4) | X | | | |
Relaxin | RXFP1 | Relaxin family peptide receptor 1 (RXFP1) | | X | | |
Relaxin | RXFP2 | Relaxin family peptide receptor 2 (RXFP2) | | X | | |
Relaxin | RXFP3 | Relaxin family peptide receptor 3 (RXFP3) | X | X | | X |
Relaxin | RXFP4 | Relaxin family peptide receptor 4 (RXFP4) | X | X | | |
Somatostatin | SSTR1 | Somatostatin receptor 1 (SST1) | X | | | |
Somatostatin | SSTR2 | Somatostatin receptor 2 (SST2) | X | X | | X |
Somatostatin | SSTR3 | Somatostatin receptor 3 (SST3) | X | X | | |
Somatostatin | SSTR4 | Somatostatin receptor 4 (SST4) | X | X | | |
Somatostatin | SSTR5 | Somatostatin receptor 5 (SST5) | X | X | | |
Somatostatin | mSSTR2 | Somatostatin receptor 2 (mSST2) | X | | | |
Somatostatin | mSSTR5 | Somatostatin receptor 5 (mSRIF1B) | X | | | |
Tachykinin | TACR1 | Tachykinin receptor 1 (NK1) | X | | X | X |
Tachykinin | TACR2 | Tachykinin receptor 2 (NK2) | X | | X | X |
Tachykinin | TACR3 | Tachykinin receptor 3 (NK3) | X | X | X | X |
Thyrotropin releasing hormone | TRHR | Thyrotropin-releasing hormone receptor (TRH1) | X | | X | X |
Trace amine | TAAR1 | trace amine associated receptor 1 (TA1) | | X | | |
Urotensin | UTR2 | Urotensin II receptor (UT) | X | | X | X |
Urotensin | mUTR2 | Urotensin II receptor (mUT) | X | | | |
Vasopressin and Oxytocin | OXTR | Oxytocin Receptor (OT) | X | | X | X |
Vasopressin and Oxytocin | mOXTR | Oxytocin recepter (OT) | X | | | |
Vasopressin and Oxytocin | AVPR1A | Vasopressin receptor 1A (V1A) | X | | X | X |
Vasopressin and Oxytocin | AVPR1B | Vasopressin receptor 1B (V1B) | X | | X | X |
Vasopressin and Oxytocin | AVPR2 | Vasopressin receptor 2 (V2) | X | X | | X |
VIP and PACAP | ADCYAP1R1 | Adenylate cyclase activating polypeptide receptor 1 (PAC1) | X | X | X | X |
VIP and PACAP | mVIPR1 | Vasoactive intestinal peptide receptor 1 (mVPAC1) | X | | | |
VIP and PACAP | mADCYAP1R1 | Adenylate Cyclase Activating Polypeptide 1 Receptor 1 (mPAC1) | X | | | |
VIP and PACAP | VIPR1 | Vasoactive intestinal peptide receptor 1 (VPAC1) | X | X | X | X |
VIP and PACAP | VIPR2 | Vasoactive intestinal peptide receptor 2 (VPAC2) | X | X | X | X |
VIP and PACAP | rVIPR1 | Vasoactive intestinal peptide receptor 1 (rVPAC1) | X | | | |