Biological Information

Background Information:

K 252a is a fungal alkaloid and analog of staurosporine that is a potent, cell-permeable inhibitor of PKC (IC50=32.9nM), calcium/calmodulin-stimulated phosphodiesterases (IC50=1.3-2.9uM), MLCK (Ki=20nM), and receptor tyrosine kinases. Promotes myogenic differentiation, neuronal culture survival, and apoptosis, among other biological effects. Provided as 200μg of dry powder.

Usage

Product Type:

Control Ligands & Inhibitors

Application:

Drug Discovery & Development

Storage Conditions:

Store at -20°C. Please avoid multiple freeze/thaw cycles.

Usage disclaimer:

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Additional Information

Brand:

Eurofins DiscoverX®