KINOMEscan® CDK12

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Panel:

Target/Description
cyclin-dependent kinase 12 isoform 2 [Homo sapiens]
Group
CMGC
Kinase Construct
Partial Length
Accession Number
NP_055898.1
Species
Human
Kinase Form
Wild Type
Expression System
Mammalian
Amino Acid Start/Stop
P697/E1077

Reference Inhibitor Information (all values in nM)

Compound
KD
BMS-357075
0.72
AT-9283
120
BMS-387032
30