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Targets / GPCR Targets / GPCR Targets by Technology
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Targets
  • Alphabetical Target List
  • GPCR Targets
    • GPCR Targets by Therapeutic/Disease Area
    • GPCR Targets by Technology
  • Kinase Targets
  • Checkpoint Receptors
  • Ion Channels
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GPCR Targets by Technology

ADCYAP1R1 ADORA1 ADORA2A ADORA2B ADORA3
ADRA1A ADRA2A ADRA2C ADRB1 ADRB2
ADRB3 AGTRL1 AVPR2 BDKRB1 BRS3
C3AR1 C5AR1 CALCR CALCRL-RAMP1 CALCRL-RAMP3
CALCR-RAMP3 CASR CCR1 CCR10 CCR5
CCR6 CCR7 CHRM2 CHRM4 CMKLR1
CNR1 CNR2 CRHR1 CRHR2 CRTH2
CXCR1 CXCR2 CXCR3 CXCR4 CXCR5
CXCR6 CYSLTR2 DRD1 DRD2L DRD2S
DRD4 DRD5 EBI2 EDG1 EDG2
EDG3 EDG4 F2RL1 FFAR1 FFAR2
FFAR3 FPR1 FPR3 FPRL1 FSHR
GABBR1-GABBR2 GALR1 GALR2 GCGR GHRHR
GIPR GLP1R GLP2R GNRHR GPBAR1
GPR109A GPR109B GPR17 GPR35 GPR39
GPR81 GPR84 GRM1 GRM2 GRM3
GRM4 GRM5 GRM6 HRH2 HRH3
HTR1A HTR1B HTR1F HTR5A HTR7A
HTR7B HTR7D LHCGR LTB4R MC1R
MC3R MC4R MC5R MCHR1 mGIPR
mGLP1R MRGPRX1 mRXFP1 mTAAR1 MTNR1A
MTNR1B NPBWR1 NPBWR2 NPFFR1 NPY2R
OPRD1 OPRK1 OPRL1 OPRM1 OXER1
OXGR1 P2RY1 PPYR1 PROKR1 PTAFR
PTGDR PTGER1 PTGER2 PTGER3 PTGFR
PTGIR PTHR1 PTHR2 rDRD1 rDRD2L
rDRD2S rTAAR1 RXFP1 RXFP2 RXFP3
RXFP4 SCTR SSTR2 SSTR3 SSTR4
SSTR5 TAAR1 TACR3 TSHR(L) VIPR1
VIPR2 XCR1
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