Biological Information

Background Information:

PFI-3 is a synthetic inhibitor of the SMARCA4 and PB1(5) bromodomains (KD=89 and 48nM, respectively). Also inhibits SMARCA2, and is otherwise selective over other bromodomain families. May play a role in SMARCA4 related cancers. Provided as 1 mg of dry powder.

Usage

Product Type:

Control Ligands & Inhibitors

Application:

Drug Discovery & Development

Storage Conditions:

Store at -20°C. Please avoid multiple freeze/thaw cycles.

Usage disclaimer:

These products may be covered by issued US and/or foreign patents, patent applications and subject to a Limited Use Label License. Please visit discoverx.com/license for a list of products that are governed by limited use label license terms and relevant patent and trademark information.

Additional Information

Brand:

Eurofins DiscoverX®