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BioMAP Recommended Benchmarks

Of the over 4,000 compounds that have been profiled using the BioMAP platform, the following compounds have been curated to provide the best starting point when identifying benchmarks for your BioMAP project. Included benchmarks were selected for their complete dosing and lack of overt cytoxicity..
 
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Agent Name :
Description :
Synonym :
Agent Name ▲CAS NumberSynonymMechanismDiversityPLUSFibrosisCRCNSCLCT Cell Panel
(+/-)-Nicotine22083-74-5NicotineNicotinic Acetylcholine Receptor Agonistx    
(5Z)-7-Oxozeaenol66018-38-0 TAK1 MAPKKK Inhibitorxx   
(D,L)-Mevalonic Acid Lactone674-26-0DL-Mevalonic Acid Lactone; MevalonolactoneHMG-CoA Reductase Inhibitorx    
(R,S)-Tocopherol10191-41-0Vitamin EAntioxidantx    
(S)-FTY720 Phosphate402616-26-6 S1P Receptor Agonistx    
(S)-Reticuline ReticulineAlkaloidx    
(S)-Reticuline 3-O-sulfate  CNS Depressantx    
(S)-Reticuline 7-O-sulfate  CNS Depressantx    
15(R)-Prostaglandin D259894-05-2PGD2DP Agonistx    
17α-Ethynylestradiol57-63-617alpha-EthynylestradiolER Agonistx    
17β-Estradiol50-28-2EstradiolER Agonistx    
1-Methyl-L-Tryptophan21339-55-9 IDO Inhibitorx    
22(R)-Hydroxycholesterol17954-98-2 LXRα Agonistxx   
24(S)-Hydroxycholesterol474-73-7CerebrosterolLXRα Agonistx    
25-Hydroxyvitamin D319356-17-325(OH)D; Calcidiol; CalcifediolVitamin D Receptor (VDR) Agonistx    
2-Chloroethyl Ethyl Sulfide693-07-2Sulfur MustardVesicantx    
2-Cl-IB-MECA163042-96-4C-Ibza-MU; Cl-IB-MECAAdenosine A3 Receptor Agonistx    
2-Iodomelatonin  Melatonin Receptor Agonistx    
2-Methoxyestradiol362-07-22-methoxy-17beta-estradiolMicrotubule Disruptorx    
4-Aminobenzoic Acid150-13-0PABA; p-Aminobenzoic AcidVitamin B Complex Memberx    
5-Aminolevulinic Acid Hydrochloride5451-09-2 Photosensitizer Precursorx    
5a-POPC  Cholesterol Efflux Promoterx    
5-ASA89-57-6Apriso; Asacol; Canasa; Delzicol; Mesalazine; Mezavant; Pentasa; Rowasa; Salofalk15-Lipoxygenase Inhibitor; COX1/2 Inhibitor; IKK1/2 Inhibitorx    
5a-SM 5A-sphingomyelinCholesterol Efflux Promoterx    
666-151433286-70-4 CREB Inhibitorx    
6-Mercaptopurine6112-76-1 Purine Nucleotide Synthesis Inhibitorx    
6-Thioguanine154-42-72-Amino-6-mercaptopurine; 6-Mercaptoguanine; Thioguanine; TioguanineAntineoplastic Agentx    
8-Azaguanine134-58-7Azaguanine; Guanazol; GuanazoloPurine Nucleotide Synthesis Inhibitor; Xanthine Oxidase Inhibitorx    
8-Br-cAMP23583-48-48-Bromoadenosine; BCAMPPKA Activatorx    
8-CPT-cAMP93882-12-3Rp-Cpt-campsPKA Activator; PKG Activatorx    
8-Hydroxy-5-nitroquinoline4008-48-4; 112-13-0; 53038-41-8NitroxolineAntimicrobial Agent; Anticancer Agentx    
8-Hydroxyquinoline148-24-3; 100-48-1; 1127-45-3Oxine; OxyquinolineAntimicrobial Agentx    
8-Prenylnaringenin (S)-8-dimethylallylnaringenin; 8-PN; Flavaprenin; HopeinPhytoestrogen; ER Agonistx    
9-cis-Retinoic Acid5300-03-8 RAR/RXR Agonistx    
A2318752665-69-7Antibiotic A23187; Calcimycin; Ionophore A23187Calcium Ionophorex    
A9395721032229-3-6SCD1 InhibitorStearoyl-CoA Desaturase 1 Inhibitorx  x 
Abacavir Sulfate188062-50-2Abacavir; Epzicom; ZiagenNucleoside Analog Reverse-transcriptase Inhibitor (NRTI)x    
Abatacept OrenciaT Cell Costimulation Modulatorx    
Abemaciclib1231930-82-7LY2835219; VerzenioCDK Inhibitorx    
Abiraterone154229-19-3CB-7598CYP17A1 Inhibitorx    
Abiraterone Acetate154229-18-2CB-7630; CB7630; ZytigaCytochrome P450 17A1 Inhibitorx    
Abitrexate59-05-2MethotrexateTetrahydrofolate Dehydrogenase Inhbitorx    
Acarbose56180-94-0Glucobay; PrecoseMaltase-glucoamylase Inhibitor; Pancreatic α-amylase Inhibitorx    
Acebutolol Hydrochloride34381-68-5Sectralβ1 Adrenergic Receptor Inhibitorx    
Acemetacin53164-05-9Acemetacinum; Acemix; Emflex; RantudilNSAIDx    
Acetaminophen103-90-24-Acetamidophenol; APAP; ParacetamolCOX-2 Inhibitorx    
Acetic Acid64-19-7Glacial Acetic AcidSolventx    
Acetonitrile75-05-8Cyanomethane; Ethanenitrile; Methyl cyanideOrganic Solventx    
Acitretin55079-83-9Ro 10-1670; Ro 10-1670/000; all-trans-AcitretinRetinoidx    
Acriflavin8048-52-0Flavine; PanflavinAntimicrobial Agentx    
Actemra375823-41-9Atlizumab; MRA; RoActemra; TocilizumabIL-6 Receptor Inhibitorx    
Actinomycin D50-76-0Cosmegen; DactinomycinRNA Polymerase Inhibitor; DNA Inhibitorx    
Actinonin13434-13-4Actinonine; Octanohydroxamic acidPeptide Deformylase Inhibitorx    
Adalimumab331731-18-1HumiraTNFα Inhibitorx    
Adapalene106685-40-9Adaferin; Adapaleno; Adapalenum; DifferinRAR/RXR Agonist; Vitamin A Derivative; Retinoic Acid Analoguex    
Adefovir Dipivoxil142340-99-6GS-0393; Hepsera; PMEA; PreveonReverse Transcriptase Inhbitorx    
Adenine73-24-56-AminopurineNucleobase; Purine Derivativex    
AEB071425637-18-9AEB-071; Sotrastaurin; UNII-7I279E1NZ8PKCΘ Inhibitorx    
AEG348263735-71-7 Hsp90 Inhibitorx    
Afamelanotide75921-69-6Scenesse; melanotan-1Melanocortin Receptor Agonistx    
Afatinib439081-18-2BIBW2992EGFR/HER2 Inhibitorx    
AG1478153436-53-4AG-1478; Tyrphostin AG 1478EGFR Inhibitorx    
AIM-100  Ack1 Inhibitor x   
Albendazole54965-21-8AlbenzaMicrotubule Inhibitor; Anthelmintic Agentx    
Aldosterone52-39-1;152-04-5;10328-70-8Aldocorten; Aldocortin; Aldosteronum; Electrocortin; ElektrocortinMineralocorticoid Receptor (MR) Agonist x    
Alectinib1256580-46-7AlecensaALK Inhibitorx xx 
Alemtuzumab Campath; LemtradaAnti-CD52 Antibodyx    
Alendronate121268-17-5FosamaxFarnesyl Diphosphate Synthase Inhibitorx    
Alfacalcidol41294-56-81-Hydroxycholecalciferol; Bondiol; Etalpha; Oxydevit; TevaboneVitamin D Analoguex    
Alprostadil745-65-3Alprostadilum; Befar; Caverject; Edex; Prostaglandin E1; Prostin vrEP Agonist; Prostanoid Receptor Agonist (EP1, EP2)x    
Altrenogest850-52-2Allyltrenbolone; Allyltrienolone; Matrix, RU-2267; RegulateProgesterone Receptor (PR) Agonist; Androgen Receptor Agonistx    
Altretamine645-05-6HexalenAlkylating Antineoplastic Agentx    
Alverine Citrate5560-59-8Oxydevit; Phenpropamine CitrateSmooth Muscle Relaxant; 5-HT1A Inhibitorx    
AM-9661228690-19-4AM966; UNII-CEO54NH393LPA1 Receptor Inhibitorxx   
AMD3465185991-07-5AMD 3465 HexahydrobromideCXCR4 Inhibitorx x  
Amfenac Sodium61618-27-72-amino-3-benzoylbenzeneacetic AcidNSAIDx    
AMG2081002304-34-8AMG 208; UNII-Y2SR66P7VMc-Met Inhibitorx    
AMG548864249-60-5AMG 548p38 MAPK Inhibitorx    
Amifampridine  Potassium Channel Blockerx    
Aminoglutethimide125-84-8Cytadren; NSC 33091Aromatase Inhibitorx    
Aminophylline317-34-0 PDE Inhibitor; Adenosine Receptor Inhibitorx    
Amitriptyline Hydrochloride549-18-8ElavilSNRI; TrkA Agonist; TrkB Agonist; SMase Inhibitorx    
Amlexanox68302-57-8Amlenanox; Amoxanox; Aphthasol; SolfaAnti-inflammatory Agent; Antiallergic Agent; Immunomodulating Agentx    
Amodiaquin86-42-0Camochin; Camoquin; Camoquine; FlavoquineAntimicrobial Agentx    
Amphotericin B1397-89-3Abelcet; Ambisome; AmphotecAntimicrobial Agentx    
Ampiroxicam99464-64-9 NSAIDx    
Amprenavir161814-49-9Agenerase; Prozei; Vertex VX478Protease Inhibitorx    
Anacetrapib875446-37-0MK-0859CETP Inhibitorx    
Anakinra143090-92-0ICIL-1RA; IL-1RN; IL-1ra; IL1 inhibitor; IRAP; KineretIL-1 Receptor Inhibitorx    
Antazoline Hydrochloride2508-72-7Vasocon-aH1 Receptor Inhibitorx    
Antimycin A1397-94-0Antimycin A1; Antimycin A1b; Antipiricullin; Fintrol; VirosinCytochrome c Reductase Inhibitor; Mitochondrial Inhibitorx    
Apelin-13  Apelin Receptor (APJ) Ligandx    
Apoptolidin194874-06-1Apoptosis Activator IV; Nocardiopsis sp.F(0)F(1) ATPase Inhibitor; Mitochondrial Inhibitorx    
Apremilast608141-41-9;Apremilastum; CC 10004; CC-10004; OtezlaPDE4 Inhibitorx    
Artemisinin63968-64-9NSC 369397Antimicrobial Agentx    
Articaine Hydrochloride23964-57-0CarticaineAnesthetic Agentx    
AS1892802928320-12-1AS 1892802; AS-1892802ROCK1, ROCK2 Inhibitorx    
AS2444697 AKOS027470180IRAK4 Inhibitorx    
AS601245345987-15-7AS 601245JNK Inhibitorx    
AS605240648450-29-7PI 3-Kgamma Inhibitor; PI3-Kγ InhibitorPI3K Inhibitorx    
Asenapine85650-56-2 Antipsychotic Agentx    
Aspirin50-78-2Acetylsalicylate; Acetylsalicylic acidCOX Inhibitorx    
Astemizole68844-77-9Astemison; Astemizol; AstemizolumAntihistamine Agentx    
Atazanavir Sulfate229975-97-7BMS 232632; CGP 73547; ReyatazHIV Protease Inhibitorx    
Atomoxetine Hydrochloride82248-59-7StratteraNorepinephrine Reuptake Inhibitorx    
Atorvastatin134523-00-5Lipitor; LipovastatinklonalHMG-CoA Reductase Inhibitorx    
Atovaquone95233-18-4AtavaquoneCytochrome b Inhibitorx    
ATP Adenosine triphosphateCoenzymex    
Atracurium Besylate64228-81-564228-81-5; Atracurium Besilate; Atracurium Besylate; TracriumNeuromuscular Blocking Agent x    
Auranofin34031-32-8NSC 321521; Ridauragold thiol; SKF 39162Thioredoxin Reductase Inhibitorx    
AVL-292 CC-292; SpebrutinibBTK Inhibitor x xx 
Axitinib319460-85-0InlytaVEGFR2 Inhibitorxxxx 
AZ876898800-26-5LPM029_300383_00LXR Agonistx    
Azaperone1649-18-9R-1929; Stresnil; SuicalmDopamine Receptor Inhibitorx    
Azatadine Dimaleate3978-86-7Azatadine Maleate; Bonamid; IdulianHistamine and Cholinergic Inhibitorx    
Azathioprine446-86-6Azasan; BW-57-322; ImuranPurine Metabolism Anatgonistxx   
AZD12081204144-28-4AZD 1208PIM Kinase Inhibitorx    
AZD45471035270-39-3AZD 4547; AZD-4547FGFR Inhibitorx    
AZD80551009298-09-2AZD 8055; AZD-8055mTOR Inhibitorx    
Azithromycin83905-01-5Azasite; Azenil; Azifast; Azigram; Azimakrol; Hemomycin; ZithromaxAntibiotic Agentxx   
Bacitracin Zinc1405-89-6 Antibiotic Agentx    
Bafilomycin A188899-55-2NSC 381866V-ATPase Inhibitorx    
Baricitinib1187594-09-7INCB 028050; LY3009104JAK1/2 Inhibitorx    
BAY-8761799753-84-6 GLUT1 Inhibitorx    
BDH35145960b  BET Inhibitorx    
BDV0005266b  Bromodomain Inhibitorx    
Beclomethasone Dipropionate4419-39-0QvarGR Agonistx    
Bedaquiline EX00040046; SirturoMycobacterial ATP Synthase Inhibitorx    
Belatacept belataceptT Cell Costimulation Modulatorx    
Bemcentinib1037624-75-1BGB324; R428AXL Inhibitorxxxx 
Benlysta belimumabBAFF Inhibitorx    
Benzethonium Chloride121-54-0Antiseptol; BZT; Diapp; Disilyn; Hyamine; Phemithyn; Phermerol; Polymine D; Quatrachlor; SalanineAntimicrobial Agent; AChE Inhibitorx    
Benzocaine94-09-7Americaine; Ethyl AminobenzoateAnestheticx    
Benztropine Mesylate132-17-2CogentinMuscarinic Acetylcholine Receptor (mAChR) Inhibitor x    
Benzydamine Hydrochloride132-69-4AF-864; TantumNSAIDx    
Beraprost MDL-201229; ProcylinProstacyclin Analoguex    
Berberine Berberin; UmbellatineDipeptidyl Peptidase IV Inhibitor; PTP1B Inhibitorx    
Bergapten484-20-85-Methoxypsoralen; Bergaptene; Heraclin; MajudiPsoralenx    
beta-Mercaptoethanol  Inorganic Compound  xx 
Betamethasone378-44-9CelestoneGlucocorticoid Receptor (GR) Agonistx    
Betamethasone Dipropionate5593-20-4DiproleneGlucocorticoid Receptor (GR) Agonistx    
Betamethasone Valerate2152-44-5BetnovateGlucocorticoid Receptor (GR) Agonistx    
Betamipron3440-28-6Benzoyl-beta-alanineCarbapenem Antibiotic Agentx    
Betapar1247-42-3Betanisona; Meprednisone; MethylprednisoneGlucocorticoid Receptor (GR) Agonistx    
Bevacizumab216974-75-3Avastin; anti-VEGFVEGFA Inhibitorx x  
BI-10n  ITK Inhibitorx    
BI2536755038-02-9 BET Inhibitor; PLK1 Inhibitorx x  
BIBX1382196612-93-8BIBX 1382; FalnidamolEGFR Inhibitorx    
Bilirubin635-65-4Bilirubin IX- α; Hematoidin; HemetoidinHeme Metabolitex    
Bindarit  CCL2/7/8 Inhibitor x   
Biperiden Hydrochloride1235-82-1Akineton; AkinophylAcetylcholine Inhibitorx    
Bisacodyl603-50-9Bicol; Brocalax; Dulcolax; DurolaxLaxativex    
Bismuth Subcitrate Potassium880149-29-1Bismuth Subcitrate; Bismuth Subcitrate Potassium; De-Noltab; Gastrodenol; Tripotassium DicitratobismuthateAntibiotic Agentx    
Bleomycin Sulfate9041-93-4Blenoxane; BleomycinAntineoplastic Agentx    
BMP7 Osteogenic Protein-1 (OP-1)Activin Receptor Agonist (Activin RIA, RIIA, RIIB; BMPR-IA, BMPR-IB, BMPR-II)x    
BMS-7776071025720-94-8BMS777607c-Met Inhibitor; Axl Inhibitor; RON Inhibitor; Tyro3 Inhibitorxxx  
BMY 45778152575-66-1 BMY 45778 is a non-prostanoid prostacyclin IP receptor partial agonist.x    
Bortezomib179324-69-7VelcadeProteasome Inhibitorxx   
Bosentan147536-97-8Bosentan Hydrate; Bosentanum; TracleerET-A Inhibitor; ET-B Inhibitorx    
Bosutinib380843-75-4Bosulif; SKI-606BCR-ABL Inhibitor; Src Inhibitorxx x 
Brefeldin A20350-15-6Ascotoxin; Cyanein; Decumbin; SynergisidinARF1 Inhibitorx    
Brequinar Bay_BioMAP_005_B2; bipenquinateDHODH Inhibitorx    
Brigatinib  ALK Inhibitor; EGFR Inhibitor  xx 
Bromfenac Sodium91714-93-1XibromNSAID; COX Inhibitorx    
Bromosporine1619994-69-2 Pan Bromo Domain Inhibitorx    
Brompheniramine Maleate980-71-2BPN; Bromfed; Bromfenex; Dimetane; Dimetapp; LodraneAntihistamine Agentx    
Broxyquinoline521-74-4DibromohydroxyquinolineAntimicrobial Agentx    
BSK_4925 Lymphocyte Specific KinaseLck Inhibitorx    
BSK_anti-CTLA4  CTLA4 Inhibitorx    
BSK_RORg1333114-08-1 RORγ Inhibitorx    
Bucladesine362-74-3Actosin; Dibutyryl cAMP; Dibutyryl cyclic AMPPDE4 Inhibitorx    
Budesonide51333-22-3Budeson; Entocort; Preferid; Pulmicort; SpirocortGlucocorticoid Receptor (GR) Agonistxx   
Bupropion Hydrochloride34841-39-9Amfebutamone; Budeprion; Bupropion; Elontril; Prexaton; Quomem; Voxra; WellbutrinNDRIx    
Busulfan55-98-1Busulfex; MyleranAlkylating Antineoplastic Agentx    
BW 245C75693-75-3BW-245C; BW245CDP Agonistx    
BW 246C65705-83-18-epi BW 245CDP Agonistx    
Cabozantinib849217-68-1BMS-907351; Cometriq; XL184VEGFR2 Inhibitorxxxx 
Calcipotriene112965-21-6Daivonex; Dovonex; SoriluxSynthetic Calcitriol Derivativex    
Calcitriol32222-06-3Calcijex; Calcitriolum; Decostriol; Rocaltrol; Silkis; VecticalVitamin D Receptor (VDR) Agonistx    
Calcium Chloride10043-52-4CaCl2; Calcium Chloride AnhydrousSaltx    
Cantharidin56-25-7CantharoneProtein Phosphatase 2A (PP2A) Inhibitorx    
CAPE104594-70-9Caffeic Acid Phenethyl Ester; Phenethyl caffeate15-Lipoxygenase Inhibitorx    
Carbimazole22232-54-8AthyromazoleAntithyroid Agentx    
Carboplatin Paraplat; Paraplatin; Paraplatin-AQDNA Repair Inhibitor  x  
Carfilzomib868540-17-4Kyprolis; PR-171Proteasome Inhibitorx    
Carmofur61422-45-51-hexylcarbamoyl-5-fluorouracil; HCFUPyrimidine Analogue; Antineoplastic Agentx    
Carprofen53716-49-7Imadyl; Imafen; Novox; Quellin; Rimadyl; Rovera; VetprofenNSAIDx    
Carvedilol72956-09-3Beta Blocker; Carvedilolum; Coreg; Coreg CR; SKF 105517Adrenergic Receptor Inhibitorx    
Caspofungin Acetate179463-17-3Cancidas; L-743,872; MK 0991Antimicrobial Agentx    
CAY10410596104-94-89,10-dihydro-15-deoxy-Δ12,14-PGJ2PPARγ Agonistx    
CCG-1423285986-88-1Myocardin-related Transcription Factor-AMRTF-A Inhibitor; Rho Kinase/ROCK Signaling Inhibitorxx   
CDDO Methyl Ester218600-53-4Bardoxolone Methyl; NSC 713200; RTA 402; TP-155Nrf2 Activator; Triterpenesx    
Ceftazidime Pentahydrate78439-06-2Fortaz; TazicefAntibiotic Agentx    
Celebrex169590-42-5; 184007-95-2Celecoxib; CelecoxibumCOX-2 Inhibitorx    
Cepharanthine481-49-2 Anti-inflammatory Agent; Antineoplastic Agentx    
Cerivastatin143201-11-0Baycol; Cerivastatin Acid; LipobayHMG-CoA Reductase Inhibitorx    
Cetirizine Dihydrochloride83881-51-0Alerlisin; Reactine; ZyrtecAntihistamine Agent; GPCR Ligandx    
Cetrimonium Bromide57-09-0CTAB; Centimide; Cetyltrimethylammonium Bromide; Hexadecyltrimethylammonium BromideAntimicrobial Agentx    
Cetuximab Anti-EGFR; Erbitux; IMC-C225EGFR Inhibitorx xx 
Cetylpyridinium Chloride123-03-5 Antiseptic Agentx    
CFM 1571 Hydrochloride  sGC Activator x   
CGP 5260887958-67-6 RORα Ligandx    
CH223191301326-22-7 AhR Inhibitorx    
CHIR-99021 Hydrochloride252917-06-9CT99021GSK-3α/β Inhibitorx x  
Chlorambucil305-03-3Ambochlorin; CHLORAMBUCIL; Chloraminophen; LeukeranAlkylating Agentx    
Chlorocresol59-50-74-chloro-3-cresol; 4-chloro-3-methylphenolAntiseptic Agentx    
Chloroquine Phosphate50-63-5Aralen; Resoquine; Reumachlor; SanoquinAntimicrobial Agentx    
Chlorothiazide58-94-6DiurilAntihypertensive Agent; Diuretic Agentx    
Chlorprothixene113-59-7Chlorprothixenum; Clorprotixeno; Taractan; TruxalAntipsychotic Agentx    
Chlorquinaldol72-80-0SterosanAntimicrobial Agentx    
Cholecalciferol67-97-0Calciol; Colecalciferol; Oleovitamin D3; Vitamin D3Vitamin D Receptor (VDR) Agonistx    
Cilnidipine132203-70-4Atelec; Cinalong; SiscardCalcium Channel Blockerx    
Cilostazol73963-72-1Cilostazole; Cilostazolum; Pletaal; PletalPDE Inhibitorx    
Cinacalcet Hydrochloride364782-34-3AMG-073 HClCalcimimetic Agent; Extracellular Calcium-sensing Receptor Agonistx    
Cinchophen132-60-5Atophan; Phenaquin; QuinophanAnalgesic Drug x    
Ciprofloxacin Hydrochloride85721-33-1BAY-o 9867; Cetraxal; Ciloxan; Cipro; Ciprol; NSC 620634Antimicrobial Agentx    
Cisplatin15663-27-1CACP; Cisplatina; Cisplatinum; DDP; Neoplatin; Platinol-AQDNA Alkylating Agentx x  
Cladribine4291-63-82-CdA; 2-Chlorodeoxyadenosine; LeustatinAntineoplastic Agentx    
Clemastine17-7-4Clemastina; ClemastinumAntihistamine Agentx    
Clexane Ardeparin; Enoxaparin; Enoxaparin Sodium; Heparin; Nadroparin; TinzaparinAnticoagulant Agentx    
CLI-095 Meclastin; Resatorvid; TAK-242TLR4 Inhibitorx    
Climbazole38083-17-9Baypival; BaysanAntimicrobial Agentx    
Clofarabine123318-82-1CAFdA; Clofarex; Clolar; EvoltraNucleic Acid Synthesis Inhibitorx    
Clofazimine2030-63-9LampreneAntimycobacterial Agentx    
Cloprostenol (+)-16-m-chlorophenoxy Tetranor Prostaglandin F2αProstaglandin F (FP) Receptor Agonist; PGF2α Analogx    
Closantel Sodium61438-64-0 Antimicrobial Agentx    
Clozapine5786-21-0Clozapinum; Clozaril; Fazaclo; VersaclozAntipsychotic Agentx    
Cobalt(II) Chloride Hexahydrate7791-13-1Cobaltous Chloride HexahydrateInorganic Compoundx x  
Cobicistat1004316-88-4GS-9350; GS-9350, Tybost; TybostCYP3A Inhibitorx    
Coffee Extract  Coffee Extractx    
Colchicine114977-28-5Colchicin; Colchicina; Colchicinum; Colcrys; MitigareMicrotubule Disruptorx xx 
Concanamycin A80890-47-7Antibiotic X 4357B; NSC 674620; X 4357BV-ATPase Inhibitorx    
Concanavalin A Type VI11028-71-0 Purified Lectinx    
Copper(II) Sulfate7758-98-7 Glucose-6-phosphate Dehydrogenase (G6PD) Inhibitor; Paraoxonase Inhibitorx    
Cortistatin-14186901-48-4Cortistatin14Steroidal Alkaloidsx    
CP 55,940  Cannabinoid (CB) Receptor Agonistx    
CPG 52364  TLR7/TLR8/TLR9 Inhibitorx    
Crisaborole EucrisaPDE4 Inhibitorx    
Crizotinib877399-52-5PF 2341066; PF-02341066; XalkoriAnticancer Agent; ALK Tyrosine Kinase Receptor Inhibitor; HGFR Inhibitorx xx 
Curcumin  Natural Phenol x   
Cyanocobalamin68-19-9Cyanocob(III)alamin; Nascobal; Vitamin B12Vitamin B12 Analoguex    
Cycloheximide66-81-9Actidione; Cicloheximide; Kaken; Naramycin AProtein Synthesis Inhibitorx    
Cyclopentyl Adenosine  Adenosine A1 Receptor Agonistx    
Cyclosporin A59865-13-3CyA; Cyclosporine; Gengraf; Neoral; Restasis; SandimmuneCalcineurin Inhibitor; Cyclophilin A Modulatorx xxx
Cystamine Dihydrochloride111625-30-0; 56-17-7EthanamineCystine Depleting Agentx    
Cysteamine Hydrochloride156-57-0; 116962-86-8; 16904-32-8 Cystine Depleting Agentx    
Cytarabine147-94-4Ara-C; Arabinosylcytosine; Cytosar; Cytosine ArabinosideDNA Synthesis Inhibitorx    
Dabrafenib GSK2118436; TafinlarBRAF Inhibitorx xx 
Dacomitinib VizimproEGFR Inhibitorx  x 
Dactolisib915019-65-7BEZ235; NVP-BEZ235PI3K Inhibitor; mTOR Inhibitorx xx 
Dalcetrapib211513-37-0JTT-705Cholesterylester Transfer Protein (CETP) Inhibitorx    
Danofloxacin Mesylate119478-55-6Advoci; CP-76136-27; NofloxacinAntimicrobial Agentx    
Darifenacin Hydrogen Bromide133099-07-7Enablex; UK 88525-04Muscarinic Acetylcholine Receptor Inhibitorx    
Darunavir Ethanolate635728-49-3Prezista; TMC114Protease Inhibitorx    
Dasatinib302962-49-8BMS-354825; SprycelMultikinase Inhibitor (Src tyr Kinase, BCR/Abl)xxxx 
Daunorubicin Hydrochloride23541-50-6Acetyladriamycin; Daunomycin; Daunorubicina; Daunorubicine ; Daunorubicinum; Leukaemomycin C; RubidomycinDNA Topoisomerase Inhibitorx x  
Decitabine2353-33-5Azadc; Dacogen; DezocitidineNucleic Acid Synthesis Inhibitorx    
Deferasirox201530-41-8Exjade; ICL670AIron Chelating Agentx    
Deferoxamine Mesylate70-51-9DFOA; DFOM; Deferoxamina; Deferoxamine; Deferoxaminum; DeferrioxamineIron Chelating Agentx    
Denosumab Prolia; XgevaRANKL Inhibitorx x  
Deoxyarbutin53936-56-4 Tyrosinase Inhibitorx    
Dequalinium Chloride522-51-0Danical; Decabis; DequafunganAntimicrobial Agent; PKC Inhibitorx    
Desloratadine100643-71-8Aerius; Clarinex; DescarboethoxyloratadineAntihistamine Agentx    
Desonide638-94-8Desowen; TridesilonGlucocorticoid Receptor (GR) Agonistx    
Dexamethasone50-02-2Baycadron; Decadron; Dexametasona; Maxidex; OzurdexGlucocorticoid Receptor (GR) Agonistx    
Dexlansoprazole138530-94-6Dexilant; KapidexProton Pump Inhibitorx    
Dexmedetomidine113775-47-6Dex; Precedexα2 Adrenergic Receptor Agonistx    
Dibucaine85-79-0Cinchocaine; Dermacaine; Nupercainal; NupercaineAnestheticx    
Diclofenac Diethylamine78213-16-8AK163134; UNII-6TGQ35Z71KNSAIDx    
Diclofenac Potassium15307-81-0Cambia; Cataflam; UNII-L4D5UA6CB4; ZipsorNSAIDx    
Dienogest65928-58-7Progestin; VisanneSemisynthetic Steroidal Progestogenx    
Difluprednate23674-86-4DurezolCorticosteroidx    
Digoxigenin1672-46-4Digitoxigenin; UzarigeninHaptenx    
Dihydrotestosterone521-18-6Anaboleen; Androlone; Androstanolone; Stanaprol; StanoloneAR Agonistx    
Dimethyl Fumarate624-49-7BG-12; DMF; TecifideraNFκB Inhibitor; Nrf2 Activatorx    
Diminazene Aceturate908-54-3Diminazeno; DiminazenumACE Activatorx    
Diphenylpyraline Hydrochloride132-18-3Allerzine; Diaphen; HistalertAntihistamine Agent; GPCR Ligandx    
Diprophylline479-18-5DilorPDE Inhibitor; Adenosine Receptor Antagonistx    
Dipyridamole58-32-2Cardoxin; Cleridium 150; Curantyl; Permole; Persantin; PersantinePDE Inhibitorx x  
Disulfiram97-77-8Antabuse; Tetraethylthiuram DisulfideAldehyde Dehydrogenase Inhibitorx    
Donepezil Hydrochloride120011-70-3Aricept; DonepezilumCholinesterase Inhibitorx    
Doramapimod285983-48-4BIRB-796; BIRB796p38 MAPK Inhibitorxx   
Dorzolamide Hydrochloride120279-96-1MK-507Carbonic Anhydrase Inhibitorx    
Doxazosin Mesylate74191-85-8Carduraα1 Adrenergic Receptor Inhibitorx    
Doxorubicin Hydrochloride25316-40-9Adriamycin; Doxorubicine; Doxorubicinum; HydroxydaunorubicinDNA Topoisomerase Inhibitorx    
D-Pantethine16816-67-4Pantethine; Pantetina; Pantomin; PantosinCofactor Precursorx    
Droperidol548-73-2Dehydrobenzperidol; Dridol; Droleptan; InapsineDopamine Receptor (D2) Inhibitor; 5-HT2A Receptor Inhibitorx    
Drospirenone67392-87-41,2-dihydrospirorenone; YasminProgesterone Receptor (PR) Agonistx    
Dydrogesterone152-62-5Duphaston; IsopregnenoneProgesterone Receptor (PR) Agonistx    
Edaravone89-25-8MCI-186; RadicutAntioxidantx    
EGF62253-63-8Epidermal Growth FactorEGFR Activatorx    
EGFR/ErbB-2/ErbB-4 Inhibitor881001-19-0 EGFR Inhibitor; HER2, HER4 Inhibitorx    
Eicosapentaenoic Acid10417-94-4EPA; Icosapentaenoic AcidOmega-3 Fatty Acid; Eicosanoid Precursorx    
Ellagic Acid476-66-4 Antioxidant Agentx    
Embelin  X-linked Inhibitor of Apoptosis Protein (XIAP) Inhibitor  x  
Emricasan254750-02-2 Caspase Inhibitorx    
Enbrel185243-69-0Etanercept; TNF-R2TNFα Inhibitorx    
Entinostat209783-80-2MS-275; SNDX-275HDAC Inhibitorx    
Epacadostat INCB024360IDO Inhibitorx xx 
Epalrestat82159-09-9ONO-2235Aldose Reductase Inhibitorxx   
Epothilone B152044-54-7EPO 906; EPO906; PatupiloneMicrotubule Disruptorx    
Epothilone D189453-10-9Desoxyepothilone BMicrotubule Disruptorx xx 
Eprazinone Dihydrochloride10402-53-6746CE; Eftapan; Mucitux; NSC 317935; Resplen; RozuplenMucolytic Agentx    
Erlotinib183321-74-6CP-358,774; Erlotinib Hydrochloride; OSI-774; TarcevaEGFR Inhibitorxxxx 
Erythromycin114-07-8Abomacetin; Eritromicina; IlotycinAntibiotic Agentx    
Ethacridine Lactate6402-23-9Acrinol; RivanolDNA Intercalating Antiseptic Agentx    
Ethacrynic Acid58-54-8EdecrinDiuretic Agentx    
Ethanol64-17-5Alcohol; Ethyl Alcohol; Ethyl HydroxideGABA-A Receptor Agonist; NMDA Receptor Inhibitorx    
Ethionamide536-33-4 Antimicrobial Agentx    
Ethosuximide77-67-8Aethosuximide; Atysmal; Ethosuximidum; EtosuximidaVoltage-gated T-type Calcium Channel Blockerx    
Ethoxzolamide452-35-7EthoxyzolamideCarbonic Anhydrase Inhibitorx    
Ethyl Pyruvate617-35-6Ethyl 2-Oxopropanoate; Pyruvic Acid Ethyl EsterAnti-inflammatory Agentx    
Ethylenediamine107-15-3 Organic Compoundx    
Etodolac41340-25-4Etodolaco; Etodolacum; Etodolic acid; LodineCOX-2 Inhibitorx    
Etomidate33125-97-2AmidateAnaesthetic Agent; GABA-A Agonistx    
Etoposide33419-42-0VP-16DNA Topoisomerase (TOPO) II Inhibitorx    
Etravirine269055-15-4Intelence; TMC-125; TMC125NNRTIx    
Everolimus159351-69-6Afinitor; Certican; Evertor; RAD001; ZortressmTOR Inhibitorxxx x
Exemestane107868-30-4AromasinSteroidal Aromatase Inhibitorx    
Ezetimibe163222-33-1Ezedoc; SCH-58235; ZetiaAntilipemic Agentx    
Famprofazone22881-35-2Gewodin; GewolenNSAIDx    
Fasudil103745-39-7Fasudil Hydrochloride; HA-1077ROCK1, ROCK2 Inhibitorxx   
FCCP370-86-5Carbonyl cyanide p-trifluoromethoxyphenylhydrazoneUncoupling Agent; Ionophorex    
Febuxostat144060-53-7Adenuric; Feburic; Goturic; UloricXanthine Oxidase Inhibitorx    
Fedratinib936091-26-8Inrebic; SAR302503; TG101348JAK2 Inhibitorx x  
Fenbendazole43210-67-9PanacurAnthelmintic Agent; Microtubule Disruptorx    
Fenoprofen Calcium Dihydrate34597-40-5Fenopron; Nalgesic; ProgesicCOX Inhibitorx    
Fenspiride Hydrochloride5053-08-7NAT-333; NDR-5998APDE Inhibitorx    
Fexofenadine Hydrochloride153439-40-8AllegraH1 Receptor Inhibitorx    
FICZ172922-91-7 AhR Agonistx x  
Fidaxomicin873857-62-6Dificid; Dificlir; OPT-80; PAR-101Antibiotic Agentx    
Filgotinib GLPG0634JAK1 Inhibitorxxx  
Finasteride98319-26-7Propecia; ProscarType II, Type III 5α-reductase Inhibitorx    
Fingolimod162359-56-0FTY720; GilenyaS1P Receptor Agonistx    
Flagellin  TLR5 Agonistx    
Fleroxacin79660-72-3FLRX; Megalone ; Megalosin; QuinodisAntimicrobial Agentx    
Flubendazole31430-15-6FlutelmiumAntimicrobial Agentx    
Fludarabine21679-14-12-Fluoro-Ara-A; F-ara-A; Fludara; NSC 118218; OfortaSTAT1 Inhibitor; DNA Synthesis Inhibitorx    
Fludrocortisone127-31-1Fludrocortisona; Fludrocortisonum; FluohydrocortisoneGlucocorticoid Receptor (GR) Agonist; Mineralocorticoid Receptor (MR Agonist)x    
Flumazenil78755-81-4Anexate; Flumazepil; LanexatGABA/Benzodiazepine Receptor Inhibitorx    
Flumethasone2002-29-1Locacorten; Locorten; Orsalin; U-10974Glucocorticoid Receptor (GR) Agonistx    
Flunarizine Dihydrochloride30484-77-6FlunarizinaCalcium Channel Blocker; Antihistamine Agentx    
Fluorometholone Acetate3801-06-7Eflone; Flarex; Fluorometholone 17-acetate; Oxylone AcetateGlucocorticoid Receptor (GR) Agonistx    
Fluorouracil51-21-8 5-FU; 5-FU; 5-Fluracil; Adrucil; Fluoro Uracil; Fluoroplex; FluouracilThymidylate Synthase (TS) Inhibitor; Pyrimidine Analogx x  
Fluoxetine54910-89-3Adofen; LY-110140; Prozac; Sarafem; SymbyaxAntidepressant; SSRI Inhibitorx    
Flurbiprofen5104-49-4Ansaid; FLP; OcufenCOX Inhibitor; NSAIDx    
Fluticasone Propionate80474-14-2Fluticason; Fluticasona; Fluticasone; FluticasonumGlucocorticoid Receptor (GR) Agonist; Progesterone Receptor (PR) Agonistxx   
Fluvastatin93957-54-1Fluvastatin Sodium; LescolHMG-CoA Reductase Inhibitorx    
Fluvoxamine Maleate61718-82-9LuvoxSSRIx    
FM-381 DRX_FM-381JAK3 Inhibitorx    
fMLP59880-97-6FMLP; N-Formylmethionyl-leucyl-phenylalanineFPR Agonistx    
Forskolin66575-29-9Coleonol; Colforsin; Colforsina; ColforsineAdenylyl Cyclase Activatorx    
Fosaprepitant Dimeglumine265121-04-8Ivemend; L 758298; UNII-6L8OF9XRDCNeurokinin-1 Receptor Inhibitorx    
Fosbretabulin Disodium168555-66-6CA4DP; ZybrestatMicrotubule Disruptorx    
Fostamatinib1025687-58-4R406Syk Inhibitorx    
FSL-1  TLR2/TLR6 Agonistx    
Ftorafur17902-23-7Tefudex; Tegafur-uracil; UFT; Uftotral; UfurChemotherapeutic Agentx    
Fucoidan9072-19-9 Caspase-3 Activatorx    
Fulvestrant129453-61-8FaslodexEstrogen Receptor (ER) Inhibitorx    
Fumagillin23110-15-8FumidilAngiogenesis Inhibitor; MetAP2 Inhibitorx    
Galeterone851983-85-2TOK-001CYP17A1 Inhibitorx    
Galunisertib700874-72-2LY2157299TGFβR1 Kinase Inhibitorxxxx 
Gandotinib1229236-86-5LY2784544JAK2 Inhibitorx x  
GDC0834 1133432-49-1BTK Inhibitorx xx 
GDC0853 RG-7845BTK Inhibitorx    
GDC0879  B-Raf/C-Raf Inhibitor  x  
GDC0941957054-30-7GDC-0941; PictilisibPI3Kα/δ Inhibitorxxx  
Gefitinib184475-35-2Iressa; ZD 1839EGFR Inhibitorx x  
Geldanamycin30562-34-6GeldanomycinHsp90 Inhibitorx    
Gemcitabine Hydrochloride122111-03-9Gemzar; LY-188011; dFdC; dFdCydNucleoside Metabolic Inhibitor x xx 
Gemfibrozil25812-30-0Gemfibrozilo; Gemfibrozilum; LopidPPARα Agonistx    
Genistein446-72-0Genisteol; Genisterin; NSC-36586Phytoestrogenx    
Gestodene60282-87-315-dehydronorgestrelProgesterone Receptor (PR) Agonistx    
GF109203X133052-90-1Bisindolylmaleimide IPKC (c+n) Inhibitorx    
Gilteritinib1254053-43-4XospataTyrosine Kinase Inhibitorx    
GKT1378311218942-37-0GKT-137831NOX1/NOX4 Inhibitorxx   
Glatimer Acetate CopaxoneImmunomodulating Agentx    
Glesatinib  Tyrosine Kinase Inhibitorx    
Gliquidone33342-05-1Beglynor; Glikvidon; Gliquidonum; GlurenormKATP Channel Blockerx    
GLP-1 Proglucagon (72-108)Glucagon-like Peptide 1 (GLP-1) Receptor Agonistx    
Glyburide  Sulfonylurea; Antihyperglycemic Agentx    
GM-CSF83869-56-1CSF2; Leukine; SargramostimCytokine; Immune Modulatorx    
Go 6983133053-19-7 PKC (c+n) Inhibitorx    
Golimumab SimponiTNFα Inhibitorx    
GRP Gastrin-releasing PeptideStimulates Gastrin Release; Neuropeptidex    
GSK Compound 181221277-91-3LPM029_300303_01LXR Agonistx    
GSK27950391415925-18-6 NOX2 Inhibitorx    
GSK2801 GSK 2801; KB-146016BAZ2 Bromodomain Inhibitorx    
GSK461364A929095-18-1GSK 461364APLK1 Inhibitorx x  
GSK690693937174-76-0GSK 690693AKT Inhibitorx    
GSKJ41373423-53-0GSK J4; GTPL8979Histone Demethylase Inhibitorx x  
GW2580870483-87-7 cFMS Kinase Inhibitorx    
GW3965405911-09-3 LXRα Agonistx    
GW501516317318-70-0GW-501516PPARδ Agonistx xx 
H-1152451462-58-1H1152ROCK2 Inhibitorxx   
H-89127243-85-05-Isoquinolinesulfonamide; Protein Kinase Inhibitor H-89PKA Inhibitorx    
Halobetasol Propionate66852-54-8UlobetasolGlucocorticoid Receptor (GR) Agonistx    
hCG Human Chorionic GonadotropinLuteinizing Hormone; Choriogonadotropin Receptor Agonistx    
Hemicholinium Bromide312-45-8HemicholineCholine Transporter (ChT) Inhibitorx    
HGF Hepatocyte Growth Factorc-Met Inhibitorx    
Histamine51-45-6 Histamine Receptor Agonistx    
Histamine Phosphate51-74-1 Histamine Receptor Agonistx    
HKLM Heat Killed Listeria monocytogenesTLR2 Agonistx x  
Homatropine Bromide51-56-9 Muscarinic Acetylcholine Receptor (mAChR) Inhibitor x    
Human anti-CD73 IgG1 MEDI9447Anti-CD73 Monoclonal Antibody  x  
Human IgG1  IgG1 Control Antibody  x  
Human IgG1 Kappa  Immunoglobulinx    
Human IgG1 mAb R347 Isotype Control  IgG1 Control Antibody  x  
Human γ-Globulin  Serum Fractionx    
Hydrochlorothiazide58-93-5 Diuretic Agentx    
Hydrocortisone50-23-717-HydroxycorticosteroneGlucocorticoid Receptor (GR) Agonistx    
Hydroxychloroquine Sulfate747-36-4Ercoquin; Oxychlorochin; Oxychloroquine; Plaquenil; ToremonilAntimicrobial Agentx    
Hydroxyfasudil155558-32-0HA 1100ROCK1, ROCK2 Inhibitorx    
Hydroxyurea127-07-1Droxia; Hydrea; Hydroxycarbamide; LitalirAntineoplastic Agent; Ribonucleotide Reductase Inhibitorx    
Hydroxyzine Dihydrochloride68-88-2Arcanax; NeurolaxAntihistamine Agentx    
Hygromycin B31282-04-9 Antibiotic Agentx    
I-BET1260907-17-2 BET Inhibitorx x  
I-BET-1511300031-49-5GDK1210151ABET Inhibitorxxxx 
Ibrutinib936563-96-1Imbruvica; PCI-32765BTK Inhibitorx xxx
Ibudilast50847-11-5AV-411; Eyevinal; Ibudilastum; KetasPDE4 Inhibitorx    
Ibuprofen15687-27-1NeoProfenCOX Inhibitorx    
Ibutamoren Mesylate159752-10-0; 159634-47-6Crescendo; Ibutamoren; Ibutamoren Mesilate; MK-677Ghrelin Receptor Agonistx    
IC-87114371242-69-2IC87114PI3Kδ Inhibitorx x  
ICG001780757-88-2;847591-62-2ICG-001β-catenin/CBP Inhibitorxxx  
ICI 6319727277-00-5 PDE4 Inhibitorx    
Idebenone58186-27-9Catena; Raxone; SovrimaSynthetic Coenzyme Q10 (CoQ10) Analogx    
Idelalisib870281-82-6CAL-101; GS-1101; ZydeligPI3Kδ Inhibitorx xxx
IDO-IN-2914471-09-3 IDO Inhibitorx xx 
IFNß-1b145155-23-3Betaseron; INF-β 1b; INFβ 1b; Interferonß-1b; Interferonß1bCytokinex    
IFNα 2a IFN-α 2a; INF-α 2a; Interferon α 2aCytokinex    
IFNα 2b IFN-α 2b; INF-α 2b; Interferon α 2bCytokinex    
IFNγ82115-62-6Actimmune; Interferon gamma-1bCytokinex x  
IgG4 Isotype  IgG4 Control Antibodyx x  
IKK 161186195-62-9IKK Inhibitor VII; IKK-16IKK2 Inhibitorx    
IKK-2 Inhibitor IV507475-17-4 IKK2 Inhibitorx    
IL-10130068-27-8Interleukin 10Cytokinex x  
IL-12632331-09-0Interleukin 12Cytokinex    
IL-13148157-34-0Interleukin 13Cytokinex    
IL-17A Interleukin 17ACytokinex    
IL-17F Interleukin 17FCytokinex    
IL-1R Antagonist566914-00-9Interleukin 1 Receptor AntagonistIL-1 Receptor Inhibitorx    
IL-1β97599-21-8Interleukin-1βCytokinex    
IL-2 Aldesleukin; Interleukin 2; ProleukinCytokinex  x 
IL-27 Interleukin 27Cytokinex    
IL-29 Interferon λ1; Interleukin 29Cytokinex    
IL-32 Interleukin 32Cytokinex    
IL-33 Interleukin 33Cytokinex    
IL-35 Interleukin 35Cytokinex    
IL-4207137-56-2Interleukin 4Cytokinex    
IL-6 Rα CD126 ; Cluster of Differentiation 126Immunomodulating Agentx    
IL-8 CXCL8; Interleukin 8CXCR1/2 Agonistx    
Iloperidone133454-47-4FanaptAntipsychotic Agentx    
Iloprost78919-13-8VentavisEP1 Agonist; Prostanoid IP Receptor Agonistx    
Imatinib152459-95-5Gleevec; Imatinib Methansulfonate; ImatinibumBCR-ABL Inhibitorxx   
Imfinzi (durvalumab)  Anti-PD-L1 Antibody  xx 
Indomethacin53-86-1Aconip; Indocin; Indometacina; Indometacine; IndometacinumCOX Inhibitorx    
Indoximod110117-83-4; 26988-72-7NLG-8189IDO Inhibitorx xx 
Infliximab170277-31-3RemicadeTNFα Inhibitorxx  x
Iniparib160003-66-7BSI 201PARP Inhibitorx  x 
Insulin Aspart NovologInsulin Receptor Agonistx    
Insulin Glargine LantusInsulin Receptor Agonistx    
Insulin Lispro Humalog; Insulin Lispro RecombinantInsulin Receptor Agonistx    
IOX15852-78-8 Histone Demethylase JMJD Inhibitorx    
Ipilimumab477202-00-9MDX-010; MDX-101; MDX-CTLA-4; MOAB-CTLA-4; YervoyCTLA-4 Inhibitorx xx 
IRAK-1/4 Inhibitor I509093-47-4 IRAK-1/4 Inhibitorx    
Irinotecan100286-90-6CPT-11; Campto; Camptosar; Camptothecin-11DNA Topoisomerase (TOPO) I Inhibitorx x  
Irsogladine57381-26-7 PDE4 Inhibitorx    
Isoetharine Mesylate530-08-5Isoetarine Mesilateβ2 Adrenergic Receptor Agonistx    
Isoniazid54-85-3Isonicotinic acid hydrazide; Isonicotinsaeurehydrazid; IsonicotinylhydrazineAntibiotic Agentx    
Isotretinoin4759-48-213-cis-retinoic acid; AccutaneRAR/RXR Agonistx    
Itraconazole84625-61-6SporanoxCytochrome P450 51 Inhibitor, Ergosterol Synthesis Inhibitorxx   
Ivacaftor873054-44-5Kalydeco; VX770CFTR Potentiatorxx   
Ixekizumab TaltzIL-17A Inhibitorx    
JAK Inhibitor 1457081-03-7CMP 6; Merck-5; Pyridone 6JAK1 Inhibitorx    
JNJ-10397049708275-58-5JNJ 10397049Orexin Receptor Type 2 (OX2) Inhibitorx    
JNK Inhibitor VIII894804-07-0 JNK Inhibitorx    
JQ11268524-70-4 BET Inhibitorxxx  
JWH-015  CB1/2 Agonist x   
K252a  Multikinase Inhibitorx    
KD025 SLx-2119ROCK2 Inhibitorx    
Ketoconazole65277-42-1Fungares; Ketoderm; Nizoral; Orifungal M; PanfungolCytochrome P450 51 Inhibitorx    
Ketoprofen22071-15-4ActronCOX Inhibitorx    
Ketotifen Fumarate34580-14-8Ketotifen; Ketotifeno; Ketotifenum; ZaditorAntihistamine Agentx    
Ki16425355025-24-0Ki 16425LPA1, LPA3 Receptor Inhibitorx    
Kisspeptin-10 MetastatinKISS1 Agonist; GPR54 Agonistx    
KN93139298-40-1 CAMKII Inhibitorxx   
KNK437218924-25-5 Hsp Modulator; Hsp Inhibitor (Hsp 72, 73, 90, 105, 27, 40)x    
L-7448321177806-11-9 Farnesyltransferase Inhibitorx    
Lansoprazole103577-45-3A-65006; AG-1749; PrevacidProton Pump Inhibitorx    
Lapatinib388082-77-7GW 572016; Lapatinib Ditosylate; Lapatinib Tosilate Hydrate; TykerbTyrosine Kinase Inhibitor (ERBB1, ERBB2)x    
L-Arginine Hydrochloride1119-34-2 Vasodilatorx    
Larotrectinib1223403-58-4VitrakviTropomyosin Kinase Receptor (Trk) Inhibitorx    
Leflunomide75706-12-6Arava; Leflunomida; Leflunomidum; LefunomideDihydroorotate Dehydrogenase (DHODH) Inhibitorx x  
Lenalidomide191732-72-6RevlimidImmunomodulating Agent; Antineoplastic Agentx x  
Lenvatinib417716-92-8LenvimaTyrosine Kinase Inhibitorx    
Letrozole112809-51-5CGS 20267; FemaraCytochrome P450 19A1 Inhibitorx    
Levamisole Hydrochloride14769-73-4(-)-Tetramisole Hydrochloride; Ergamisol; Levamisole HCl; TramisolAntihelminthic Agentx    
LFM-A1362004-35-7 BTK Inhibitorx    
Linezolid165800-03-3PNU 100766; ZyvoxAntibiotic Agentx    
Linsitinib867160-71-2OSI-906IGF-1R Inhibitorx    
Liothyronine6893-02-3Liothyronin; Tresitope; TriiodothyronineThyroid Hormone Receptor Agonistx    
Liraglutide Liraglutida; Liraglutidum; Saxenda; VictozaGlucagon-like Peptide 1 (GLP-1) Receptor Agonistx    
Lithium Chloride7447-41-8 Inorganic Compoundxxxx 
Lofexidine Hydrochloride21498-08-8Lucemyraα2A Adrenergic Receptor Agonistx    
Lonidamine50264-69-2Diclondazolic acid; DoridaminaHexokinase Inhibitor; Glycolysis Inhibitorx    
Loperamide Hydrochloride34552-83-5 Opioid-receptor Agonistx    
Lopinavir192725-17-0A-157378.0; ABT-378; Aluviran; KoletraAntiretroviral Agent; Protease Inhibitorx    
Lorlatinib  ALK/ROS1 Inhibitor   x 
Lornoxicam70374-39-9Chlortenoxicam; XefoNSAID; Analgesic Agent; Anti-inflammatory Agentx    
Loteprednol Etabonate82034-46-6Alrex; LotemaxGlucocorticoid Receptor (GR) Agonistx    
Lovastatin75330-75-5Altoprev; Mevacor; MevinolinHMG-CoA Reductase Inhibitorx    
Loxapine Succinate27833-64-3Adasuve; LoxitaneAntipsychotic Agentx    
LP99  Bromodomain Inhibitorx    
LPS  TLR4 Agonistx xx 
Lumacaftor936727-05-8VX-809CFTR Modulatorx    
Luminespib747412-49-3AUY-922; NVP-AUY922Hsp90 Inhibitorx    
LY294002154447-36-6 CK2 Inhibitor; PI3K Inhibitorx x  
M344251456-60-7D237; Histone Deacetylase Inhibitor III; MS 344HDAC Inhibitorx    
Macitentan441798-33-0OpsumitET-A Inhibitor; ET-B Inhibitorx    
Manidipine89226-50-6ManyperCalcium Channel Blocker; Antihypertensive Agentx    
MCC950  NLRP3 Inhibitorx    
MDV3100915087-33-1Enzalutamide; MDV-3100; XtandiAndrogen Receptor (AR) Inhibitorx    
Meclocycline Sulfosalicylate73816-42-9Meclan; Meclan Cream; Mecloderm; MeclutinAntibiotic Agentx    
Medetomidine Hydrochloride86347-15-1Domitor; MPV 785; Medetomidineα2 Adrenergic Receptor Agonistx    
Medrysone2668-66-8HMS; HydroxymesteroneGlucocorticoid Receptor (GR) Agonistx    
Mefenamic Acid61-68-7CI-473; PonstelCOX Inhibitorx    
Megestrol Acetate595-33-5Megace; Megestrol; OvaridProgesterone Receptor (PR) Agonistx    
Menadione58-27-5Vitamin K3Phosphatase Inhibitor; Mitochondrial DNA Polymerase γ (pol γ) Inhibitorx    
Mepivacaine Hydrochloride1722-62-9Carbocaina; Meaverin; MepivastesinSodium Channel α Subunit Blocker; Topical Anesthetic Agentx    
Mequinol150-76-54-Methoxyphenol; MEHQDepigmentation Agentx    
Mesoridazine Besylate5588-33-0Benzenesulfonate; MesoridazineAntipsychotic Agentx    
Metaproterenol Sulfate5874-97-5Alupent; Metaprel; Orciprenalineβ2 Adrenergic Receptor Agonistx    
Metformin Hydrochloride657-24-9Haurymellin; Metformina; Metformine Pamoate; MetforminumAMPK Activator; Antihyperglycemic Agent x    
Methacholine Chloride Acetyl-beta-methylcholine Chloride; Amechol; Mecholyl Chloride; Methacholine; ProvocholineMuscarinic Acetylcholine Receptor Agonistx    
Methapyrilene Hydrochloride135-23-9Capathyn; Histadyl; Methacon; Methapyrilene; MethoxyleneAntihistamine Agentx    
Methazolamide554-57-4Naptazane; Neptazane; NeptazaneatCarbonic Anhydrase Inhibitorx    
Methocarbamol532-03-6Delaxin; Forbaxin; Miolaxin; Neuraxin; RobaxinMuscle Relaxerx    
Methotrexate59-05-2Abitrexate; Amethopterin; Emtexate; Ledertrexate; MTX; Metoject; Otrexup; RasuvoDihydrofolate Reductase (DHFR) Inhibitorx xx 
Methyclothiazide135-07-9 Diuretic; Antihypertensive Agentx    
Methyldopa555-30-6Aldomet; Alphamethyldopa; Dopamet; Medometα2 Adrenergic Receptor Agonistx    
Methylene Blue61-73-4 NOS Inhibitor; Guanylate Cyclase Inhibitorx    
Mevastatin73573-88-3CompactinHMG-CoA Reductase Inhibitorx    
Mianserine Hydrochloride21535-47-7Bolvidon; Lerivon; TolvonH1 Receptor Inhibitor; Antidepressantx    
Mifamurtide83461-56-7Mepact; Mifamurtide HydrateNOD2 Activatorx    
Milrinone78415-72-2 PDE3 Inhibitorx    
Mitoxantrone NovantroneTOPO II Inhibitor; Antineoplastic Agentx    
Mizolastine108612-45-9MizollenH1 Receptor Inhibitorx    
Mizoribine50924-49-7BredininImmunosuppressive Agent; DNA Synthesis Inhibitorx    
MK-22061032350-13-2 AKT Inhibitorx    
MK-8457  SYK Inhibitorx    
MLN8054869363-13-3 Aurora Kinase Inhibitorx    
Momelotinib CYT-387; GS-0387JAK1/2 Inhibitorxx   
Mometasone Furoate83919-23-7Asmanex; Elomet; NasonexGlucocorticoid Receptor (GR) Agonistx    
Monensin Sodium22373-78-0Coban; RumensinNa+ Ionophorex    
Monobenzone103-16-2Benoquin; MBEHSkin Whitening Agentx    
Montelukast158966-92-8MK 0476; MK-0476; SingulairCysLT1 Receptor Inhibitor; GPCR Ligandx    
Mosapride Citrate112885-42-4AS-4370; DSSTox_CID_26207; Gasmotin5-HT4 Receptor Agonistx    
Motilin  Motilin Receptor Agonistx    
Moxifloxacin Hydrochloride186826-86-8Avalox; Avelox; Moxeza; VigamoxAntimicrobial Agentx    
MRL-SYKi DRX_MRL-SYKiSYK Inhibitorx    
MRT673071190378-57-4 IKKε, MARK1-4, NUAK1 , TBK-1 Inhibitorxx   
Mycophenolic Acid24280-93-1Cellcept; Melbex; Mycophenolate; Mycophenolsaeure; MyforticIMPDH Inhibitorx    
Myxothiazol76706-55-3 Cytochrome c Reductase Inhibitor; Mitochondrial Inhibitorx    
N-Acetyl Cysteine616-91-1616-91-1; Acetadote; Acetylcysteine; Fluimucil; N-AcetylcysteineAntioxidantxx   
Nafcillin Sodium Monohydrate985-16-06-(2-Ethoxy-1-naphthamido)penicillinAntibiotic Agentx    
Nalmefene Hydrochloride58895-64-0NalmetreneOpioid Receptor Inhibitorx    
Naproxen22204-53-1Anaprox; Naprelan; Naprolag; NaprosynCOX Inhibitorx    
Navoximod1402836-58-1GDC-0919; NLG-919; NLG919; RG6078IDO Inhibitorx xx 
Nebivolol152520-56-4Bystolic; Lobivon; Nebilet; Nebivololum; R 67555β1 Adrenergic Receptor Inhibitorx    
Nefazodone83366-66-9Nefazodona; Nefazodone Hydrochloride; NefazodonumAntidepressant Agent; 5-HT2A Inhibitorx    
Neflamapomid209410-46-8VX 745; VX745p38 MAPK Inhibitorx x  
Nefopam Hydrochloride23327-57-3Acupan; Ajan; Nefadol; SilentanNon-opioid Analgesic Drugx    
Nelarabine121032-29-9ArranonDNA Inhibitorx    
Neomycin Sulfate1405-10-3Fradiomycin; Framycetin; Mycifradin; SoframycinAntibiotic Agentx    
Neostigmine Bromide114-80-7Eustigmin Bromide; Neo-Proserin; Neoserine Bromide; Proserine Bromide; ProstigminAcetylcholinesterase Inhibitorx    
Neuromedin B Beta-Neurokinin; Neuromedin K; Porcine Neurokinin BNMBR Agonistx    
NI-57 GTPL8573Bromodomain Inhibitorx    
Nialamide51-12-7Niamid; Niamide; Nuredal; SurgexMonoamine Oxidase Inhibitor (MAOI)x    
Nifuroxazide965-52-6RC-27109; SJ000287313STAT Inhibitorx    
Nintedanib656247-17-5BIBF 1120; Ofev; VargatefVEGFR, FGFR, PDGFR Kinase Inhibitorxx   
Nithiamide140-40-9Acinitrazole; AminitrozoleAntimicrobial Agentx    
Nitrofural59-87-0Furacilin; Furacin; NitrofurazoneAntibiotic Agentx    
Nitroprusside13755-38-9Nipride; Nitroferricyanide; NitropressVasodilatorx    
Nivolumab946414-94-4OpdivoPD-1 Inhibitorx xx 
Nodinitib-1799264-47-4CID-1088438; ML130NOD1 Inhibitorx    
Norethindrone68-22-4Norethisterone; UtovlanProgesterone Receptor (PR) Agonistx    
Nortriptyline Hydrochloride72-69-5Ateben; Avantyl; Demethylamitriptyline; Noritren; Psychostyl; SensavalSNRIx    
Nutlin-3  MDM2 Antagonist  x  
NVP-TAE684761439-42-3NVP-TAE 684; TAE684ALK Inhibitor; Kinase Modulatorx    
NVS1-PAK1-1 DRX_NVS1-PAK1-1PAK1 Inhibitorx    
Obeticholic Acid  FXR Agonist x   
Octadecanoic acid57-11-4 Organic Compoundx    
Odanacatib603139-19-1MK0822Cathepsin K Inhibitorxx   
ODN2006  TLR9 Agonistx    
ODN2395  TLR9 Agonistx    
OEA OleoylethanolaminePPARα Agonistx    
Ofloxacin82419-36-1Floxin; Ocuflox; Ofloxacine; TarividAntimicrobial Agentx    
Olaparib763113-22-0AZD 2281; AZD-2281; LynparzaPARP Inhibitorx xx 
Oligomycin A579-13-5MCH 32F0/F1 ATPase Inhibitor; Mitochondrial Inhibitorx x  
Olmutinib1353550-13-6BI-1482694Tyrosine Kinase Inhibitorx xx 
Omeprazole73590-58-6Antra; H-168/68; PrilosecProton Pump Inhibitorx    
Omipalisib1086062-66-9GSK-2126458; GSK2126458PI3K Inhibitor; mTOR Inhibitorxxxx 
ONC201  DRD2 Inhibitorx  x 
Oncostatin M106956-32-5 LIFR-α; OSMR Agonistx    
Ondansetron Hydrochloride99614-02-5ZofranAntinausea Agentx    
ONX 0914960374-59-8PR-957Immunoproteasome Inhibitorx    
Orlistat96829-58-2Alli; XenicalPI3K Inhibitor; mTOR Inhibitorx    
OTX015202590-98-5MK-8628BET Inhibitorxx x 
Oxaliplatin61825-94-3Diaminocyclohexane Oxalatoplatinum; Eloxatin; L-OHPAntineoplastic Agent; DNA Synthesis Inhibitorx x  
Oxaprozin21256-18-8Alvo; Daypro; Deflam; OxaprozineCOX Inhibitorx    
Oxethazaine126-27-2Betalgil; Mucaine; Oxaethacainum; OxetacaineLocal Anaestheticx    
Oxibendazole20559-55-1 Polymerase Inhibitorx    
Oxybuprocaine Hydrochloride5987-82-6Benoxinate HydrochlorideSodium Channel α Subunit Blocker; Topical Anesthetic Agentx    
Oxybutynin Chloride1508-65-2Ditropan; Oxibutinina; Oxibutyninum; Oxybutynin; OxytrolMuscarinic Acetylcholine Receptor (mAChR) Inhibitor x    
Ozagrel Hydrochloride78712-43-3Sodium Ozagrel; UNII-L256JB984DAntiplatelet Agent; Thromboxane A2 Synthesis (TXAS) Inhibitorx    
P22077 DUB InhibitorUSP47 Inhibitorx    
P7C3301353-96-8AK340958NAMPT Activator; Proneurogenic; Neuroprotectivex    
Paclitaxel33069-62-4Anzatax; Asotax; Bristaxol; Praxel; Taxol; Taxol KonzentratMicrotubule Disruptorx xx 
Palbociclib827022-33-3Ibrance; PD0332991CDK4/6 Inhibitorx xx 
Paliperidone144598-75-4InvegaDopamine (D2) Receptor Inhibitor; 5-HT2A Receptor Inhibitorx    
Palonosetron Hydrochloride135729-62-3Aloxi5-HT3A Receptor Inhibitorx    
Pam3CSK4  TLR1/TLR2 Agonistx    
Pamoic Acid Disodium6640-22-8Embonic AcidGPR35 Agonistx    
Panitumumab ABX-EGF; VectibixEGFR Inhibitorx xx 
Panobinostat404950-80-7Faridak; Farydak; LBH-589; LBH589HDAC Inhibitorx    
Paromomycin Sulfate1263-89-4Aminosidine Sulfate; Humatin; Paromomycin; Paromomycin Sulfate SaltAntibiotic Agentx    
Paroxetine Hydrochloride110429-35-1Aropax 20; Paroxat; Paroxetine HclSSRIx    
Pazopanib444731-52-6GW 78603; GW786034; Pazopanibum; VotrientMulti Tyrosine Kinase Receptor Inhibitor (c-KIT, FGFR, PDGFR, VEGFR) xx   
PBI-4050  Antifibrotic Agentxx   
PD098059167869-21-8 MEK Inhibitorx    
PD123319130663-39-7 Angiotensin II (AT2) Receptor Inhibitorx    
PD184352212631-79-3CI-1040MEK Inhibitorx    
PDGF-BB  PDGFRβ Activatorx    
Pembrolizumab KeytrudaPD-1 Inhibitorx xx 
Pemetrexed Disodium150399-23-8 Dihydrofolate Reductase (DHFR) Inhibitor; GAR Transformylase Inhibitor; Thymidylate Synthase Inhibitorx xx 
Penciclovir39809-25-1DenavirGuanosine Analogue; Antiviral Agentx    
Pentamidine50357-45-4Nebupent; PentamAntimicrobial Agentx    
Pergolide Mesylate66104-23-2Pergolide; Pergolide Methanesulfonate; PermaxDopamine Receptor Agonistx    
Perindopril Erbumine107133-36-8AceonAngiotensin-converting Enzyme Inhibitorx    
Pertuzumab 2C4 Antibody; MOAB 2C4; Omnitarg; Perjeta; rhuMAb-2C4HER2 Dimerization Inhibitorx    
PF-04217903956905-27-4 c-Met Inhibitorx    
PF-06297470  mGluR5 Inhibitorx    
PF-066508331817626-54-2 IRAK4 Inhibitorx    
PFI-11403764-72-6PF-06405761; PF-6405761BET Inhibitorxxx  
PFI-3  SMARCA2/4 Inhibitor; Polybromo 1 (PBRM1) Inhibitorx x  
PFI-4 PFI4Bromodomain Inhibitorx    
PHA-408503555-55-3 IKK2 Inhibitorx    
Phenazopyridine Hydrochloride136-40-3Bisteril; Mallophene; Phenazopyridine HCl; UrodineSodium Channel α Subunit Blocker; Topical Anesthetic Agentx    
Pheniramine Maleate132-20-7Avil-retard; Daneral; Inhiston; Naphcon; TrimetoseAntihistamine Agentx    
Phenylbutazone50-33-9Butatron; ButazolidinCOX Inhibitorx    
Phenylephrine Cyclomydril; Mydfrinα1 Adrenergic Receptor Agonistx    
Phorbol 12-myristate 13-acetate16561-29-8PMAPKC Activatorx    
Piclamilast144035-83-6Cpodpmb; RP 73401PDE4 Inhibitorx    
Picropodophyllin477-47-4AXL1717; PicropodophyllotoxinMicrotubule Disruptorx    
Pimasertib1236699-92-5AS 703026; AS703026MEK Inhibitorx    
Pimobendan74150-27-9VetmedinPDE3 Inhibitorx    
Pioglitazone111025-46-8Actos; Glustin; Pioglitazona; PioglitazonumPPARγ Agonistx    
Pirfenidone53179-13-8Esbriet; Etuary; KitosCell; Pirespa; PirfenexAntifibrotic Agentxx   
Pironetin151519-02-7 Microtubule Disruptorx    
Pizotifen Malate5189-11-7Pizotyline; Sandomigran5-HT Receptor Antagonistx    
Plerixafor155148-31-5AMD 3100CXCR4 Inhibitorxx   
PLX4720918505-84-7PLX-4720BRAF Inhibitorx    
PNU 74654113906-27-7 Wnt/β-catenin Pathway Inhibitorx    
Poly(I:C)HMW  TLR3 Agonistx    
Pomalidomide19171-19-83-amino Thalidomide; CC-4047Immunomodulating Agent; Antineoplastic Agentx    
Ponatinib 3-amino Thalidomide; AP 24534; AP24534; IclusigBCR-ABL Inhibitorxx   
Posaconazole171228-49-2Noxafil; Sch 56592CYP51 Inhibitorx    
PP1172889-26-8Mutant Kinases Inhibitor II; PP1 Analog IISrc Family Inhibitorx    
PP2421092351-67-1PP 242mTOR Inhibitorx    
Pralatrexate146464-95-1FolotynDHFR Inhibitorx    
Pramoxine Hydrochloride637-58-1 Topical Anestheticx    
Pranlukast103177-37-3OnonCysteinyl Leukotriene Receptor 1 (CYSLTR1) Antagonist x    
Praziquantel55268-74-1BiltricideAntimicrobial Agentx    
Prednisolone50-24-8Hydroretrocortine; Metacortandralone; Millipred; Omnipred; Orapred; PRDL; Pediapred; PrednisolonaGlucocorticoid Receptor (GR) Agonistx   x
Prednisone53-03-2Adasone; Dehydrocortisone; Deltasone; Meticorten; PrednisonumGlucocorticoid Receptor (GR) Agonistx    
Prilocaine Hydrochloride721-50-6CitanestAnaesthetic Agentx    
Primaquine Diphosphate90-34-6NSC 149765; TronolaneQuinone Reductase 2 Inhibitorx    
Probenecid57-66-9Benecid; Benemid; Probalan; Probecid; Probenecid AcidUricosuric Agentx    
Procarbazine Hydrochloride671-16-9Matulane; Nathulane; Natunalar; PROCARBAZINE HClAntineoplastic Agentx    
Progesterone57-83-0PrometriumProgesterone Receptor (PR) Agonistx    
Prostaglandin D241598-07-6PGD2DP Agonistx    
Prostaglandin E2363-24-6Cervidil; Dinoprostone; Prepidil; Prostin E2EP Agonistx    
PrRP-31 Prolactin Releasing Peptide-31hGR3/GPR10 Agonistx    
PRT062607 PRT-062607Syk Inhibitorx    
Pyridostigmine Bromide101-26-8Kalimin; Mestinon; Mestinon Bromide; RegonolCholinesterase Inhibitorx    
Pyrithioxin1098-97-11098-97-1; Bonifen; Encefabol; Pyrithioxine; PyritinolNeurotropic Agentx    
QRFP-26 P518GPR 103 Agonistx    
Quinacrine Dihydrochloride Dihydrate83-89-6Atabrine HydrochloridePLA2 (phophoslipase A2) Inhibitorx    
Quizartinib950769-58-1AC220FLT3 Inhibitorx    
R(-)rolipram85416-73-5Adeo; Rolipramum; ZK 62711PDE4 Inhibitorx    
RA11740397 (MLI2)  LRRK2 Inhibitorx    
Radicicol12772-57-5MonordenHSP90 Inhibitorxx   
Raltitrexed112887-68-0Tomudex; ZD1694Dihydrofolate Reductase Inhibitor; Thymidylate Synthase Inhibitorx    
Rapamycin53123-88-9AY 22989; Rapamune; SILA 9268A; Sirolimus; WY-090217mTOR Inhibitorxxxx 
RDEA119923032-37-5BAY 869766; RDEA-119; RefametinibMEK Inhibitorx    
Reboxetine Mesylate98769-84-7 Noradrenalin Uptake Inhibitorx    
Regorafenib755037-03-7BAY 73-4506Multikinase Inhibitor (VEGFR2-TIE2 Tyrosine Kinase)x    
Repaglinide135062-02-1GlucoNorm; NovoNorm; Prandin; RepaglinidumAntidiabetic Agentx    
Resiquimod144875-48-9 TLR7/TLR8 Agonistx    
Resveratrol501-36-0 CYP1A1 Inhibitorxx   
Retapamulin224452-66-8Altabax; AltargoAntimicrobial Agentx    
Retinol68-26-8 Vitamin Ax    
rhM-CSF Recombinant Human Macrophage-colony Stimulating Factor M-CSF Receptor Agonistx    
Rimonabant158681-13-1SR141716CB1 Inverse Agonist; GPCR Ligandx    
Riociguat AdempassGC Activator x   
Risedronate Sodium115436-72-1Actonel; Atelvia; BenetBiphosphonate; Bone Density Conservation Agentx    
Ritonavir155213-67-5A-84538; ABT-53; ABT-538; Abbott 84538; NorvirHIV Protease Inhibitorx    
RN486  BTK Inhibitorx    
Ro 106-992062645-28-7 Ubiquitin Ligase Inhibitorx    
Ro 20-172429925-17-5 PDE4 Inhibitorx    
Ro 320-1195  p38 MAPK Inhibitorx    
Ro 32-0432151342-35-7 PKC (c+n) Inhibitorx    
Ro 5126766946128-88-7RO5126766BRAF Inhibitor; MEK Inhibitorx    
Rofecoxib162011-90-7Ceoxx; MK 966; VioxxCOX-2 Inhibitorx    
Roflumilast162401-32-3Daliresp; Daxas; ROF; RoflumilastumPDE4 Inhibitorxx   
Roflumilast N-Oxide292135-78-5 PDE4 Inhibitorxx   
Rolipram61413-54-5Adeo; Rolipramum; ZK 62711PDE4 Inhibitorx    
Rosiglitazone122320-73-4 TZD; AvandiaPPARγ Agonistxxx  
Rosuvastatin287714-41-4 Rosuvastatin; CrestorHMG-CoA Reductase Inhibitorx    
Rotenone83-79-4Barbasco; Dactinol; Paraderil; TubatoxinMitochondrial Inhibitor; NADH Dehydrogenase Inhibitorx    
Roxadustat FG-4592HIF-PHI Inhibitorx    
Rucaparib Phosphate  PARP Inhibitor x   
Ruxolitinib941678-49-5INCB018424; JakafiJAK1/2 Inhibitorxxx  
RXDX-106  TAM Receptor Inhibitorx    
R-α-Methylhistamine6986-90-9 H3 Histamine Receptor Agonistx    
S31-201501919-59-1Nsc 74859STAT3 Inhibitorx    
Salbutamol Sulfate51022-70-9Albuterolβ2 Adrenergic Receptor Agonistx    
Salicylanilide87-17-22-Hydroxybenzanilide; N-PhenylsalicylamideAntimicrobial Agentx    
Salicylic Acid69-72-72-Carboxyphenol; 2-Hydroxybenzoic acid; O-hydroxybenzoic acidCOX Inhibitorx    
Salinomycin Monosodium55721-31-8Coxistac; SalinomycinP-glycoprotein 1 Inhibitorx    
Salmeterol Xinafoate94749-08-3Arial; Asmerole; Salmetedur; Serevent Diskusβ2 Adrenergic Receptor Agonistxx   
Saracatinib379231-04-6AZD 0530; AZD0530Src/Abl Inhibitorxx   
Sarafloxacin Hydrochloride91296-87-6 Antimicrobial Agentx    
Saxagliptin361442-04-8OnglyzaDPP-4 Inhibitor; Antidiabetic Agentx    
SB203580152121-47-6 p38 MAPK Inhibitorx    
SB431542301836-41-9 TGFβR1 Kinase Inhibitor; ALK Inhibitorxxxx 
SB525334 TGFβ RI Kinase Inhibitor VIIITGFβR1 Kinase Inhibitor; ALK Inhibitorx    
SB939929016-96-6PracinostatHDAC Inhibitorx    
SC-514354812-17-2 IKK2 Inhibitorx    
Scriptaid287383-59-9ScriptideHDAC Inhibitorx    
Secukinumab CosentyxIL-17A Inhibitorx    
Selonsertib1448428-04-3 ASK1 Inhibitorxx   
Selumetinib606143-52-6ARRY-142886; AZD6244MEK Inhibitorx x  
Semagacestat425386-60-3LY450139γ-Secretase Inhibitorx    
Serotonin 5-HT; 5-Hydroxytryptamine; Antemovis; EnteramineMonoamine Neurotransmitterx    
Sertraline79617-96-2ZoloftSSRIx    
SGC-CBP30  CREBBP/EP300 Bromodomain Inhibitorx x  
SGC-I-CBP112  CBP/p300 Bromodomain Inhibitorx    
SGI-17761025065-69-3Pim Kinase Inhibitor IXPIM Kinase Inhibitorx    
Shaoguamycin B2738-64-9Piericidin A; Piericidin A1; Piericidine AMitochondrial Inhibitor; NADH Dehydrogenase Inhibitorx    
Sildenafil Citrate171599-83-0ViagraPDE5 Inhibitorxx   
Simvastatin79902-63-9ZocorHMG-CoA Reductase Inhibitorxx   
SL 327305350-87-2 MEK Inhibitorx    
SLPI ALK1; ALP; BLPI; HUSI; HUSI-I; MPI; WAP4; WFDC4Peptidase Inhibitor Protein  x  
Sodium Hydroxide1310-73-2Caustic Soda; Lye; Sodium HydrateInorganic Compoundx    
Somatostatin 28  Somatostatin Receptor Agonistx    
Sonidegib  Smoothened (SMO) Inhibitor x   
Sorafenib Tosylate475207-59-1BAY 43-9006; Nexavar; Tosylate SaltMultikinase Inhibitor (RAF/VEGFR-2/PDGFRβ)xxx  
Sotagliflozin ZynquistaSGLT1/SGLT2 Inhibitorx    
SP600125129-56-61,9-PyrazoloanthroneJNK Inhibitorx    
SPD-304  TNFα Inhibitorx    
Sphingosine-1-phosphate26993-30-6C18-Sphingosine 1-phosphate; D-erythro-Sphingosine-1-phosphateS1P Receptor Agonistx    
Spiramycin8025-81-8RovamycineAntimicrobial Agentx    
Spironolactone52-01-752-01-7; Aldactone; Spiroctan; Spirolactone; VerospironAldosterone Inhibitorx    
SR2211  RORγ Inhibitorx    
SRT2104 Sirtuin ModulatorSIRT1 Activatorx    
ssRNA40 R-1075TLR8 Agonistx    
STA 5326541550-19-0ApilimodIL-12/IL-23 Inhibitorx    
Staurosporine62996-74-1AM-2282; STSMultikinase Inhibitorx  x 
SU6656330161-87-0 Src Family Inhibitorx    
Succinate Succinic AcidChemical Intermediatex    
Sulfasalazine599-79-1Azopyrin; Colo-Pleon; Salazosulfapyridine; Salicylazosulfapyridine; SulcolonAnti-inflammatory Agentx    
Sulforaphane  Phytochemical; Antioxidant; Detoxifying Enzyme Inducerx    
Sunitinib Malate341031-54-7SU011248; SU11248; SutentMultikinase Inhibitor (VEGFR2, CSF-1R, PDGFR, SCFR, FLT3, RET)xxx  
Synta66 CLC001531CRAC Channel Inhibitorx    
T0901317293754-55-9T 0901317LXR Agonist; FXR Agonistxx   
Tacrolimus104987-11-3FK-506; FR900506; NCGC00179232-01Calcineurin Inhibitor; FK506-binding Protein 1A Inhibitorx    
Tadalafil171596-29-5ADCIRCA; Cialis; Ic351; TadanafilPDE5 Inhibitorx    
Tafenoquine106635-81-8KrintafelAntimalarial Agentx    
Talazoparib1207456-01-6TalzennaPARP Inhibitorx  x 
Tamoxifen10540-29-1Genox; Nolvadex; Soltamox; TamifenEstrogen Receptor Modulatorx    
Tanespimycin75747-14-717-AAGHsp90 Inhibitorx x  
Taurolithocholic Acid6042-32-6 G Protein-coupled Bile Acid Receptor 1 Agonistx    
Teicoplanin61036-62-2Targocid; TicosinAntibiotic Agentx    
Telbivudine3424-98-4Epavudine; Sebivo; TyzekaAntiviral Agent; Thymidine β-L-nucleoside Analoguex    
Telmisartan144701-48-4BIBR 277; MicardisAngiotensin II (AT2) Receptor Inhibitorxx   
Temsirolimus162635-04-3CCI 779; ToriselFK506-binding Protein 1A (FKBP1A) Inhibitor; mTOR Inhibitorx    
Tenidap120210-48-29K7CJ74ONH; Tenidapum5-Lipoxygenase Inhibitor; COX1/2 Inhibitorx    
Tepotinib1100598-32-0EMD-1214063c-Met Inhibitorx    
Terbinafine91161-71-6Lamasil; Lamisil; Lamisil AT; SF-86-327; TerbinexAntimicrobial Agentx    
Teriflunomide108605-62-5A771726; Aubagio; Flucyamide; HMR1726Pyrimidine Synthesis Inhibitor; DHODH Inhibitorx    
Tetracycline Hydrochloride60-54-8Abramycin; Achromycin; Deschlorobiomycin; Tetracyclinum; TsiklomitsinAntibiotic Agentx    
TGFβ  TGFβRI/II Agonistx    
TGFβ2  TGFRI, TGFRII Agonistx    
TGFβ3  TGFRI, TGFRII Agonistx    
TGF-βRI Kinase Inhibitor396129-53-6 TGFβR1 Kinase Inhibitorx    
TGX-221663619-89-4Tgx 221PI3Kβ Inhibitorx    
Thapsigargin67526-95-8 SERCA Inhibitorxx   
Thiostrepton1393-48-2Alaninamide; Antibiotic A 8506; Antibiotic X 146; Bryamycin; ThiactinOligopeptide Antibioticx    
Tianeptine Sodium30123-17-2Coaxil; Stablon; TatinolTricyclic Antidepressantx    
Tigecycline220620-09-7GAR-936; TBG-MINO; Tygacil; WAY-GAR-936Antibiotic Agentx    
Tilorone Dihydrochloride27591-69-1 Antiviral Agent; Type I Interferon Inducerx xx 
Tin Protoporphyrin IX14325-05-4NSC 267099Heme Oxygenase Inhibitorx    
Tin(II) Chloride7772-99-8Stannous Chloride; Tin Protochloride; Tin SaltChemical Compoundx    
Tioxolone4991-65-5ThioxoloneCarbonic Anhydrase Inhibitorx    
Tipiracil HCl  Thymidine Phosphorylase Inhibitor  x  
Tiratricol51-24-1TriacThyroid Hormone Analogue; Physiologic Thyroid Hormonex    
TMP-153128831-46-9 Acetyl-coA Cholesterol Acyltransferase (ACAT) Inhibitorx    
TNP-470129298-91-5AGM-1470; Agm 1470; DRG-0148Antineoplastic Agentx    
Tofacitinib477600-75-2Tasocitinib; Tofacitinibum; XeljanzJAK1/3 Inhibitorxxx x
Topotecan Hydrochloride119413-54-6Hycamptamine; Hycamtin; SKF S-104864-ATOPO I Inhibitorx x  
Torcetrapib262352-17-0CP 529414; CP-529414CETP Inhibitorx    
Torin-11222998-36-8Torin1mTOR Inhibitorxx   
Torin-21223001-51-1Torin2mTOR Inhibitorxx   
Torsemide56211-40-6Demadex; TORSEMIDE; Torasemida; TorasemidumDiuretic Agentx    
Tozadenant870070-55-6SYN-115Adenosine A2a Receptor Inhibitorx xx 
Trametinib871700-17-3GSK1120212; MekinistMEK Inhibitorx xx 
Tranexamic Acid1197-18-8Cyklokapron; TranexamsaeurePlasminogen Inhibitorx    
Tranilast53902-12-8RizabenAntiallergic Agentxx   
trans-Triprolidine486-12-4 Antihistamine Agentx    
Trastuzumab Herceptin; HerclonHER2/neu Receptor Inhibitor  x  
Tretinoin302-79-4ATRA; Aberela; Retinoic Acid; Trans-Retinoic Acid; Vitamin A Acid; all-trans-Retinoic AcidRAR/RXR Agonistx    
Triamcinolone124-94-7 Glucocorticoid Receptor (GR) Agonistx    
Trichostatin A58880-19-658880-19-6; TSA; TrichostatinHDAC Inhibitorx    
Triflusal322-79-2Aflex; Disgren; Grendis; TrifluxPlatelet Antiaggregantx    
Trilostane13647-35-313647-35-3; Desopan; Trilostano; Trilostanum; Vetoryl3 β-Hydroxysteroid Dehydrogenase Inhibitor x    
Tropine120-29-6 3-Tropanol Atropine Precursorx    
Trypan Blue72-57-1Direct Blue 14; Membraneblue; TRYPAN BLUE; UNII-I2ZWO3LS3; VisionBlueDiazo Dyex    
Tubastatin A1252003-15-8 HDAC Inhibitorx    
Tunicamycin11089-65-9 Antibiotic Agentx    
TWEAK Human TWEAK; TNF-like Weak Inducer; TNFSF12Cytokinex    
Tyr[SO3H]27)-CCK825126-32-3C-Terminal Octapeptide of Cholecystokinin (CCK); Kinevac; SincalideStimulates Pancreatic Secretionx    
Tyrphostin AG 1296146535-11-7AG-1296PDGFR Inhibitorx    
U-75302119477-85-9 Leukotriene B4 (LTB4) Receptor Inhibitorx    
UK 14, 304  α2 Adrenergic Receptor Agonistx    
UNC0642  G9a and GLP Inhibitorx    
UNC20251429881-91-3 Mer Inhibitor; FLT3 Inhibitorx    
UO126109511-58-2U0126MEK Inhibitorx    
Upadacitinib1310726-60-3ABT-494JAK1 Inhibitorx    
Urolithin A  Microflora Metabolitex    
Ursodeoxycholic Acid128-13-2Actigall; Delursan; Ursodiol; UrsolvanBile Acidx    
Ursolic Acid77-52-1 Urson; Malol; PrunolCosmetic Additivex    
UTP Uridine triphosphateNucleotide x    
Vadimezan117570-53-35,6-Mexaa; DMXAADT-Diaphorase Inhibitorx x  
Valdecoxib181695-72-7BextraCOX2 Inhibitorx    
Valinomycin2001-95-8 Antibiotic Agentx    
Valnemulin Hydrochloride133868-46-9 Pleuromutilin Antibiotic x    
Valproic Acid1069-66-5Depakene; Depakine; Dipropylacetic acidHDAC Inhibitor; GABA Transaminase Inhibitorxx   
Vandetanib443913-73-3AZD6474; Caprelsa; ZD6474VEGFR2, EGFR Inhibitorx x  
Vardenafil330808-88-3Levitra; Staxyn; VardenafilumPDE5 Inhibitorx    
Vasopressin ADH; AVP; Antidiuretic Hormone; ArgipressinVasopressin Receptor Agonistx    
Vegetable Extract HI_V19  Vegetable Extractx    
VEGF-165127464-60-2 VEGF Receptor Agonistx    
Vemurafenib1029872-54-5BRAF(V600E) Kinase Inhibitor; PLX4032; RO5185426; ZelborafBRAF Inhibitorx x  
Venetoclax1257044-40-8ABT199; GDC-0199; VenclextaBcl-2 Inhibitorxxxx 
Verapamil52-53-9CP-165331; Calan; Covera-hs; Iproveratril; Isoptin; Tarka; VerelanL-type Calcium Channel Blockerx    
Vinblastine865-21-4VLB; VincaleukoblastineMicrotubule Disruptorx    
Vincristine Sulfate2068-78-2Leurocristine; Vincristin; Vincristina; Vincristine; VincristinumMicrotubule Disruptorx    
Vinorelbine71486-22-1Exelbine; Navelbine; UNII-Q6C979R91Y; Vinorelbina; VinorelbinumMicrotubule Inhibitorx    
Vinpocetine42971-09-5Apovincaminic Acid Ethyl Ester; Cavinton; TCV-3BPDE1 Inhibitorx    
Vismodegib 879085-55-9Erivedge; GDC-0449Hedgehog Pathway Inhibitorxx x 
Vitamin D250-14-6 Vitamin D Receptor (VDR) Agonistx    
VLX15701431280-51-1 DUB Inhibitorx    
Vorinostat149647-78-9SAHA; Suberoylanilide Hydroxamic Acid; ZolinzaHDAC Inhibitor (HDAC1, HDAC2, HDAC3, HDAC6)x x  
Voxtalisib1123889-87-1PI3K-IN-1; XL765PI3K Inhibitor; mTOR Inhibitorx    
VX702479543-46-9VX 702p38 MAPK Inhibitorx    
WKYMVm-NH2 BDBM86297Formyl Peptide Receptor (FPR1, FPR2) Agonistx    
Wortmannin19545-26-7Antibiotic SL-2052; KY 12420; SL-2052; WartmanninPI3Kinase Inhibitorx    
WS61421227-53-3 EBP1/IKK Inhibitorx    
XAV939284028-89-3 Tankyrase (TNKS) Inhibitorxxxx 
XL019945755-56-6 JAK2 Inhibitorx    
XL147956958-53-5PI3K Inhibitor X; PilaralisibPI3K Inhibitorx    
XL880849217-64-7EXEL-2880; Foretinib; GSK089; GSK1363089; XL-880VEGFR2 Inhibitorxxxx 
Y27632146986-50-7 ROCK1, ROCK2 Inhibitorxx   
YM155781661-94-7 Survivin Inhibitorx    
YM201636371942-69-7 PIKfyve Inhibitorx    
Zaprinast37762-06-4 PDE5/PDE6/PDE9 Inhibitorx    
Zinc Chloride7646-85-7 Chemical Compoundx    
Zinc Protoporphyrin IX15442-64-5ZPPHeme Oxygenase Inhibitorx    
Ziprasidone Hydrochloride122883-93-6Zeldox; ZiprasidoneAntipsychotic Agentx    
ZM4498294452-06-6 JAK3 Inhibitorx    
α-Amanitin23109-05-9Alpha-Amanitine; Alpha-Amatoxin; HSDB 3458RNA Polymerase II Inhibitorx