Target Gene ▲ | Common Name | Arrestin | cAMP | Calcium | Internalization |
| | X | | | |
ADCYAP1R1 | Adenylate cyclase activating polypeptide receptor 1 (PAC1) | X | X | X | X |
ADORA1 | Adenosine receptor A1 (A1) | X | X | | |
ADORA3 | Adenosine receptor A3 (A3) | X | X | | |
ADRA1B | Adrenergic receptor alpha 1B (α1B-adrenoceptor) | X | | X | |
ADRA2A | Adrenergic receptor alpha 2A (α2A-adrenoceptor) | X | X | | |
ADRA2C | Adrenergic receptor alpha 2C (α2C-adrenoceptor) | X | X | | X |
ADRB1 | Adrenergic receptor beta 1 (β1-adrenoreceptor) | X | X | | |
ADRB2 | Adrenergic receptor beta 2 (β2-adrenoreceptor) | X | X | | X |
AGTR1 | Angiotensin II receptor, type 1 (AT1) | X | | X | |
AGTRL1 | Apelin receptor (APJ) | X | X | | X |
AVPR1A | Vasopressin receptor 1A (V1A) | X | | X | X |
AVPR1B | Vasopressin receptor 1B (V1B) | X | | X | X |
AVPR2 | Vasopressin receptor 2 (V2) | X | X | | X |
BDKRB1 | Bradykinin receptor B1 (B1) | X | | X | |
BDKRB2 | Bradykinin receptor B2 (B2) | X | | X | X |
BRS3 | Bombesin receptor, subtype 3 (BB3) | X | | X | |
C5AR1 | Complement component 5a receptor 1 (C5A) | X | X | | X |
C5L2 | G-Protein Coupled Receptor 77 (C5L2) | X | | | X |
CALCR | Calcitonin receptor (CT) | X | X | | |
CALCRL-RAMP1 | Calcitonin receptor-like (Calcitonin receptor-like receptor) | X | X | | |
CALCRL-RAMP3 | Calcitonin receptor-like (Calcitonin receptor-like receptor) | X | X | | |
CALCR-RAMP3 | Calcitonin receptor (CT) | X | X | | |
CCKAR | Cholecystokinin A receptor (CCK1) | X | | X | X |
CCKBR | Cholecystokinin B receptor (CCK2) | X | | X | X |
CCR1 | Chemokine (C-C motif) receptor 1 (CCR1) | X | X | | X |
CCR10 | Chemokine (C-C motif) receptor 10 (CCR10) | X | X | | X |
CCR2 | Chemokine (C-C motif) receptor 2 (CCR2) | X | | | X |
CCR4 | Chemokine (C-C motif) receptor 4 (CCR4) | X | | | X |
CCR5 | Chemokine (C-C motif) receptor 5 (CCR5) | X | X | | X |
CCR6 | Chemokine (C-C motif) receptor 6 (CCR6) | X | X | | X |
CCR7 | Chemokine (C-C motif) receptor 7 (CCR7) | X | X | | X |
CHRM1 | Cholinergic receptor, muscarinic 1 (M1) | X | | X | X |
CHRM2 | Cholinergic receptor, muscarinic 2 (M2) | X | X | | X |
CHRM3 | Cholinergic receptor, muscarinic 3 (M3) | X | | X | X |
CHRM4 | Cholinergic receptor, muscarinic 4 (M4) | X | X | | X |
CHRM5 | Cholinergic receptor, muscarinic 5 (M5) | X | | X | X |
CMKLR1 | Chemokine-like receptor 1 (CMKLR1) | X | X | | X |
CNR1 | Cannabinoid receptor 1 (CB1) | X | X | | |
CNR2 | Cannabinoid receptor 2 (CB2) | X | X | | |
CRHR1 | Corticotropin releasing hormone receptor 1 (CRF1) | X | X | | X |
CRHR2 | Corticotropin releasing hormone receptor 2 (CRF2) | X | X | | X |
CRTH2 | prostaglandin D2 receptor 2 (PTGDR2) | X | X | | |
CXCR1 | Chemokine (C-X-C motif) receptor 1 (CXCR1) | X | X | | X |
CXCR2 | Chemokine (C-X-C motif) receptor 2 (CXCR2) | X | X | | X |
CXCR3 | Chemokine (C-X-C motif) receptor 3 (CXCR3) | X | X | | X |
CXCR4 | Chemokine (C-X-C motif) receptor 4 (CXCR4) | X | X | | X |
CXCR5 | Burkitt lymphoma receptor (CXCR5) | X | X | | |
CXCR7 | Chemokine (C-X-C motif) receptor 7 (CXCR7) | X | | | X |
DRD1 | Dopamine receptor D1 (D1) | X | X | | X |
DRD2L | Dopamine Receptor D2 (long isoform) (D2L) | X | X | | |
DRD2S | Dopamine Receptor D2 (short isoform) (D2S) | X | X | | |
DRD4 | Dopamine Receptor D4 (D4) | X | X | | |
DRD5 | Dopamine receptor D5 (D5) | X | X | | |
EBI2 | G protein-coupled receptor 183 (GPR183) | X | X | | X |
EDG1 | Sphingosine 1-phosphate receptor 1 (S1P1) | X | X | | X |
EDG2 | Lysophosphatidic acid receptor 1 (LPA1) | | | X | X |
EDG3 | Sphingosine 1-phosphate receptor 3 (S1P3) | X | | X | X |
EDG4 | Lysophosphatidic acid receptor 2 (LPA2) | X | | X | |
EDG5 | Sphingosine 1-phosphate receptor 2 (S1P2) | X | | | X |
EDG7 | Lysophosphatidic acid receptor 3 (LPA3) | X | | X | X |
EDNRA | Endothelin receptor type A (ETA) | X | | X | |
EDNRB | Endothelin receptor type B (ETB) | X | | | X |
F2RL1 | Coagulation factor II (thrombin) receptor-like 1 (PAR2) (PAR2) | X | | X | X |
F2RL3 | Coagulation factor II (thrombin) receptor-like 3 (PAR4) (PAR4) | X | | X | X |
FFAR1 | Free fatty acid receptor 1 (FFA1) | X | | X | |
FPR1 | Formylpeptide receptor 1 (FPR1) | X | X | | X |
FPRL1 | Formylpeptide receptor-like 1 (FPR2/ALX) | X | X | | X |
FSHR | Follicle stimulating hormone receptor (FSHR) | X | X | | |
GALR1 | Galanin receptor 1 (GALR1) | X | X | | X |
GALR2 | Galanin receptor 2 (GALR2) | X | | X | |
GCGR | Glucagon receptor (glucagon) | X | X | | X |
GHSR | Ghrelin receptor (ghrelin) | X | | X | |
GIPR | Gastric inhibitory polypeptide receptor (GIP) | X | X | | |
GLP1R | Glucagon-like peptide receptor 1 (GLP-1) | X | X | | X |
GLP2R | Glucagon-like peptide receptor 2 (GLP-2) | X | X | | X |
GPBAR1 | G protein-coupled bile acid receptor 1 (GPBA) | X | X | | |
GPR1 | G-protein coupled receptor 1 (GPR1) | X | | | X |
GPR103 | pyroglutamylated RFamide peptide receptor (QRFPR) | X | | X | |
GPR109A | Hydroxycarboxylic acid receptor 2 (HCA2) | X | X | | |
GPR109B | Hydroxycarboxylic acid receptor 3 (HCA3) | X | X | | |
GPR120 | G-protein coupled receptor 120, long isoform (FFA4) | X | | | X |
GPR35 | G-protein coupled receptor 35 (GPR35) | X | X | | X |
GPR92 | Lysophosphatidic acid receptor 5 (GPR92) | X | | X | |
GRPR | Gastrin releasing peptide receptor (BB2) | X | | X | X |
HCRTR1 | Orexin receptor 1 (OX1) | X | | X | X |
HCRTR2 | Orexin receptor 2 (OX2) | X | | X | X |
HRH1 | Histamine receptor H1 (H1) | X | | X | |
HRH2 | Histamine receptor H2 (H2) | X | X | X | |
HRH3 | Histamine receptor H3 (H3) | X | X | | |
HTR1A | 5-hydroxytryptamine receptor 1A (5HT1A) | X | X | | |
HTR1B | 5-hydroxytryptamine receptor 1B (5HT1B) | X | X | | |
HTR1F | 5-hydroxytryptamine receptor 1F (5HT1F) | X | X | | |
HTR2A | 5-hydroxytryptamine receptor 2A (5HT2A) | X | | X | |
HTR2C | 5-hydroxytryptamine receptor 2C (5HT2C) | X | | X | X |
HTR5A | 5-hydroxytryptamine receptor 5A (5HT5A) | X | X | | |
LHCGR | Choriogonadotropin receptor (LH) | X | X | | |
LTB4R | Leukotriene B4 receptor (BLT1) | X | X | X | X |
MC1R | Melanocortin receptor 1 (MC1) | X | X | | |
MC3R | Melanocortin receptor 3 (MC3) | X | X | | X |
MC4R | Melanocortin receptor 4 (MC4) | X | X | | |
MC5R | Melanocortin receptor 5 (MC5) | X | X | | |
MCHR1 | Melanin concentrating hormone receptor 1 (MCH1) | X | X | | X |
MCHR2 | Melanin-concentrating hormone receptor 2 (MCH2) | X | | X | |
MLNR | Motilin receptor (motilin) | X | | X | X |
MRGPRX1 | MAS-related GPR, member X1 (MRGPRX1) | X | | X | |
MRGPRX2 | MAS-related GPR, member X2 (MRGX2) | X | | X | |
MTNR1A | Melatonin receptor 1A (MT1) | X | X | | X |
MTNR1B | Melatonin receptor 1B (MT2) | X | X | | X |
NMBR | Neuromedin B Receptor (BB1) | X | | X | X |
NMU1R | Neuromedin U receptor 1 (NMU1) | X | | X | X |
NPBWR1 | Neuropeptides B/W receptor 1 (NPBW1) | X | X | | |
NPBWR2 | Neuropeptides B/W receptor 2 (NPBW2) | X | X | | |
NPFFR1 | Neuropeptide FF receptor 1 (NPFF1) | X | X | | |
NPY2R | Neuropeptide Y receptor Y2 (Y2) | X | X | X | X |
NTSR1 | Neurotensin receptor 1 (NTS1) | X | | X | X |
OPRD1 | Opioid receptor delta (δ) | X | X | | X |
OPRK1 | Opioid receptor kappa (κ) | X | X | | X |
OPRL1 | Opioid receptor-like receptor (NOP) | X | X | | X |
OPRM1 | Opioid receptor mu (μ) | X | X | | X |
OXER1 | Oxoeicosanoid (OXE) receptor 1 (OXE) | X | X | | X |
OXTR | Oxytocin Receptor (OT) | X | | X | X |
P2RY1 | Purinergic receptor P2Y, G-protein coupled, 1 (P2RY1) | X | | X | X |
P2RY11 | Purinergic receptor P2Y, G-protein coupled, 11 (P2Y11) | X | | | |
P2RY2 | Purinergic receptor P2Y, G-protein coupled, 2 (P2Y2) | X | | X | X |
P2RY4 | Pyrimidinergic receptor P2Y, G-protein coupled, 4 (P2Y4) | X | | | X |
PPYR1 | Pancreatic polypeptide receptor 1 (Y4) | X | X | | |
PRLHR | Prolactin releasing hormone receptor (PRRP) | X | | X | X |
PROKR1 | Prokineticin receptor 1 (PKR1) | X | X | X | X |
PROKR2 | Prokineticin receptor 2 (PKR2) | X | | | X |
PTAFR | Platelet activating receptor (PAF) | X | | X | X |
PTGER3 | Prostaglandin E receptor 3 (subtype EP3) (EP3) | X | X | X | |
PTGER4 | Prostaglandin E receptor 4 (subtype EP4) (EP4) | X | | | X |
PTGFR | Prostaglandin F receptor (FP) (FP) | X | | X | X |
PTGIR | Prostaglandin I2 (prostacyclin) receptor (IP) (IP1) | X | X | | X |
PTHR1 | Parathyroid hormone receptor 1 (PTH1) | X | X | X | X |
PTHR2 | Parathyroid hormone receptor 2 (PTH2) | X | X | X | X |
RXFP3 | Relaxin family peptide receptor 3 (RXFP3) | X | X | | X |
RXFP4 | Relaxin family peptide receptor 4 (RXFP4) | X | X | | |
SCTR | Secretin receptor (secretin) | X | X | | X |
SSTR2 | Somatostatin receptor 2 (SST2) | X | X | | X |
SSTR3 | Somatostatin receptor 3 (SST3) | X | X | | |
SSTR4 | Somatostatin receptor 4 (SST4) | X | X | | |
SSTR5 | Somatostatin receptor 5 (SST5) | X | X | | |
TACR1 | Tachykinin receptor 1 (NK1) | X | | X | X |
TACR2 | Tachykinin receptor 2 (NK2) | X | | X | X |
TACR3 | Tachykinin receptor 3 (NK3) | X | X | X | X |
TBXA2R | Thromboxane A2 receptor (TP) | X | | X | X |
TRHR | Thyrotropin-releasing hormone receptor (TRH1) | X | | X | X |
TSHR(L) | Thyroid Stimulating Hormone Receptor (TSH) | X | X | | |
UTR2 | Urotensin II receptor (UT) | X | | X | X |
VIPR1 | Vasoactive intestinal peptide receptor 1 (VPAC1) | X | X | X | X |
VIPR2 | Vasoactive intestinal peptide receptor 2 (VPAC2) | X | X | X | X |