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BioMAP Recommended Benchmarks

Of the over 4,000 compounds that have been profiled using the BioMAP platform, the following compounds have been curated to provide the best starting point when identifying benchmarks for your BioMAP project. Included benchmarks were selected for their complete dosing and lack of overt cytoxicity..
 
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Agent Name :
Description :
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Agent Name ▲DescriptionSynonymDiversityPLUSFibrosisCRCNSCLC
(+/-)-NicotineNicotinic Acetylcholine Receptor Agonist 1   
(R,S)-TocopherolAntioxidant; Lipid SolubleVitamin E1   
(S)-FTY720 PhosphateS1P1 Agonist 1   
(S)-ReticulineAlkaloid 1   
(S)-Reticuline 3-O-sulfateCNS Depressant 1   
(S)-Reticuline 7-O-sulfateCNS Depressant 1   
15(R)-Prostaglandin D2DP Agonist 1   
1-Methyl-L-TryptophanIDO Inhibitor 1   
22(R)-Hydroxy CholesterolLXRα Agonist 1   
24(S)-HydroxycholesterolLXRα Agonist 1   
2-Chloroethyl Ethyl SulfideVesicantSulfur Mustard1   
2-Cl-IB-MECAAdenosine A3 Receptor Agonist 1   
2-IodomelatoninMelatonin Receptor Agonist 1   
2-MethoxyestradiolMicrotubule Disruptor2-methoxy-17beta-estradiol1   
4-Aminobenzoic AcidAntifibrotic; Vitamin B Complex Member 1   
5a-POPCCholesterol Efflux Promoter; Apolipoprotein 1   
5A-SMCholesterol Efflux Promoter5A-sphingomyelin1   
8-Br-cAMPPKA Activator 1   
8-CPT-cAMPPKA Activator; PKG Activator 1   
8-Hydroxy-5-nitroquinolineAntimicrobial Agent; Anticancer AgentNitroxoline1   
8-HydroxyquinolineAntimicrobial Agent 1   
9-cis-Retinoic AcidRAR/RXR Agonist 1   
Abacavir SulfateHuman Immunodeficiency Virus Type 1 Reverse Transcriptase Inhibitor 1   
AbirateroneCYP17A1 InhibitorCB75981   
Abiraterone AcetateCYP17A1 InhibitorCB76301   
AcadesineAMPK ActivatorAICAR1   
AcarboseMaltase-glucoamylase Inhibitor; Pancreatic α-amylase Inhibitor 1   
AcemetacinNSAIDEmflex1   
AcetaminophenCOX InhibitorTylenol; Paracetamol; Acephen; APAP1   
Acetic AcidOrganic SolventGlacial Acetic Acid1   
AcetonitrileOrganic Solvent 1   
AcetylcysteineMucolytic Agent 1   
Acetylsalicylic acidCOX 1/2 Inhibitor; NSAIDAcetylsalicylate; Aspirin1   
AcitretinRAR/RXR Agonist; Oral Retinoid 1   
AcriflavinAntiseptic Agent 1   
Actinomycin DRNA Polymerase Inhibitor; DNA InhibitorCosmegen; Dactinomycin1   
ActinoninPeptide Deformylase Inhibitor 1   
AdalimumabTNFα AntagonistHumira1   
AdapaleneRAR/RXR Agonist; Vitamin A Derivative; Retinoic Acid Analogue 1   
Adefovir DipivoxilntRT Inhibitor; Nucleotide Analog Reverse Transcriptase InhibitorPreveon, Hepsera1   
AdenineNucleobase; Purine Derivative 1   
AEG3482Hsp90 Inhibitor 1   
AfatinibEGFR/HER2 InhibitorBIBW29921   
AG1478EGFR Inhibitor 1   
AlbendazoleMicrotubule Inhibitor; Anthelmintic AgentZental; Valbazen; SK&F 62979; Albenza1   
AldosteroneMR AgonistAldocorten; Aldocortin; Electrocortin1   
AlendronateFarnesyl Diphosphate Synthase InhibitorFosamax1   
AlfacalcidolVitamin D Analogue 1   
all-trans-Retinoic AcidRAR/RXR Agonist 1   
AlprostadilEP Agonist; Prostanoid Receptor Agonist (EP1, EP2)Alprostadilum; Prostaglandin E11   
AltretamineAntineoplastic AgentHexalen1   
Alverine CitrateSmooth Muscle Relaxant; 5-HT1A AntagonistPhenpropamine Citrate1   
AM966LPA1 Receptor Antagonist 11  
AMD 3465CXCR4 Antagonist AMD 3465 Hexahydrobromide1 1 
AmfebutamoneNorepinephrine-dopamine Reuptake Inhibitor (NDRI)Budeprion; Elontril; Wellbutrin; Quomem; Prexaton; Voxra; Bupropion1   
Amfenac SodiumCOX Inhibitor; NSAID 1   
AMG-208c-MET Inhibitor 1   
AMG548p38 MAPK Inhibitor 1   
AminoglutethimideAdrenal Steroidogenesis InhibitorCytadren1   
AminophyllinePDE Inhibitor; Adenosine Receptor AntagonistTruphylline; Theophyllamine1   
AmlexanoxAnti-inflammatory Agent; Antiallergic Agent; Immunomodulator 1   
AmodiaquinHistamine N-methyltransferase Inhibitor 1   
Amphotericin BAntifungal AgentAmbisome; Abelcet; Amphotec1   
AmprenavirProtease Inhibitor Agenerase1   
AnacetrapibCETP Inhibitor 1   
AnakinraIL-1 Receptor AntagonistICIL-1RA; IL-1RN; IL-1ra; IL1 inhibitor; IRAP; Kineret1   
Antazoline HClHistamine (H1) Receptor Antagonist 1   
Antimycin ACytochrome c Reductase Inhibitor; Mitochondrial Inhibitor 1   
Apelin-13Apelin Receptor (APJ) Ligand 1   
ApilimodIL-12/IL-23 AntagonistSTA 53261   
ApoptolidinF(0)F(1) ATPase Inhibitor; Mitochondrial Inhibitor 1   
ApremilastPhosphodiesterase 4 (PDE4) Inhibitor 1   
ArtemisininAntimalaria Agent 1   
AS1892802ROCK1/2 Inhibitor 1   
AS2444697IRAK4 Inhibitor 1   
AS601245JNK Inhibitor 1   
AS605240PI3K Inhibitor (α, β, γ) 1   
AsenapineAtypical Antipsychotic; Multi Receptor Antagonist 1   
AstemizoleHistamine (H1) Receptor AntagonistAstemison; Astemizolum1   
Atazanavir SulfateAntiretroviral Agent; Protease Inhibitor  1   
AtorvastatinHMG-CoA Reductase InhibitorLipitor; Lipovastatinklonal1   
AtovaquoneCytochrome b InhibitorAtavaquone1   
ATPCoenzymeAdenosine triphosphate;1   
Atracurium BesylateMuscle-type Nicotinic Acetylcholine Receptor Antagonist 1   
AxitinibVEGFR2 InhibitorInlyta1   
Azaguanine-8Purine Nucleotide Synthesis Inhibitor; Xanthine Oxidase Inhibitor 1   
AzaperoneDopamine Receptor AntagonistSuicalm; Stresnil; R-19291   
Azatadine DimaleateHistamine and Cholinergic InhibitorAzatadine Maleate; Bonamid; Idulian1   
AzathioprinePurine Metabolism AnatgonistImuran; BW-57-322; Azasan1   
AZD1208PIMK Inhibitor 1   
AZD4547FGFR Inhibitor 1   
AZD8055mTOR Inhibitor 1   
AzithromycinBacterial 70S Ribosome InhibitorAzasite; Azenil; Azifast; Azigram; Azimakrol; Hemomycin; Zithromax1   
Bacitracin ZincC55-isoprenyl Pyrophosphate Inhibitor 1   
Bafilomycin A1V-ATPase Antagonist 1   
Bardoxolone MethylNRF2 ActivatorCDDO-methyl Ester1   
BaricitinibJAK Inhibitor 1   
BDH35145960bBET Inhibitor 1   
BDV0005266bBromodomain Inhibitor 1   
Benzethonium ChloridenAChR Inhibitor; Nicotinic Acetylcholine Receptor InhibitorPhemerol Chloride; Microklenz1   
BenzocaineAnesthetic 1   
Benzydamine HClNSAIDAF-864; Tantum1   
BeraprostProstacyclin Analogue 1   
BerberineDipeptidyl Peptidase IV Inhibitor; PTP1B Inhibitor 1   
BergaptenPsoralen 1   
BetamethasoneGlucocorticoid Receptor (GR) AgonistAlphatrex; Uticort; Taclonex; SCH-4831; Celestone1   
Betamethasone DipropionateGlucocorticoid Receptor (GR) AgonistDiprolene1   
Betamethasone ValerateGlucocorticoid Receptor (GR) AgonistBetnovate1   
BetamipronCarbapenem Antibiotic 1   
BevacizumabVEGFA InhibitorAvastin; anti-VEGF1   
BI 2536BET Inhibitor; PLK1 Inhibitor 1 1 
BI-10nIL-2 Inducible T-cell Kinase (ITK) Antagonist 1   
BIBX1382EGFR Inhibitor 1   
BilirubinHeme Metabolite 1   
Biperiden HClAcetylcholine Inhibitor 1   
BisacodylLaxative 1   
Bismuth Subcitrate PotassiumAntibiotic 1   
Bleomycin SulfateDNA Inhibitor 1   
BMP-7Activin Receptor Agonist (Activin RIA, RIIA, RIIB; BMPR-IA, BMPR-IB, BMPR-II)Osteogenic Protein-1 (OP-1)1   
BMS-777607cMET, AXL, RON and TYRO3 Inhibitor 1   
BortezomibProteasome InhibitorVelcade11  
BosentanEndothelin Receptor Antagonist (ET-A, ET-B)Bosentan Hydrate; Bosentanum; Tracleer1   
BosutinibMultikinase Inhibitor ( Bcr-Abl, SRc)SKI-6061  1
Brefeldin AARF1 Inhibitor 1   
Bromfenac SodiumNSAID; COX Inhibitor 1   
BromosporineBRD Inhibitor 1   
BrompheniramineAntihistamine; Histamine (H1) Receptor AntagonistBromfed; Dimetapp; Bromfenex; Dimetane; BPN; Lodrane1   
BroxyquinolineAntiprotozoal AgentDibromohydroxyquinoline1   
BSI-201PARP Inhibitor 1   
BSK_4925Lck InhibitorLymphocyte Specific Kinase1   
BSK_anti-CTLA4Anti-CTLA-4 Monoclonal Antibody; CTLA-4 Inhibitor 1   
BSK_RORgRORγ Inhibitor 1   
BucladesinePDE4 Inhibitor 1   
BudesonideGlucocorticoid Receptor (GR) Agonist 11  
BusulfanAntineoplastic AgentMyleran, Busulfex1   
BW 245CDP Agonist 1   
BW 246CDP Agonist 1   
CabozantinibVEGFR2 InhibitorXL184; Cometriq1   
CalcifediolVitamine D3 Metabolite 1   
CalcimycinCalcium IonophoreA231871   
CalcitriolVitamin D Receptor (VDR) AgonistCalcijex; Calcitriolum; Decostriol; Rocaltrol1   
Calcium ChlorideSaltCaCl2; Calcium Chloride Anhydrous1   
CantharidinProtein Phosphatase 2A (PP2A) InhibitorCantharone1   
CAPE15-Lipoxygenase Inhibitor 1   
CarbimazoleAntithyroid AgentAthyromazole1   
CarboplatinDNA Repair InhibitorParaplat; Paraplatin; Paraplatin-AQ  1 
CardarinePPARd AgonistGW5015161 11
Carfilzomib20S Proteasome Inhibitor; 26S Proteosome InhibitorKyprolis; PR-1711   
CarmofurPyrimidine Analogue; Antineoplastic AgentHCFU (1-hexylcarbamoyl-5-fluorouracil)1   
CarprofenCOX Inhibitor; NSAIDRimadyl; Imadyl; Quellin; Novox; Imafen; Rovera1   
CarvedilolAdrenergic Receptor Antagonist (α1,β1, β2) Carvedilolum; Coreg; SKF 105517; Beta Blocker1   
CAY10410PPARγ Agonist 1   
CCG 1423MRTF-A Inhibitor; Rho Kinase/ROCK Signaling InhibitorMyocardin-related Transcription Factor-A11  
CDDO Methyl EsterNrf2 Activator; TriterpenesRTA 402; NSC 713200; TP-155; Bardoxolone Methyl1   
Ceftazidime PentahydrateAntibioticFortaz; Tazicef1   
CelecoxibCOX2 InhibitorCelebrex; Celecoxibum1   
CepharanthineAnti-inflammatory Agent; Antineoplastic Agent 1   
CerivastatinHMG-CoA Reductase InhibitorBaycol; Lipobay1   
Cetirizine DihydrochlorideAntihistamine; GPCR Ligand; Histamine (H1) Receptor Antagonist 1   
Cetrimonium BromideAntiseptic Agent 1   
CetuximabEpidermal Growth Factor Receptor erbB1 InhibitorAnti-EGFR; Erbitux; IMC-C2251 11
CGP 52608RORα Ligand 1   
CH 223191AhR Inhibitor 1   
CHIR-99021 HClGSK-3α/β InhibitorCT990211 1 
ChlorambucilDNA InhibitorAmbochlorin; Chloraminophen; Leukeran1   
ChlorocresolRyanodine Receptor Activator 1   
Chloroquine PhosphateAntimalarial Agent; Quinone Reductase 2 InhibitorAralen; Sanoquin; Reumachlor; Resoquine1   
ChlorothiazideDiuretic; Antihypertensive AgentDiuril; Uroflux; Mechlozid1   
ChlorprothixeneAntipsychotic Agent 1   
ChlorquinaldolAntimicrobial Agent 1   
CholecalciferolVitamin D Receptor (VDR) AgonistOleovitamin D3; Vitamin D3; Calciol1   
CilnidipineCalcium Antagonist; Calcium Channel Blocker 1   
CilostazolPDE3 Inhibitor; Phosphodiesterase ModulatorPletal; OPC-21; OPC-130131   
Cinacalcet HClCalcimimetic Agent; Extracellular Calcium-sensing Receptor AgonistAMG-073 HCl 1   
CinchophenAnalgesic Drug Atophan; Quinophan; Phenaquin1   
CiprofloxacinBacterial DNA Gyrase InhibitorCipro1   
CisplatinDNA Alkylating AgentPlatinol-AQ; Cisplatinum; Neoplatin; CACP; DDP1 1 
CladribineAntineoplastic Agent 1   
ClemastineHistamine (H1) Receptor AntagonistClemastina; Clemastinum; Meclastin1   
CLI-095TLR4 InhibitorTAK2421   
ClimbazoleAntifungal Agent 1   
ClofarabineDNA Inhibitor 1   
ClofazimineAntimycobacterial AgentLamprene1   
CloprostenolProstaglandin F (FP) Receptor Agonist; PGF2α Analog(+)-16-m-chlorophenoxy tetranor Prostaglandin F2α1   
ClosantelAntibacterial Activity Inhibitor 1   
ClozapineAntipsychotic AgentChlorpromazine; Clozaril; Fazaclo; Versacloz1   
Cobalt(II) Chloride HexahydrateInorganic CompoundCobaltous Chloride Hexahydrate1 1 
CobicistatCYP3A InhibitorGS-93501   
Coffee ExtractCoffee Extract 1   
ColchicineMicrotubule DestabilizerColchicina; Colchicinum; Colcrys; Mitigare1 11
Concanamycin AVacuolar Type H+-ATPase (V-ATPase) Inhibitor 1   
Concanavalin A Type VILectin 1   
Copper(II) SulfateGlucose-6-phosphate Dehydrogenase (G6PD) Inhibitor; Paraoxonase Inhibitor 1   
CP 55,940Cannabinoid (CB) Receptor Agonist 1   
CPG 52364TLR7/8/9 Inhibitor 1   
CrizotinibAnticancer Agent; ALK Tyrosine Kinase; HGFR Inhibitor PF-02341066; Xalkori1   
CyanocobalaminVitamin B12 AnalogueCyanocob(III)alamin; Nascobal; Vitamin B121   
CycloheximideProtein Synthesis Inhibitor 1   
Cyclopentyl AdenosineAdenosine A1 Receptor Agonist 1   
Cyclosporin ACalcineurin Inhibitor; Cyclophilin A ModulatorCyA; Cyclosporine; Gengraf; Neoral; Restasis1 1 
Cystamine 2HClCystine Depleter 1   
Cysteamine HClCystine Hydrolytic Enzyme 1   
CytarabineDNA Synthesis Inhibitor 1   
DabrafenibBRAF InhibitorTafinlar; GSK21184361 1 
DactolisibPI3K Inhibitor; mTOR InhibitorNVP-BEZ235; BEZ-2351 11
Dalcetrapib Cholesterylester Transfer Protein (CETP) Inhibitor 1   
Danofloxacin MesylateAntibacterial Agent; Selective Topoisomerase (TOPO) Ligase InhibitorAdvoci; Nofloxacin; CP-76136-271   
Darunavir EthanolateProtease InhibitorPrezista1   
DasatinibMultikinase Inhibitor (Src tyr Kinase, BCR/Abl)BMS-354825; Sprycel111 
Daunorubicin HydrochlorideDNA Inhibitor; DNA Topoisomerase (TOPO) II Alpha InhibitorAcetyladriamycin; Daunomycin; Daunorubicinum; Leukaemomycin C; Rubidomycin1   
DecitabineDNA (cytosine-5)-methyltransferase 1 Inhibitor; DNA (cytosine-5)-methyltransferase 3A Inhibitor; DNA InhibitorAzadc; Dacogen; Dezocitidine1   
DeferasiroxIron Chelating AgentExjade1   
Deferoxamine MesylateIron Chelating AgentDFOA; DFOM; Deferoxamina; Deferoxaminum1   
DenosumabRANKL InhibitorProlia, Xgeva1 1 
DeoxyarbutinTyrosinase Inhibitor 1   
Dequalinium ChlorideAntibacterial Agent 1   
DesloratadineHistamine (H1) Receptor AntagonistAerius; Clarinex; Descarboethoxyloratadine1   
DesonideGlucocorticoid Receptor (GR) Agonist 1   
DexamethasoneGlucocorticoid Receptor (GR) AgonistBaycadron; Decadron; Maxidex; Ozurdex1   
DexlansoprazoleProton Pump Inhibitor 1   
Dibucaine HCLAnesthetic 1   
DienogestSemisynthetic Steroidal ProgestogenProgestin; Visanne1   
DifluprednateDifluorinated Prednisolone Derivative 1   
DigoxigeninHaptenUzarigenin; Digitoxigenin1   
DihydrotestosteroneAR AgonistAnaboleen; Androlone; Stanaprol; Stanolone1   
Dimethyl FumarateNF-kappaB Inhibitor; Nrf2 ActivatorTecifidera; DMF1   
Diminazene AceturateAntiparasitic 1   
DinoprostoneEP AgonistCervidil; Prepidil; Prostin E2; Prostaglandin E21   
Diphenylpyraline HClAntihistamine; Histamine (H1) Receptor Antagonist 1   
DipyridamolePDE InhibitorCardoxin; Cleridium 150; Curantyl; Persantin; Permole1 1 
DisulfiramAldehyde Dehydrogenase InhibitorAntabuse; Tetraethylthiuram Disulfide1   
DL-Mevalonic Acid LactoneHMG-CoA Reductase Inhibitor Mevalonolactone1   
Donepezil HCl Cholinesterase InhibitorAricept; Donepezilum1   
Doramapimodp38 MAPK InhibitorBIRB-79611  
Dorzolamide HCLCarbonic Anhydrase InhibitorMK-5071   
Doxazosin Mesylateα1 Adrenergic Receptor InhibitorDoxazosinum; Doxazosine; Cardura1   
Doxorubicin HydrochlorideDNA Inhibitor; DNA Topoisomerase (TOPO) II Alpha InhibitorAdriamycin; Doxorubicinum; Hydroxydaunorubicin1   
D-PantethineCofactor Precursor 1   
DroperidolD2-like Dopamine Receptor Antagonist; 5-HT2A Receptor Antagonist 1   
DrospirenoneProgesterone Receptor (PR) Agonist 1   
DydrogesteroneProgesterone Receptor (PR) AgonistIsopregnenone; Gynorest; Dydrogesterone1   
DyphyllinePDE Inhibitor; Adenosine Receptor AntagonistDilor1   
EdaravoneAntioxidant MCI-1861   
EGFEGFR Activator 1   
EGFR/ErbB-2/ErbB-4 InhibitorEGFR Inhibitor; HER2, HER4 Inhibitor 1   
Eicosapentaenoic AcidOmega-3 Fatty Acid; Eicosanoid PrecursorEPA; Icosapentaenoic Acid1   
Ellagic acidAntioxidant  1   
EmbelinX-linked Inhibitor of Apoptosis Protein (XIAP) Inhibitor   1 
EMD-1214063cMET Inhibitor 1   
EntinostatHDAC InhibitorMS-2751   
EnzalutamideAndrogen Receptor AntagonistMDV31001   
EpacadostatIDO Inhibitor (IDO1)INCB0243601 11
EpalrestatAldose Reductase Inhibitor 1   
Epothilone BMicrotubule StabilizerEPO 906; EPO906; Patupilone1   
Epothilone DMicrotubule StabilizerDesoxyepothilone B1 1 
Eprazinone 2HClMucolytic Agent746CE; Mucitux; Eftapan; Resplen; Rozuplen; NSC 3179351   
ErlotinibEGFR InhibitorTarceva; CP-358,774; OSI-7741111
ErythromycinBacterial 70S Ribosome InhibitorAbomacetin; Eritromicina; Ilotycin1   
EstradiolER Agonist (α,β)17β-Estradiol1   
EtanerceptTNFα AntagonistEnbrel; TNF-R21   
Ethacridine Lactate MonohydrateDNA Intercalating Antiseptic AgentAcrinol; Rivanol1   
Ethacrynic AcidDiuretic AgentEthacrynic Acid; Edecrin1   
EthanolGABA-A Receptor Agonist; NMDA Receptor Antagonist 1   
EthionamideAntibiotic; Nicotinamide DerivativeTrecator; Amidazine; Thioamide1   
EthosuximideVoltage-gated T-type Calcium Channel BlockerAethosuximide; Atysmal; Etosuximida1   
EthoxzolamideCarbonic Anhydrase InhibitorEthoxyzolamide1   
Ethyl PyruvateAnti-inflammatory AgentPyruvic Acid Ethyl Ester; Ethyl 2-Oxopropanoate1   
EtodolacCOX-2 InhibitorEtodolaco; Etodolacum; Etodolic acid; Lodine1   
EtomidateAnaesthetic AgentEtomidatum; Etomidato; Etomidate; Amidate1   
Etoposide DNA Topoisomerase (TOPO) II InhibitorVP-161   
EverolimusmTOR InhibitorZortress; Certican; Afinitor; Evertor; RAD001111 
ExemestaneSteroidal Aromatase InhibitorAromasin1   
EzetimibeCholesterol Absorption InhibitorZetia; SCH-58235; Ezedoc1   
FamprofazoneNSAIDGewodin; Gewolen1   
FasudilROCK1/2 InhibitorFasudil Hydrochloride; HA-107711  
FCCPUncoupling Agent; Ionophore 1   
FebuxostatXanthine Oxidase InhibitorUloric1   
FenbendazoleAnthelmintic; Microtubule Disruptor; TubulinPanacur1   
Fenoprofen Calcium DihydrateCOX1/2 Inhibitor 1   
Fenspiride HClPDE InhibitorNDR-5998A; NAT-3331   
FICZAhR Agonist 1 1 
FidaxomicinAntibioticDificid; Dificlir; OPT-80; PAR-1011   
FinasterideType II and Type III 5α-reductase InhibitorProscar; Propecia1   
FingolimodSphingosine 1-phosphate (S1P) Receptor ModulatorGilenya; FTY7201   
FlagellinTLR5 Agonist 1   
FlavapreninPhytoestrogen; ER Agonist8-Prenylnaringenin; Hopein; 8-PN 1   
FleroxacinBactericidal Agent; DNA Replication InhibitorFLRX; Quinodis; Megalosin; Megalone 1   
FlubendazoleAnthelminticFlutelmium1   
FludarabineSTAT1 Inhibitor; DNA Synthesis InhibitorOforta; 2-Fluoro-Ara-A; Fludara1   
FludrocortisoneGlucocorticoid Receptor (GR) Agonist; Mineralocorticoid Receptor AgonistFludrocortisonum; Fluohydrocortisone1   
FlumazenilGABA/Benzodiazepine Receptor AntagonistAnexate; Flumazepil; Lanexat1   
FlumethasoneGlucocorticoid Receptor (GR) AgonistU-10974; Flumetasone1   
Flunarizine 2HClCalcium Channel Blocker; Histamine (H1) Receptor AntagonistFlunarizina1   
Fluorometholone AcetateGlucocorticoid Receptor (GR) Agonist 1   
FluorouracilThymidylate Synthase (TS) Inhibitor; Pyrimidine Analog 5-FU; Fluoroplex; 5-Fluracil; Adrucil1 1 
Fluoxetine HClSSRI Symbyax; Sarafem; Prozac; LY-1101401   
Flurbiprofen COX Inhibitor; NSAIDOcufen; FLP; Ansaid1   
Fluticasone PropionateGlucocorticoid Receptor (GR) Agonist; Progesterone Receptor (PR) AgonistFluticason; Fluticasona; Fluticasonum11  
FluvastatinHMG-CoA Reductase InhibitorFluvastatin Sodium; Lescol1   
Fluvoxamine MaleateSSRI Luvox; DU-230001   
fMLPFPR Agonist 1   
Foretinibc-MET and VEGFR2 InhibitorXL880; EXEL-2880; GSK1363089; GSK0891   
ForskolinAdenylyl Cyclase Activator 1   
Fosbretabulin DisodiumMicrotubule Disruptor 1   
Fostamatinib_R406Syk Inhibitor 1   
FSL-1TLR2/6 Agonist 1   
FtorafurChemotherapeutic Agent 1   
FucoidanCaspase-3 Activator 1   
FulvestrantEstrogen Receptor (ER) AntagonistFaslodex1   
FumagillinAngiogenesis Inhibitor; MetAP2 InhibitorFumidil; Fumagillin1   
GaleteroneCYP17A1 Inhibitor 1   
GalunisertibTGFbR1 Kinase InhibitorLY215729911  
GandotinibJAK InhibitorLY27845441 1 
GDC-0834BTK Inhibitor 1   
GDC-0879B-Raf/C-Raf Inhibitor   1 
GefitinibEGFR Inhibitor; erbB1 InhibitorIressa; ZD 18391 1 
GeldanamycinHsp90 Inhibitor 1   
Gemcitabine HClNucleoside Metabolic Inhibitor dFdC; Gemzar; LY-188011; dFdC; dFdCyd1 11
GemfibrozilPPARα AgonistGemfibrozilo; Gemfibrozilum; Lopid1   
GenisteinPhytoestrogenGenisterin; Genisteol; NSC-365861   
GestodeneProgesterone Receptor (PR) Agonist 1   
GF 109203XPKC (c+n) Inhibitor 1   
GKT137831NOX1/NOX4 Inhibitor 11  
GleevecBCR-ABL Tyrosine Kinase Inhibitor; PDGFR Inhibitor; SCFR InhibitorImatinib; Imatinibum11  
GLP-1Glucagon-like Peptide 1 (GLP1) Receptor Agonist 1   
Glyburide Sulfonylurea; Antidiabetic AgentDiabeta1   
GM-CSFCytokine; Immune ModulatorCSF2; Leukine; Sargramostim1   
Go 6983PKC (c+n) Inhibitor 1   
GRPStimulates Gastrin Release; NeuropeptideGastrin-releasing Peptide1   
GSK2801BAZ2 Bromodomain Inhibitor 1   
GSK461364APLK1 Inhibitor 1 1 
GSK690693AKT Inhibitor 1   
GSKJ4Histone Demethylase Inhibitor 1 1 
GW2580cFMS Kinase Inhibitor 1   
GW3965LXRα Agonist 1   
H-1152ROCK2 Inhibitor; Rho/ROCK Inhibitor 11  
Halobetasol PropionateAnti-inflammatory Agent 1   
hCGLuteinizing Hormone/Choriogonadotropin Receptor AgonistHuman Chorionic Gonadotropin1   
Hemicholinium BromideCholine Transporter (ChT) Inhibitor 1   
HGFc-MET/MET/HGF Receptor AgonistHepatocyte Growth Factor1   
HistamineHistamine (H1, H2, H3, H4) Receptor Agonist  1   
Histamine PhosphateHistamine (H1) Receptor Agonist 1   
HKLMTLR2 agonistHeat Killed Listeria monocytogenes1   
Human anti-CD73 IgG1Anti-CD73 Monoclonal AntibodyMEDI9447  1 
Human IgG1IgG1 Control Antibody   1 
Human IgG1 mAb R347 Isotype ControlIgG1 Control Antibody   1 
Human IgG1kIgG1 Control Antibody 1   
Human IgG4 IsotypeIgG4 Control Antibody 1 1 
Human γ-GlobulinAntibody 1   
HydrochlorothiazideDiuretic; Antihypertensive AgentEsidrix; Urozide; Microzide; HCTZ1   
HydrocortisoneGlucocorticoid Receptor (GR) Agonist17-Hydroxycorticosterone1   
HydroxyfasudilROCK1/2 Inhibitor 1   
HydroxyureaAntineoplastic Agent; Ribonucleotide Reductase InhibitorHydroxycarbamide; Hydrea; Litalir; Droxia1   
Hydroxyzine 2HClHistamine (H1) Receptor Antagonist 1   
Hygromycin BAntibiotic 1   
I-BETBET Inhibitor (BRD2, 3, 4)GSK525762A1 1 
I-BET-151BET InhibitorGSK1210151A111 
IbrutinibBTK InhibitorPCI-32765; Imbruvica1 11
IbudilastPDE4 InhibitorAV-411; Eyevinal; Ibudilastum; Ketas1   
IbuprofenCOX Inhibitor; NSAID 1   
Ibuprofen LysineCOX Inhibitor; NSAIDNeoProfen1   
IbutamorenGhrelin Receptor AgonistMK-06771   
IC-87114PI3Kd Inhibitor 1 1 
I-CBP112CBP/p300 Bromodomain InhibitorSGC-I-CBP1121   
ICG-001β-catenin/CBP Inhibitor 111 
ICI 63197PDE4 Inhibitor 1   
IdebenoneSynthetic Coenzyme Q10 (CoQ10) AnalogCatena; Raxone; Sovrima1   
IdelalisibPI3Kδ InhibitorCAL-101; Zydelig; GS-1101 1 1 
IDO-IN-2IDO Inhibitor (IDO1) 1 11
IFNα 2aIFNα Receptor Agonist 1   
IFNα 2bIFNα Receptor Agonist 1   
IFNβ 1bIFNβ Receptor Agonist 1   
IFNγIFNγ Receptor AgonistActimmune; Interferon gamma-1b1 1 
IKK 16IKK2 Inhibitor 1   
IKK-2 Inhibitor IVIKKβ (IKK-2) Inhibitor 1   
IL-10IL-10 Receptor Agonist 1 1 
IL-12IL-12 Receptor Agonist 1   
IL-13IL-13 Receptor Agonist 1   
IL-17AIL-17 Receptor Agonist 1   
IL-17A/FIL-17 Receptor Agonist 1   
IL-17FIL-17 Receptor Agonist 1   
IL-1R AntagonistIL-1 Receptor Antagonist 1   
IL-1βIL-1β Receptor Agonist 1   
IL-2IL-2 Receptor AgonistAldesleukin; Proleukin1  1
IL-22IL-22 Receptor Agonist 1   
IL-27IL-27 Receptor Agonist 1   
IL-29IL-29 Receptor Agonist 1   
IL-33IL-33 Receptor Agonist 1   
IL-35IL-35 Receptor Agonist 1   
IL-4IL-4 Receptor Agonist 1   
IL-6 RαImmunomodulating AgentCD126 (Cluster of Differentiation 126)1   
IL-8CXCR1/2 Agonist 1   
IloperidoneAntipsychotic AgentFanapt1   
IloprostEP1 Agonist; Prostanoid IP Receptor AgonistVentavis1   
ImatinibBCR-ABL Tyrosine Kinase Inhibitor; PDGFR Inhibitor; SCFR InhibitorGleevec1   
IndomethacinCOX1/2 InhibitorAconip; Indocin; Indometacina; Indometacinum1   
IndoximodIDO Inhibitor (IDO2)NLG-81891 11
InfliximabTNFα AntagonistRemicade; Biosimilars (Inflectra, Remsima, Infimab)11  
Insulin AspartInsulin Receptor AgonistNovolog 1   
Insulin GlargineInsulin Receptor AgonistLantus1   
Insulin LisproInsulin Receptor AgonistHumalog; Insulin Lispro Recombinant1   
IOX 1Histone Demethylase JMJD Inhibitor 1   
IpilimumabAnti-CTLA-4 Monoclonal Antibody; CTLA-4 InhibitorYervoy, MDX-010, MDX-101; MDX-CTLA-4; MOAB-CTLA-41 1 
IRAK1/4 Inhibitor IIRAK 1/4 InhibitorIRAK-1/4 Inhibitor1   
IrinotecanDNA Topoisomerase (TOPO) I InhibitorCamptosar; Campto; CPT-11; Camptothecin-11; Irinotecan1 1 
IrsogladineM1 Muscarininc Receptor 1   
Isoetharine Mesylateβ2 Adrenergic Receptor AgonistIsoetarine Mesilate1   
IsoniazidEnoyl-[acyl-carrier-protein] Reductase InhibitorIsonicotinic acid hydrazide; Isonicotinylhydrazine1   
IsotretinoinRAR/RXR Agonist13-cis-Retinoic acid; 13-RA; Accutane1   
ItraconazoleCytochrome P450 51 InhibitorSporanox11  
IvacaftorCFTR PotentiatorVX-770; Kalydeco11  
JAK Inhibitor IJAK InhibitorJAK Inhibitor 11   
JNJ 10397049Orexin Receptor Type 2 (OX2) Antagonist 1   
JNK Inhibitor VIIIJNK Inhibitor 1   
JQ1BET Inhibitor 1 1 
KetoconazoleCytochrome P450 51 Inhibitor 1   
KetoprofenCOX Inhibitor; NSAIDActron; RP-19583; Oruvail; Orudis; Nexcede1   
Ketotifen Fumarate Histamine (H1) Receptor AntagonistKetotifeno; Ketotifenum; Zaditor1   
Ki16425LPA1 Receptor Antagonist; LPA3 Receptor Antagonist 1   
Kisspeptin-10/MetastatinKISS1 Agonist; GPR54 Agonist 1   
KN93CAMKII Inhibitor 11  
KNK437Hsp Modulator; Hsp Inhibitor (Hsp 72, 73, 90, 105, 27, 40) 1   
L-744832Farnesyltransferase Inhibitor 1   
LansoprazoleProton Pump InhibitorA-65006; Prevacid; AG-17491   
LapatinibTyrosine Kinase Inhibitor (ERBB1, ERBB2)GW 572016; Tykerb1   
L-Arginine HClVasodilator; Source of NO 1   
LeflunomideDihydroorotate Dehydrogenase (DHODH) InhibitorArava; Leflunomida; Leflunomidum1   
LenalidomideImmunomodulating Agent; Antineoplastic AgentRevlimid1 1 
LetrozoleCytochrome P450 19A1 Inhibitor 1   
Levamisole HydrochlorideNicotinic Acetylcholine Receptor Alpha Subunit AgonistErgamisol1   
LFM-A13BTK Inhibitor 1   
LinezolidAntibiotic AgentZyvox1   
LinsitinibIGF-1R InhibitorOSI-9061   
Liothyronine SodiumThyroid Hormone Receptor Agonist 1   
LiraglutideGlucagon-like Peptide 1 (GLP-1) Receptor AgonistVictoza; Liraglutidum; Saxenda1   
LonidamineHexokinase Inhibitor; Glycolysis Inhibitor 1   
LopinavirAntiretroviral Agent; Protease Inhibitor ABT-3781   
LoratadineHistamine (H1) Receptor Inhibitor 1   
LornoxicamCOX Inhibitor; NSAID; Analgesic Agent; Anti-inflammatory AgentXefo; Chlortenoxicam1   
Loteprednol EtabonateGlucocorticoid Receptor (GR) Agonist 1   
LovastatinHMG-CoA Reductase InhibitorAltoprev; Mevacor; Mevinolin1   
Loxapine SuccinateAntipsychotic AgentCL-71563; Loxitane1   
LP99BRD7/9 Inhibitor 1   
LPSTLR4 Agonist 1   
LumacaftorCFTR ModulatorVX-8091   
LuminespibHsp90 InhibitorNVP-AUY-9221   
LY294002CK2 Inhibitor; PI3K Inhibitor 1 1 
LY364947TGFβ/Smad Inhibitor 1   
M344HDAC Inhibitor 1   
MacitentanEndothelin Receptor Antagonist (ET-A, ET-B)Opsumit1   
ManidipineCalcium Channel Blocker; Antihypertensive AgentManyper1   
Meclocycline SulfosalicylateAntibiotic 1   
MedrysoneAnti-inflammatory Corticoidsteroid (Ocular)Hydroxymesterone; HMS1   
Mefenamic AcidCOX Inhibitor; NSAIDCI-473; Ponstel; CN 35355; CI-4731   
Megestrol AcetateProgesterone Receptor (PR) AgonistVolidan; Ovarid; Ovaban; Niagestin; BDH-12981   
MenadionePhosphatase Inhibitor; Mitochondrial DNA Polymerase γ (pol γ) InhibitorVitamin K31   
Mepivacaine HClSodium Channel Alpha Subunit Blocker; Topical Anesthetic Agent 1   
MeprednisoneGlucocorticoid Receptor (GR) Agonist; Methylated Derivative of PrednisoneBetapar1   
MequinolDepigmentation Agent 1   
MercaptopurinePurine Nucleotide Synthesis Inhibitor 1   
Mesalazine15-Lipoxygenase Inhibitor; COX1/2 Inhibitor; IKK1/2 InhibitorApriso; Asacol; Canasa; Delzicol; 5-ASA; Mezavant1   
Mesoridazine BesylateAntipsychotic Agent; D2 Receptor Antagonist; 5-HT2A Receptor AntagonistMesoridazine Benzenesulfonate1   
Metaproterenol Sulfateβ2-Adrenergic Receptor AgonistAlupent1   
Metformin HydrochlorideAMPK Activator; Mitochondrial Complex I (NADH dehydrogenase) InhibitorHaurymellin; Metformine Pamoate; Metforminum1   
Methapyrilene HClHistamine (H1) Receptor AntagonistMethapyrilene1   
MethazolamideCarbonic Anhydrase InhibitorNeptazane; Methazolamide1   
MethocarbamolMuscle RelaxerDelaxin; Robaxin; Neuraxin; Miolaxin; Forbaxin1   
MethotrexateDihydrofolate Reductase (DHFR) InhibitorAbitrexate; Amethopterin; Emtexate; Ledertrexate; MTX; Metoject1 11
MethyclothiazideDiuretic; Antihypertensive Agent 1   
MethyldopaAdrenergic Receptor α2 AgonistAldomet1   
MevastatinHMG-CoA Reductase InhibitorCompactin1   
MianserinHistamine (H1) Receptor Antagonist; 5-HT Serotonin Receptor Antagonist 1   
MifamurtideNOD2 Activator 1   
MizolastineHistamine (H1) Receptor InhibitorMizollen1   
MizoribineImidazole Nucleoside; Immuno-suppressant; DNA Synthesis InhibitorBredinin1   
MK-2206AKT Inhibitor 1   
MLN8054Aurora Kinase Inhibitor 1   
Mometasone FuroateGlucocorticoid Receptor (GR) Agonist 1   
Monensin SodiumNa+ Ionophore 1   
MonobenzoneDepigmentation AgentBenoquin1   
MontelukastCysLT1 Receptor Antagonist; GPCR Ligand 1   
Mosapride CitrateMosapride Citrate 1   
MotilinMotilin Receptor Agonist 1   
Moxifloxacin HClAntibacterial Agent 1   
MRT67307IKKe and TBK-1 Inhibitor 11  
Mycophenolate Mofetil Inosine Monophosphate Dehydrogenase I/II InhibitorCellCept1   
Mycophenolic AcidIMPDH Inhibitor 1   
MyxothiazolCytochrome c Reductase Inhibitor; Mitochondrial Inhibitor 1   
N-Acetyl CysteineAntioxidant 11  
Nafcillin Sodium MonohydrateAntibiotic6-(2-Ethoxy-1-naphthamido)penicillin1   
Nalmefene HClOpioid Receptor Antagonist Nalmetrene1   
NaproxenCOX Inhibitor; NSAIDAnaprox; Naprelan; Naprolag; Naprosyn1   
NDP-α-MSHMelanocortin Receptor Agonist 1   
Nebivololβ1-Adrenergic Receptor InhibitorBystolic1   
Nefazodone5-HT2A AntagonistNefazodone Hydrochloride; Nefazodonum1   
Nefopam HClNon-opioid Analgesic Drug Acupan; Silentan; Nefadol; Ajan1   
NelarabineDNA InhibitorArranon1   
Neomycin SulfateBacterial 70S Ribosome Inhibitor 1   
Neostigmine BromideAcetylcholinesterase InhibitorProstigmin1   
Neuromedin BNMBR Agonist 1   
NI-57BRPF Bromodomain Inhibitor 1   
NialamideMonoamine Oxidase Inhibitor (MAOI)Niamid; Niamide; Nuredal; Surgex1   
NifuroxazideSTAT InhibitorSJ000287313; RC-271091   
NintedanibVEGFR, FGFR, PDGFR Kinase InhibitorOfev; Vargatef; BIBF 112011  
NithiamideAntiprotozoan AgentAcinitrazole; Aminitrozole1   
NitrofurazoneAnti-infective AgentNitrofural1   
NitroprussideVasodilator; Source of NONipride; Nitroferricyanide; Nitropress1   
NivolumabAnti-PD-1 AntibodyOpdivo1 1 
NLG919IDO Inhibitor 1 1 
Nodinitib-1NOD1 Inhibitor 1   
Non_StimNo stimuli added to any system 1   
NorethindroneProgesterone Receptor (PR) AgonistNorethisterone; Utovlan1   
Nortriptyline HydrochlorideNorepinephrine Transporter Inhibitor; SERT Antagonist; Serotonin Transporter InhibitorAteben; Avantyl; Noritren; Psychostyl; Sensaval1   
Nutlin-3MDM2 Antagonist   1 
NVP-TAE684ALK Inhibitor; Kinase Modulator 1   
OdanacatibCathepsin K Inhibitor 11  
ODN2006TLR9 Agonist 1   
ODN2395TLR9 Agonist 1   
OEAPPARα AgonistOleoylethanolamine1   
OfloxacinBacterial DNA gyrase InhibitorFloxin1   
OlaparibPARP InhibitorAZD22811   
Oligomycin AF0/F1 ATPase Inhibitor; Mitochondrial Inhibitor 1 1 
OmeprazoleProton Pump InhibitorAntra; Prilosec; H-168/681   
OmipalisibPI3K Inhibitor; mTOR InhibitorGSK-21264581111
Oncostatin MLIFRα; OSMR Agonist 1   
Ondansetron5-HT3A Receptor AntagonistZuplenz; Zofran1   
OrlistatLipase InhibitorAlli, Xenical1   
OTX015BET Inhibitor 1   
OxaliplatinAntineoplastic Agent; DNA Synthesis InhibitorEloxatin; L-OHP1 1 
OxaprozinCOX Inhibitor; NSAID; Anti-inflammatory Agent 1   
OxethazaineLocal Anaesthetic 1   
OxibendazolePolymerase Inhibitor 1   
Oxybuprocaine HClSodium Channel Alpha Subunit Blocker; Topical Anesthetic Agent 1   
OzagrelAntiplatelet Agent; Thromboxane A2 Synthesis (TXAS) InhibitorOKY-0461   
P 22077 USP7/USP47 Inhibitor; DUB Inhibitor 1   
P7C3NAMPT Activator; Proneurogenic; Neuroprotective 1   
Paclitaxel Microtubule StabilizerTaxol; Anzatax; Asotax; Bristaxol; Praxel1 11
PalbociclibCDK4/6 InhibitorIbrance1   
PaliperidoneD2 Receptor Antagonist; 5-HT2A Receptor AntagonistInvega1   
Palonosetron HCl5-HT3A Receptor Antagonist 1   
Pam3CSK4TLR1 Agonist 1   
Pamoic Acid DisodiumGPR35 Agonist 1   
PanitumumabEGFR Inhibitor; erbB1 InhibitorABX-EGF; Vectibix1   
PanobinostatHDAC Inhibitor 1   
Paromomycin SulfateBacterial 70S Ribosome Inhibitor 1   
Paroxetine HClSERT Antagonist; Serotonin Transporter 1   
PazopanibMultikinase Inhibitor (c-KIT, FGFR, PDGFR, VEGFR) GW 78603; GW786034; Pazopanibum; Votrient1   
PBI - 4050Antifibrotic Agent 11  
PD098059MEK Inhibitor 1   
PD123319AT2 Antagonist 1   
PD184352MEK InhibitorCI-10401   
PDGF-BBPDGFRβ Activator 1   
PembrolizumabAnti-PD-1 AntibodyKeytruda1 11
Pemetrexed DisodiumDihydrofolate Reductase (DHFR) Inhibitor; GAR Transformylase Inhibitor; Thymidylate Synthase Inhibitor 1   
PenciclovirGuanosine Analogue; Antiviral AgentDenavir1   
Pergolide MesylateDopamine Receptor Agonist 1   
Perindopril ErbumineAngiotensin-converting Enzyme InhibitorAceon1   
PertuzumabReceptor Protein-tyrosine Kinase erbB-2 Inhibitor2C4 Antibody;Omnitarg; Perjeta; rhuMAb-2C41   
PF-04217903c-Met Inhibitor 1   
PFI-1BET Inhibitor (BRD2/4) PF-6405761; PF-064057611 1 
PFI-3SMARCA2/4 Inhibitor; Polybromo 1 (PBRM1) Inhibitor 1 1 
PFI-4BRPF1 Bromodomain Inhibitor 1   
PHA-408IKK2 Inhibitor 1   
Phenazopyridine HClSodium Channel Alpha Subunit Blocker; Topical Anesthetic Agent 1   
Pheniramine MaleateHistamine (H1) Receptor Antagonist 1   
PhenylbutazoneCOX Inhibitor; NSAIDButazolidin, Butatron1   
Phenylephrineα1-Adrenergic Receptor AgonistCyclomydril; Mydfrin1   
Phorbol 12-myristate 13-acetatePKC ActivatorPMA1   
PiclamilastPDE4 Inhibitor 1   
PicropodophyllinMicrotubule Disruptor 1   
PictilisibPI3Kα/δ InhibitorGDC-09411 1 
PictilisibPI3K InhibitorGDC-0941 11 
PilaralisibPI3K InhibitorXL1471   
PimasertibMEK InhibitorAS7030261   
PimobendanPDE3 InhibitorVetmedin1   
PioglitazonePPARγ AgonistActos1   
PirfenidoneAntifibrotic AgentPirespa; Pirfenex; Esbriet; Etuary; KitosCell11  
PironetinMicrotubule Disruptor 1   
Pizotifen malate5-HT Receptor Anatagonist 1   
PlerixaforCXCR4 InhibitorAMD 31001   
PLX4720BRAF Inhibitor 1   
PNU 74654Wnt/β-catenin Pathway Inhibitor 1   
Poly(I:C)HMWTLR3 Agonist 1   
PomalidomideTNFα Inhibitor 1   
PonatinibBCR-ABL InhibitorAP 24534; AP24534; Iclusig1   
PosaconazoleCYP51 Inhibitor 1   
PP 242mTOR Inhibitor 1   
PP1Src Family Inhibitor 1   
PracinostatHDAC InhibitorSB9391   
PralatrexateDHFR InhibitorFolotyn1   
PramoxineTopical Anaesthetic Agent; Antipuritic AgentTronothane; Tronolane; Pramocaine1   
PraziquantelAntihelmintic AgentBiltricide; EMBAY-8440; Droncit; Cestocur; Cesol1   
PrednisoloneGlucocorticoid Receptor (GR) AgonistHydroretrocortine; Metacortandralone; Omnipred; Orapred; Pediapred1   
PrednisoneGlucocorticoid Receptor (GR) AgonistRayos; Adasone; Cortan; Sterapred1   
PrilocaineAnaesthetic Agent 1   
Primaquine DiphosphateQuinone Reductase 2 Inhibitor 1   
ProbenecidUricosuric AgentBenemid; Probalan1   
Procarbazine HClDNA InhibitorMatulane1   
ProgesteroneProgesterone Receptor (PR) AgonistPrometrium1   
Prostaglandin D2DP Agonist 1   
PrRP-31hGR3/GPR10 AgonistProlactin Releasing Peptide-311   
PRT-062607SYK Inhibitor 1   
Pyridostigmine BromideCholinesterase InhibitorMestinon1   
PyrithioxinNeurotropic Agent 1   
Quinacrine Dihydrochloride DihydratePLA2 (phophoslipase A2) InhibitorAtabrine hydrochloride1   
QuizartinibFLT3 InhibitorAC2201   
R(-)rolipramPDE4 Inhibitor 1   
R428AXL Inhibitor 1   
RadicicolHSP90 InhibitorMonorden11  
RaltitrexedDihydrofolate Reductase Inhibitor; Thymidylate Synthase InhibitorRaltitrexed; Tomudex; ZD16941   
Reboxetine MesylateNoradrenalin Uptake Inhibitor 1   
Refametinib MEK1/2 InhibitorRDEA-1191   
RegorafenibMultikinase Inhibitor; VEGFR2-TIE2 Tyrosine Kinase InhibitorBAY 73-4506; Stivarga1   
RepaglinideAntidiabetic Agent; Meglitinide 1   
ResiquimodTLR7/8 Agonist 1   
ResveratrolCYP1A1 Inhibitor 1   
RetapamulinAntibiotic; Protein Synthesis InhibitorAltabax; Altargo1   
RetinolVitamin A MetaboliteAquasol A1   
rhM-CSF M-CSF Receptor AgonistRecombinant Human Macrophage-colony Stimulating Factor; CSF-1 1   
RimonabantCB1 Inverse Agonist; GPCR LigandSR1417161   
Risedronate SodiumBiphosphonate; Bone Density Conservation AgentActonel; Atelvia; Benet1   
RitonavirHIV Type 1 Protease InhibitorNorvir1   
RN486BTK Inhibitor 1   
Ro 106-9920Ubiquitin Ligase Inhibitor 1   
Ro 20-1724PDE4 Inhibitor 1   
Ro 320-1195p38 MAPK Inhibitor 1   
Ro 32-0432PKC (c+n) Inhibitor 1   
RO5126766BRAF Inhibitor; MEK Inhibitor 1   
RofecoxibCOX2 InhibitorVioxx1   
RoflumilastPDE4 InhibitorDaxas; Daliresp; ROF; Roflumilastum 11  
Roflumilast N-OxidePDE4 Inhibitor 11  
Ropivacaine HClLocal Anaesthetic AgentNaropin1   
RosiglitazonePPARγ AgonistAvandia; TZD111 
RosuvastatinHMG-CoA Reductase InhibitorCrestor; Rosuvastatin1   
RotenoneMitochondrial Inhibitor; NADH Dehydrogenase Inhibitor 1   
RuxolitinibJAK InhibitorINCB018424; Jakafi1   
R-α-MethylhistamineHistamine (H3) Receptor Agonist 1   
S31-201STAT3 Inhibitor 1   
Salbutamol Sulfateβ2 Adrenergic Receptor AgonistAlbuterol1   
SalicylanilideAntimycobacterial Agent2-Hydroxybenzanilide; N-Phenylsalicylamide 1   
Salinomycin MonosodiumP-glycoprotein 1 Inhibitor 1   
Salmeterol Xinafoateβ2-Adrenergic Receptor Agonist 11  
SaracatinibABL InhibitorAZD053011  
Sarafloxacin HClAntibacterial Agent; Bacterial Topoisomerase Inhibitor 1   
SaxagliptinDPP-4 Inhibitor; Anti-diabetic AgentOnglyza1   
SB203580p38 MAPK Inhibitor 1   
SB431542TGFβR1 Kinase Inhibitor; ALK Inhibitor 111 
SB525334TGFβR1 Kinase Inhibitor; ALK InhibitorTGFβ RI Kinase Inhibitor VIII1   
ScriptaidHDAC Inhibitor 1   
SelumetinibMEK1/MEK2 InhibitorAZD6244; ARRY-1428861 1 
Semagacestatγ-Secretase InhibitorLY4501391   
Sepantronium BromideSurvivin InhibitorYM1551   
Sertraline HClSSRI 1   
SGC-CBP30CREBBP/EP300 Bromodomain Inhibitor 1 1 
SGI-1776PIM1/2/3 Inhibitor 1   
Shaoguamycin BMitochondrial Inhibitor; NADH Dehydrogenase Inhibitor 1   
Sildenafil CitratePDE5 InhibitorViagra11  
SimvastatinHMG CoA Reductase InhibitorZocor11  
Sirolimus mTOR Inhibitor; FK506-binding Protein 1A InhibitorRapamycin; Rapamune; AY 22989; SILA 9268A; WY-0902171111
SL 327MEK Inhibitor 1   
SLPIPeptidase Inhibitor ProteinALP; MPI; ALK1; BLPI; HUSI; WAP4; WFDC4; HUSI-I  1 
Sodium HydroxideInorganic CompoundLye; Caustic Soda; Sodium Hydrate1   
Somatostatin 28Somatostatin Receptor Agonist 1   
Sorafenib TosylateMultikinase Inhibitor (RAF/VEGFR-2/PDGFRβ)Nexavar; BAY 43-9006; Tosylate Salt1 1 
SotrastaurinPKC InhibitorAEB0711   
SP600125JNK Inhibitor 1   
SPD-304TNFα Inhibitor 1   
SpebrutinibBTK InhibitorAVL-292; CC-2921 1 
Sphingosine-1-phosphateS1P1 Agonist 1   
SpiramycinAntibiotic Agent; Antiparasitic Agent 1   
SpironolactoneAldosterone AntagonistAldactone1   
SR2211RORγ Inhibitor 1   
SRT2104SIRT1 Activator 1   
ssRNA40TLR8 Agonist 1   
SU6656Src Family Inhibitor 1   
SuccinateChemical IntermediateSuccinic acid1   
SulfasalazineAnti-inflammatory AgentAzulfidine1   
SulforaphanePhytochemical; Antioxidant; Detoxifying Enzyme Inducer 1   
Sunitinib MalateMultikinase Inhibitor (VEGFR2, CSF-1R, PDGFR, SCFR, FLT3, RET)Sutent; SU11248; SU0112481 1 
Synta66CRAC Channel InhibitorCLC0015311   
T0901317LXR/FXR Agonist; LXRα Agonist 1   
Tacrolimus Calcineurin Inhibitor; FK506-binding Protein 1A InhibitorFK-5061   
TadalafilPDE5 InhibitorCialis1   
TanespimycinHSP90 Inhibitor17-AAG 1 1 
Taurolithocholic AcidG Protein-coupled Bile Acid Receptor 1 Agonist 1   
TeicoplaninAntibioticTargocid; Ticosin 1   
TelbivudineAntiviral Agent; Thymidine β-L-nucleoside AnalogueSebivo, Tyzeka1   
TelmisartanType-1 Angiotensin II Receptor (AT2R) AntagonistBIBR 277; Micardis1   
TemsirolimusFK506-binding Protein 1A (FKBP1A) Inhibitor; mTOR InhibitorCCI 779; Torisel1   
Tenidap5-Lipoxygenase Inhibitor; COX1/2 Inhibitor 1   
TerbinafineAntifungal AgentLamisil, Terbinex1   
TeriflunomidePyrimidine Synthesis Inhibitor; DHODH InhibitorA7717261   
Tetracycline HClBacterial 70S Ribosome Inhibitor 1   
TG-101348JAK InhibitorSAR3025031 1 
TGFβTGFβRI/II Agonist 1   
TGFβ2TGFRI, TGFRII Agonist 1   
TGFβ3TGFRI, TGFRII Agonist 1   
TGFβRI Kinase InhibitorTGFβR1 Kinase Inhibitor 1   
TGX-221PI3Kβ Inhibitor 1   
ThapsigarginSR Ca++ ATPase Inhibitor; SERCA Inhibitor 11  
ThioguanineDNA Inhibitor; Inosine-5'-monophosphate Dehydrogenase (IMPDH) Inhibitor 1   
ThiostreptonOligopeptide AntibioticAlaninamide; Bryamycin; Thiactin1   
Tianeptine SodiumAntidepressant 1   
TigecyclineAntibiotic 1   
Tilorone DihydrochlorideAntiviral; IFN Type I Inducer 1 11
Tin(II) ChlorideChemical CompoundStannous Chloride; Tin Salt; Tin Protochloride1   
TioxoloneCarbonic Anhydrase InhibitorThioxolone1   
TiratricolThyroid Hormone Analogue; Physiologic Thyroid Hormone TRIAC; Triiodothyroacetic Acid1   
TMP-153Acetyl-coA Cholesterol Acyltransferase (ACAT) Inhibitor 1   
TocilizumabInterleukin-6 Receptorα Subunit InhibitorAtlizumab; MRA; RoActemra; Actemra1   
TofacitinibJAK InhibitorTasocitinib; Tofacitinibum; Xeljanz1   
Topotecan HClTopoisomerase (TOPO) I InhibitorHycamtin, Hycamptamine, SKF S-104864-A1 1 
TorcetrapibCETP Inhibitor 1   
Torin-1mTOR Inhibitor 1   
Torin-2mTOR Inhibitor 1   
TorsemideSodium-(potassium)-chloride Cotransporter 2 InhibitorDemadex1   
TozadenantAdenosine A2a Receptor Antagonist 1 11
TrametinibMEK InhibitorMekinist; GSK1120212 1 1 
Tranexamic acidPlasminogen InhibitorTransamin1   
TranilastAntiallergic AgentRizaben11  
trans-TriprolidineHistamine (H1) Receptor Antagonist 1   
TrastuzumabAnti-HER2/neu Monoclonal AntibodyHerclon; Herceptin; Biosimilars (PF-05280014, ABP 980 and SB3)  1 
TretinoinRAR/RXR Receptor AgonistAberela1   
Triamcinolone AcetonideGlucocorticoid Receptor (GR) Agonist 1   
Trichostatin AHDAC Inhibitor 1   
Trilostane3β-hydroxysteroid Dehydrogenase Inhibitor 1   
TropineAtropine Precursor 3-Tropanol 1   
Tubastatin AHDAC Inhibitor 1   
TunicamycinAntibiotic 1   
TWEAKTWEAKR (Fibroblast growth factor-inducible 14 (Fn14)) Agonist; CytokineTNFSF12; TNF-like Weak Inducer; Human TWEAK1   
Tyr[SO3H]27)-CCK8Stimulates Pancreatic SecretionC-Terminal Octapeptide of Cholecystokinin (CCK); Sincalide; Kinevac 1   
Tyrphostin AG 1296PDGFRα/β Inhibitor 1   
U0126MEK Inhibitor 1   
U-75302Leukotriene B4 (LTB4) Receptor Antagonist 1   
UK 14, 304α2-Adrenergic Receptor Agonist 1   
UNC0642G9a and GLP Inhibitor 1   
Urolithin AMicroflora Metabolite 1   
Ursodeoxycholic AcidBile Acid Receptor FXR Agonist 1   
Ursolic AcidCosmetic AdditiveUrson; Prunol; Malol1   
VadimezanDT-DiaphoraseDMXAA1 1 
ValdecoxibNSAID; COX-2 InhibitorBextra1   
ValinomycinAntibiotic 1   
Valnemulin HClPleuromutilin Antibiotic  1   
Valproic AcidHDAC Inhibitor; GABA Transaminase InhibitorDepakene; Stavzor; Sodium Divalproex11  
VandetanibVEGFR2/EGFR InhibitorCaprelsa; AZD6474; ZD64741 1 
VardenafilPDE5 InhibitorLevitra; Staxyn; Vardenafil; Vardenafilum1   
VasopressinVasopressin Receptor AgonistADH; AVP; Antidiuretic Hormone; Argipressin1   
Vegetable Extract HI_V19Vegetable Extract 1   
VemurafenibBRAF InhibitorBRAF(V600E) Kinase Inhibitor RO5185426; PLX4032; Zelboraf1 1 
VenetoclaxBcl-2 InhibitorABT-199; GDC-01991   
VerapamilL-type Ca++ Channel AntagonistCP-165331; Calan; Iproveratril; Isoptin; Verelan1   
VinblastineMicrotubule DisruptorVincaleukoblastine; VLB1   
Vincristine SulfateMicrotubule DisruptorLeurocristine; Vincristin; Vincristina1   
VinorelbineMicrotubule InhibitorNavelbine1   
VinpocetineVoltage Sensitive Sodium Channel Inhibitor; PDE InhibitorCavinton1   
VismodegibHedgehog Pathway InhibitorErivedge; GDC-044911 1
VorinostatHDAC Inhibitor (HDAC1, HDAC2, HDAC3, HDAC6)Zolinza; Suberoylanilide Hydroxamic Acid (SAHA)1 1 
VoxtalisibPI3K Inhibitor; mTOR InhibitorXL7651   
VX-702p38 MAPK Inhibitor 1   
VX-745p38α MAPK Inhibitor 1 1 
WKYMVm-NH2Formyl Peptide Receptor (FPR1, FPR2) Agonist 1   
WortmanninPI3K InhibitorKY 124201   
WS6EBP1/IKK Inhibitor 1   
XAV-939Tankyrase (TNKS) Inhibitor 1111
XL019JAK Inhibitor 1   
Y-27632ROCK1/2 Inhibitor 11  
YM201636PIKfyve InhibitorYM-2016361   
ZaprinastPDE Inhibitor (PDE9, PDE6, PDE5) 1   
ZidovudineReverse Transcriptase InhibitorAZT; Retrovir; Azidothymidine1   
Zileuton5-Lipoxygenase InhibitorArachidonate 5-lipoxygenase Inhibitor; Zyflo1   
Zinc ChlorideChemical Compound 1   
Ziprasidone5-HT Receptor Anatagonist 1   
ZM449829JAK Inhibitor 1   
αAmanitinRNA Polymerase II Inhibitor 1