my cart
log-in
Search for:
Search for:
applications / products
Applications
Drug Discovery & Development
Cell Banks for Bioassays
Potency & QC Lot Release
Detect Neutralizing Abs
Cytotoxicity Assays
Target Engagement
Translocation Assays
Targeted Protein Degradation
Signaling Pathway Reporters
Pharmacotrafficking Assays
Do-It-Yourself Assays
Therapeutic/Disease Area
Custom Development Capabilities
Products
Cells & Cell Lines
Assay Ready Kits
Bioassay Kits
eXpress Kits
Frozen Cells
Membrane Preps
Proteins & Kinases
Cell Culture Reagents
Detection Reagents
Biochemical Assays
Control Ligands & Inhibitors
targets
A-Z List of Target List
GPCRs
Kinases
Checkpoint Receptors
Ion Channels
Cytokines & Interleukins
Signaling Pathways
Nuclear Proteins
Epigenetics Proteins
technologies / platforms
Enzyme Fragment Complementation
Human Primary Cell Screening
Competition Binding Platform
tools / resources
Document Resource Library
Flyers & Brochure
User Manuals & Protocols
White Papers & Applications
Scientific Posters
Presentations
Webinars
Knowledge-Based Videos
Blogs
Scientific FAQs
Publications & References
CRO/CDMO Certification
Reagent Calculators
Instrument Compatibility
services
Contact Us
Customer & Technical Support
Submit an Order
Technical Resources
Literature & Email Signup
Legal & Policies
Locations
Distributors
Procurement Partners
about us
Company
Contact Us
Careers
Announcements
Events
Targets
/
EPHA2
Contact a Specialist
Services
Drug Discovery & Development Services
Custom Assay Development Services
KINOME
scan
®
EPHA2
Request a Quote
Explore Our Panels & Assays
Related Group Members:
TK
Available Technology Platforms:
KINOMEscan
Panel:
KdMAX
;
KdELECT
;
scanEDGE
;
scanMAX
;
scanELECT
;
scanTK
;
Specifications
Target/Description
EPH receptor A2
Group
TK
Kinase Construct
Partial Length
Accession Number
NP_004422.2
Species
Human
Kinase Form
Wild Type
Expression System
Bacterial
Amino Acid Start/Stop
T593/V891
How it works
Assay Information
Average Z' Panel
0.79
Reference Inhibitor Information
(all values in nM)
Compound
K
D
Dasatinib
0.85
AST-487
160
ZD-6474
1100