GPCR Targets by Technology

ADCYAP1R1 ADORA1 ADORA2B ADORA3 ADRA1B
ADRA1D(82-572) ADRA2A ADRA2B ADRA2C ADRB1
ADRB2 AGTR1 AGTRL1 AVPR1A AVPR1B
AVPR2 BAI1 BAI2 BAI3 BDKRB1
BDKRB2 BRS3 C3AR1 C5AR1 C5L2
CALCR CALCRL-RAMP1 CALCRL-RAMP2 CALCRL-RAMP3 CALCR-RAMP2
CALCR-RAMP3 CCKAR CCKBR CCR1 CCR10
CCR2 CCR3 CCR4 CCR5 CCR6
CCR7 CCR8 CCR9 CCRL1 CCRL2
cEDG5 cGPR91 CHRM1 CHRM2 CHRM3
CHRM4 CHRM5 CMKLR1 CNR1 CNR2
CRHR1 CRHR2 CRTH2 CX3CR1 CXCR1
CXCR2 CXCR3 CXCR4 CXCR5 CXCR6
CXCR7 cyno CXCR1 cyno CXCR2 cyno GPR120 DARC
DRD1 DRD2L DRD2S DRD3 DRD4
DRD5 EBI2 EDG1 EDG2 EDG3
EDG4 EDG5 EDG6 EDG7 EDNRA
EDNRB F2R F2RL1 F2RL3 FFAR1
FFAR2 FPR1 FPRL1 FSHR GALR1
GALR2 GCGR GHSR GHSR1b GIPR
GLP1R GLP2R GPBAR1 GPR1 GPR101
GPR103 GPR107 GPR109A GPR109B GPR119
GPR12 GPR120 GPR120S GPR123 GPR132
GPR135 GPR137 GPR139 GPR141 GPR142
GPR143 GPR146 GPR148 GPR149 GPR15
GPR150 GPR151 GPR152 GPR157 GPR161
GPR162 GPR17 GPR171 GPR173 GPR176
GPR18 GPR182 GPR20 GPR22 GPR23
GPR25 GPR26 GPR27 GPR3 GPR30
GPR31 GPR32 GPR35 GPR37 GPR37L1
GPR39 GPR4 GPR45 GPR50 GPR52
GPR55 GPR6 GPR61 GPR65 GPR75
GPR78 GPR79 GPR83 GPR84 GPR85
GPR88 GPR92 GPR97 GRPR HCRTR1
HCRTR2 HRH1 HRH2 HRH3 HRH4
HTR1A HTR1B HTR1E HTR1F HTR2A
HTR2C HTR2C(VGV) HTR2C(VNV) HTR2C(VSV) HTR5A
HTR6 KISS1R LGR4 LGR5 LGR6
LHCGR LTB4R mADCYAP1R1 mADORA2B mADORA3
mADRA1B mAGTRL1 mAVPR2 mBRS3 MC1R
MC3R MC4R mC5AR1 MC5R mCCKAR
mCCR1 mCCR2 mCCR3 mCCR4 mCCR5
mCCR6 mCCR7 mCCR8 mCCR9 MCHR1
MCHR2 mCMKLR1 mCNR1 mCNR2 mCRHR1
mCRTH2 mCXCR2 mCXCR3 mCXCR4 mCXCR5
mCXCR6 mCXCR7 mDRD5 mEBI2 mEDG1
mEDG3 mEDG5 mEDNRA mEDNRB mFFAR1
mFPR1 mFPR2 mGALR1 mGALR2 mGCGR
mGHSR mGIPR mGLP1R mGPR1 mGPR120
mGPR84 mHCRTR1 mHTR2A mHTR2C MLNR
mLTB4R mMC3R mMC4R mMC5R mMCHR1
mNPY1R mNPY2R mOPRD1 mOPRK1 mOPRM1
mOXTR mP2RY12 mP2RY6 mPPYR1 mPTAFR
mPTGER4 mPTGIR MRGPRD MRGPRE MRGPRF
MRGPRX1 MRGPRX2 MRGPRX4 mRXFP3 mRXFP4
mSSTR2 mSSTR5 mTACR1 MTNR1A MTNR1B
mUTR2 mVIPR1 NMBR NMU1R NPBWR1
NPBWR2 NPFFR1 NPSR1b NPY1R NPY2R
NTSR1 OPN5 OPRD1 OPRK1 OPRL1
OPRM1 OXER1 OXGR1 OXTR P2RY1
P2RY11 P2RY12 P2RY2 P2RY4 P2RY6
P2RY8 PPYR1 PRLHR PROKR1 PROKR2
PTAFR PTGER1 PTGER2 PTGER3 PTGER4
PTGFR PTGIR PTHR1 PTHR2 rCHRM4
rCRTH2 rDRD1 rDRD2L rDRD2S rEDG5
rFFAR1 rGPR120 rGPR35 rHTR2C rOPRM1
rPROKR1 rPROKR2 rPTGER4 rVIPR1 RXFP3
RXFP4 SCTR sEDG5 SSTR1 SSTR2
SSTR3 SSTR4 SSTR5 TAAR5 TACR1
TACR2 TACR3 TBXA2R TRHR TSHR(L)
UTR2 VIPR1 VIPR2 XCR1