Improving the Predictive Power of GPCR Assays Webinar | Oct. 29th Presented by Terry Kenakin, Ph.D.

Thursday, October 29th, 2026 · 8am PT | 11am ET | 3pm GMT. Tuning GPCR System Sensitivity Webinar – Revealing True Drug Activity through Functional Volume Control. Presented by Terry Kenakin, Ph.D., Prof. of Pharmacology, U. N. Carolina, School of Medicine, Chapel Hill, NC, USA. The webinar highlights how functional volume control facilitates mechanistic differentiation of allosteric modulators by distinguishing effects on affinity versus efficacy. Approaches discussed provide a framework for improving the quantitative interpretation of pharmacological data and enhancing the predictive value of in vitro assays for in vivo drug activity.