Targets by Family


ABL1(E255K)-phosphorylated ABL1(F317I)-nonphosphorylated ABL1(F317I)-phosphorylated ABL1(F317L)-nonphosphorylated ABL1(F317L)-phosphorylated
ABL1(H396P)-nonphosphorylated ABL1(H396P)-phosphorylated ABL1(M351T)-phosphorylated ABL1(Q252H)-nonphosphorylated ABL1(Q252H)-phosphorylated
ABL1(T315I)-nonphosphorylated ABL1(T315I)-phosphorylated ABL1(Y253F)-phosphorylated ABL1-nonphosphorylated ABL1-phosphorylated
ABL2 ALK ALK(1151Tins) ALK(C1156Y) ALK(F1174L)
ALK(L1196M) BMX BRK CSF1R-autoinhibited CSK
CTK DDR2(T654M) EGFR EGFR(E746-A750del) EGFR(G719C)
EGFR(G719S) EGFR(L747-E749del, A750P) EGFR(L747-S752del, P753S) EGFR(L747-T751del,Sins) EGFR(L858R)
EGFR(L858R,T790M) EGFR(L861Q) EGFR(S752-I759del) EGFR(T790M) EPHA1
EPHA2 EPHA3 EPHA6 EPHA8 EPHB6
ERBB2 ERBB3 FAK FER FES
FGFR2(N550K) FGFR3 FGFR3(G697C) FGFR3(K650E) FGFR3(V555M)
FGFR4 FLT1 FLT3(D835H) FLT3(D835V) FLT3(D835Y)
FLT3(ITD) FLT3(ITD,D835V) FLT3(ITD,F691L) FLT3(K663Q) FLT3(N841I)
FLT3(R834Q) FLT3-autoinhibited FRK FYN INSR
INSRR ITK JAK1(JH1domain-catalytic) JAK1(JH2domain-pseudokinase) JAK2(JH1domain-catalytic)
JAK3(JH1domain-catalytic) KIT KIT(A829P) KIT(D816H) KIT(D816V)
KIT(L576P) KIT(V559D) KIT(V559D,T670I) KIT(V559D,V654A) KIT-autoinhibited
LCK LTK LYN MERTK MET
MET(M1250T) MET(Y1235D) MST1R MUSK RET
RET(A883F) RET(M918T) RET(V804E) RET(V804L) RET(V804M)
ROS1 SRC SRMS TEC TIE1
TIE2 TNK1 TNK2 TXK TYK2(JH1domain-catalytic)
TYK2(JH2domain-pseudokinase) TYRO3 VEGFR2 YES ZAP70