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Kinase Targets by Technology

AAK1 ABL1(E255K)-phosphorylated ABL1(F317I)-nonphosphorylated ABL1(F317I)-phosphorylated ABL1(F317L)-nonphosphorylated
ABL1(F317L)-phosphorylated ABL1(H396P)-nonphosphorylated ABL1(H396P)-phosphorylated ABL1(M351T)-phosphorylated ABL1(Q252H)-nonphosphorylated
ABL1(Q252H)-phosphorylated ABL1(T315I)-nonphosphorylated ABL1(T315I)-phosphorylated ABL1(Y253F)-phosphorylated ABL1-nonphosphorylated
ABL1-phosphorylated ABL2 ACVR1 ACVR1B ACVR2A
ACVR2B ACVRL1 ADCK3 ADCK4 AKT1
AKT2 AKT3 ALK ALK(1151Tins) ALK(C1156Y)
ALK(F1174L) ALK(L1196M) AMPK-alpha1 AMPK-alpha2 ANKK1
ARK5 ASK1 ASK2 AURKA AURKB
AURKC BIKE BMPR1A BMPR1B BMPR2
BMX BRAF BRAF(V600E) BRK BRSK1
BRSK2 BUB1 CAMK1 CAMK1B CAMK1D
CAMK1G CAMK2A CAMK2B CAMK2D CAMK2G
CAMK4 CAMKK1 CAMKK2 CASK CDC2L1
CDC2L2 CDC2L5 CDK1 CDK10 CDK11
CDK12 CDK2 CDK20 CDK3 CDK4
CDK4-cyclinD1 CDK4-cyclinD1(F93L) CDK4-cyclinD3 CDK5 CDK6
CDK7 CDK8 CDK9 CDKL1 CDKL2
CDKL3 CDKL5 CHEK1 CHEK2 CIT
CLK3 CLK4 CSF1R-autoinhibited CSK CSNK1A1
CSNK1A1L CSNK1E CSNK1G1 CSNK1G2 CSNK1G3
CSNK2A1 CSNK2A2 CTK DAPK1 DAPK2
DAPK3 DCAMKL1 DCAMKL2 DCAMKL3 DDR2(T654M)
DLK DMPK DMPK2 DRAK1 DRAK2
DYRK1A DYRK1B DYRK2 EGFR EGFR(E746-A750del)
EGFR(G719C) EGFR(G719S) EGFR(L747-E749del, A750P) EGFR(L747-S752del, P753S) EGFR(L747-T751del,Sins)
EGFR(L858R) EGFR(L858R,T790M) EGFR(L861Q) EGFR(S752-I759del) EGFR(T790M)
EIF2AK1 EPHA1 EPHA2 EPHA3 EPHA6
EPHA8 EPHB6 ERBB2 ERBB3 ERK1
ERK1(Q122L) ERK2 ERK3 ERK4 ERK5
ERK8 ERN1 FAK FER FES
FGFR2(N550K) FGFR3 FGFR3(G697C) FGFR3(K650E) FGFR3(V555M)
FGFR4 FLT1 FLT3(D835H) FLT3(D835V) FLT3(D835Y)
FLT3(ITD) FLT3(ITD,D835V) FLT3(ITD,F691L) FLT3(K663Q) FLT3(N841I)
FLT3(R834Q) FLT3-autoinhibited FRK FYN GAK
GCN2(Kin.Dom.2,S808G) GRK1 GRK2 GRK3 GRK4
GRK7 GSK3A GSK3B HASPIN HIPK1
HIPK2 HIPK3 HIPK4 HPK1 HUNK
ICK IKK-alpha IKK-beta IKK-epsilon INSR
INSRR IRAK1 IRAK2 IRAK3 IRAK4
ITK JAK1(JH1domain-catalytic) JAK1(JH2domain-pseudokinase) JAK2(JH1domain-catalytic) JAK3(JH1domain-catalytic)
JNK1 JNK2 JNK3 KIT KIT(A829P)
KIT(D816H) KIT(D816V) KIT(L576P) KIT(V559D) KIT(V559D,T670I)
KIT(V559D,V654A) KIT-autoinhibited LATS1 LATS2 LCK
LIMK1 LIMK2 LKB1 LOK LRRK2
LRRK2(G2019S) LTK LYN LZK MAK
MAP3K1 MAP3K15 MAP3K2 MAP3K3 MAP3K4
MAP4K2 MAP4K3 MAP4K4 MAP4K5 MAPKAPK2
MAPKAPK5 MARK1 MARK2 MARK3 MARK4
MAST1 MEK2 MEK3 MEK4 MEK5
MEK6 MELK MERTK MET MET(M1250T)
MET(Y1235D) MINK MKK7 MKNK1 MKNK2
MLCK MLK1 MLK2 MLK3 MLKL
MLKL(full-length) MRCKA MRCKB MST1 MST1R
MST2 MST3 MST4 MTOR MUSK
MYLK MYLK2 MYLK4 MYO3A MYO3B
NDR1 NDR2 NEK1 NEK10 NEK11
NEK2 NEK3 NEK4 NEK5 NEK6
NEK7 NEK9 NIM1 NLK OSR1
p38-alpha p38-beta p38-delta p38-gamma PAK1
PAK2 PAK3 PAK4 PAK6 PAK7
PASK PCTK1 PCTK2 PCTK3 PDPK1
PFCDPK1(P.falciparum) PFPK5(P.falciparum) PFTAIRE2 PFTK1 PHKG1
PHKG2 PIK3C2B PIK3C2G PIK3CA PIK3CA(C420R)
PIK3CA(E542K) PIK3CA(E545A) PIK3CA(E545K) PIK3CA(H1047L) PIK3CA(H1047Y)
PIK3CA(I800L) PIK3CA(M1043I) PIK3CA(Q546K) PIK3CB PIK3CD
PIK3CG PIK4CB PIKFYVE PIM2 PIM3
PIP5K1A PIP5K1C PIP5K2B PIP5K2C PKAC-alpha
PKAC-alpha(L206R) PKAC-beta PKMYT1 PKN1 PKN2
PKNB(M.tuberculosis) PLK1 PLK2 PLK3 PLK4
PRKCD PRKCE PRKCH PRKCI PRKCQ
PRKD1 PRKD2 PRKD3 PRKG1 PRKG2
PRKR PRKX PRP4 QSK RAF1
RET RET(A883F) RET(M918T) RET(V804E) RET(V804L)
RET(V804M) RIOK1 RIOK2 RIOK3 RIPK1
RIPK3 RIPK4 RIPK5 ROCK1 ROCK2
ROS1 RPS6KA4(Kin.Dom.1-N-terminal) RPS6KA4(Kin.Dom.2-C-terminal) RPS6KA5(Kin.Dom.1-N-terminal) RPS6KA5(Kin.Dom.2-C-terminal)
RSK1(Kin.Dom.1-N-terminal) RSK1(Kin.Dom.2-C-terminal) RSK2(Kin.Dom.1-N-terminal) RSK2(Kin.Dom.2-C-terminal) RSK3(Kin.Dom.1-N-terminal)
RSK3(Kin.Dom.2-C-terminal) RSK4(Kin.Dom.1-N-terminal) RSK4(Kin.Dom.2-C-terminal) S6K1 SBK1
SGK SgK110 SGK2 SGK3 SIK
SIK2 SLK SNARK SNRK SRC
SRMS SRPK1 SRPK2 SRPK3 STK16
STK33 STK35 STK36 STK39 TAK1
TAOK1 TAOK2 TAOK3 TBK1 TEC
TESK1 TGFBR1 TGFBR2 TIE1 TIE2
TLK1 TLK2 TNIK TNK1 TNK2
TNNI3K TRPM6 TSSK1B TSSK3 TTK
TXK TYK2(JH1domain-catalytic) TYK2(JH2domain-pseudokinase) TYRO3 ULK1
ULK2 ULK3 VEGFR2 VPS34 VRK2
WEE1 WEE2 WNK1 WNK2 WNK3
WNK4 YANK1 YANK2 YANK3 YES
YSK1 YSK4 ZAK ZAP70