Explore our Assay Panels

DiscoverX services offer a comprehensive portfolio of cell-based and biochemical assay formats against a broad range of target classes.  View available assays and assay panels below.  Don't see the assay you need?  Contact us if you don't see your target of interest in our list below as additional catalog items may be available for screening and profiling as a custom service.
 

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Kinases, Cell based

Browse Complete Target List

Listed below are the assays currently available for screening and profiling.  Assays may be sorted by column name. Contact us if you don't see your target of interest in list below as additional catalog assays may be available for screening and profiling as a custom service.
Target Gene ▲Common NameTarget ClassFamilySpecies
ADCYAP1R1PAC1GPCRVIP and PACAPHuman
ADORA1A1GPCRAdenosineHuman
ADORA2AA2AGPCRAdenosineHuman
ADORA2BA2BGPCRAdenosineHuman
ADORA3A3GPCRAdenosineHuman
ADRA1Aα1A-adrenoreceptorGPCRAdrenoceptorsHuman
ADRA1Bα1B-adrenoreceptorGPCRAdrenoceptorsHuman
ADRA2Aα2A-adrenoreceptorGPCRAdrenoceptorsHuman
ADRA2Bα2B-adrenoreceptorGPCRAdrenoceptorsHuman
ADRA2Cα2C-adrenoreceptorGPCRAdrenoceptorsHuman
ADRB1β1-adrenoreceptorGPCRAdrenoceptorsHuman
ADRB2β2-adrenoreceptorGPCRAdrenoceptorsHuman
ADRB3β3-adrenoreceptorGPCRAdrenoceptorsHuman
AGTR1AT1GPCRAngiotensinHuman
AGTRL1APJGPCRApelinHuman
ARARNHRNHRHuman
AVPR1AV1AGPCRVasopressin and OxytocinHuman
AVPR1BV1BGPCRVasopressin and OxytocinHuman
AVPR2V2GPCRVasopressin and OxytocinHuman
AXLEGFRKINASERTKHuman
BAI1BAI1GPCRClass B OrphanHuman
BAI2BAI2GPCRClass B OrphanHuman
BAI3BAI3GPCRClass B OrphanHuman
BDKRB1B1GPCRBradykininHuman
BDKRB2B2GPCRBradykininHuman
BLKNULLKINASECTKHuman
BRS3BB3GPCRBombesinHuman
C3AR1C3AGPCRComplement peptideHuman
C5AR1C5AGPCRComplement peptideHuman
C5L2C5L2GPCRComplement peptideHuman
CALCRCTGPCRCalcitoninHuman
CALCRL-RAMP1Calcitonin receptor-like receptorGPCRCalcitoninHuman
CALCRL-RAMP2Calcitonin receptor-like receptorGPCRCalcitoninHuman
CALCRL-RAMP3Calcitonin receptor-like receptorGPCRCalcitoninHuman
CALCR-RAMP1CTGPCRCalcitoninHuman
CALCR-RAMP2CTGPCRCalcitoninHuman
CALCR-RAMP3CTGPCRCalcitoninHuman
CASRCaSGPCRCalcium sensingHuman
CCKARCCK1GPCRCholecystokininHuman
CCKBRCCK2GPCRCholecystokininHuman
CCR1CCR1GPCRChemokineHuman
CCR10CCR10GPCRChemokineHuman
CCR2CCR2GPCRChemokineHuman
CCR3CCR3GPCRChemokineHuman
CCR4CCR4GPCRChemokineHuman
CCR5CCR5GPCRChemokineHuman
CCR6CCR6GPCRChemokineHuman
CCR7CCR7GPCRChemokineHuman
CCR8CCR8GPCRChemokineHuman
CCR9CCR9GPCRChemokineHuman
CCRL2CCRL2GPCRClass A OrphanHuman
CDC25ANULLPathwayPathwayHuman
cEDG5cS1P2GPCRLysophospholipid (S1P)Canine
CHRM1M1GPCRAcetylcholineHuman
CHRM2M2GPCRAcetylcholineHuman
CHRM3M3GPCRAcetylcholineHuman
CHRM4M4GPCRAcetylcholineHuman
CHRM5M5GPCRAcetylcholineHuman
c-KITKITKINASERTKHuman
c-METMETKINASERTKHuman
CMKLR1CMKLR1GPCRChemerinHuman
CNR1CB1GPCRCannabinoidHuman
CNR2CB2GPCRCannabinoidHuman
c-Ret-GFRα2RETKINASERTKHuman
CRHR1CRF1GPCRCorticotropin-releasing factorHuman
CRHR2CRF2GPCRCorticotropin-releasing factorHuman
CRTH2PTGDR2GPCRProstanoidHuman
CSF3R-JAK1NULLKINASECTKHuman
CX3CR1CX3CR1GPCRChemokineHuman
CXCR1CXCR1GPCRChemokineHuman
CXCR2CXCR2GPCRChemokineHuman
CXCR3CXCR3GPCRChemokineHuman
CXCR4CXCR4GPCRChemokineHuman
CXCR5CXCR5GPCRChemokineHuman
CXCR6CXCR6GPCRChemokineHuman
CXCR7CXCR7GPCRChemokineHuman
CYSLTR2CYSLT2GPCRLeukotriene Human
DARCFYGPCRNon-signalling 7TM chemokine-binding proteinsHuman
DDR1CD167aKINASERTKHuman
DRD1D1GPCRDopamineHuman
DRD2LD2LGPCRDopamineHuman
DRD2SD2SGPCRDopamineHuman
DRD3D3GPCRDopamineHuman
DRD4D4GPCRDopamineHuman
DRD5D5GPCRDopamineHuman
EBI2GPR183GPCRClass A OrphanHuman
EDG1S1P1GPCRLysophospholipid (S1P)Human
EDG2LPA1GPCRLysophospholipid (LPA)Human
EDG3S1P3GPCRLysophospholipid (S1P)Human
EDG4LPA2GPCRLysophospholipid (LPA)Human
EDG5S1P2GPCRLysophospholipid (S1P)Human
EDG6S1P4GPCRLysophospholipid (S1P)Human
EDG7LPA3GPCRLysophospholipid (LPA)Human
EDG8S1P5GPCRLysophospholipid (S1P)Human
EDNRAETAGPCREndothelinHuman
EDNRBETBGPCREndothelinHuman
EphA4EphA4KINASERTKHuman
EphA5EphA5KINASERTKHuman
EphA7EphA7KINASERTKHuman
EphB1EphB1KINASERTKHuman
EphB2EphB2KINASERTKHuman
EphB3EphB3KINASERTKHuman
EphB4EphB4KINASERTKHuman
ErbB1EGFRKINASERTKHuman
ErbB2-ErbB3HER2KINASERTKHuman
ErbB4HER4KINASERTKHuman
ERRαESRRANHRNHRHuman
ERαESR1NHRNHRHuman
F2RPAR1GPCRProtease activatedHuman
F2RL1PAR2GPCRProtease activatedHuman
F2RL3PAR4GPCRProtease activatedHuman
FFAR1FFA1GPCRFree Fatty AcidHuman
FFAR2GPR43GPCRFree Fatty AcidHuman
FFAR3GPR41GPCRFree Fatty AcidHuman
FGFR1FGFR1KINASERTKHuman
FGRNULLKINASECTKHuman
FLT4EGFRKINASERTKHuman
FOXO3forkhead box O3PathwayPathwayHuman
FPR1FPR1GPCRFormylpeptideHuman
FPR3FPRL2GPCRFormylpeptideHuman
FPRL1FPR2/ALXGPCRFormylpeptideHuman
FSHRFSHRGPCRGlycoprotein hormone receptorHuman
FXRNR1H4NHRNHRHuman
GABBR1-GABBR2GABB1GPCRGABABHuman
GALR1GALR1GPCRGalaninHuman
GALR2GALR2GPCRGalaninHuman
GCGRglucagonGPCRGlucagonHuman
GHRHRGHRHGPCRGlucagonHuman
GHR-JAK1NULLKINASECTKHuman
GHR-JAK2NULLKINASECTKHuman
GHSRghrelinGPCRGhrelinHuman
GHSR1bGHSR1bGPCRClass A OrphanHuman
GIPRGIPGPCRGlucagonHuman
GLP1RGLP-1GPCRGlucagonHuman
GLP2RGLP-2GPCRGlucagonHuman
GNRHRGnRHGPCRGonadotropin-releasing hormoneHuman
GPBAR1GPBAGPCRBile acidHuman
GPR1GPR1GPCRClass A OrphanHuman
GPR101GPR101GPCRClass A OrphanHuman
GPR103QRFPRGPCRPeptide P518Human
GPR107GPR107GPCROther 7TM proteinsHuman
GPR109AHCA2GPCRHydroxycarboxylic acidHuman
GPR109BHCA3GPCRHydroxycarboxylic acidHuman
GPR119GPR119GPCRClass A OrphanHuman
GPR12GPR12GPCRClass A OrphanHuman
GPR120FFA4GPCRFree fatty acidHuman
GPR120SFFA4GPCRFree fatty acidHuman
GPR123GPR123GPCRClass B OrphanHuman
GPR132GPR132GPCRClass A OrphanHuman
GPR135GPR135GPCRClass A OrphanHuman
GPR137TM7SF1GPCRClass A OrphanHuman
GPR139GPR139GPCRClass A OrphanHuman
GPR141GPR141GPCRClass A OrphanHuman
GPR142GPR142GPCRClass A OrphanHuman
GPR143GPR143GPCROther 7TM proteinsHuman
GPR146GPR146GPCRClass A OrphanHuman
GPR148GPR148GPCRClass A OrphanHuman
GPR149GPR149GPCRClass A OrphanHuman
GPR15GPR15GPCRClass A OrphanHuman
GPR150GPR150GPCRClass A OrphanHuman
GPR151GPR151GPCRClass A OrphanHuman
GPR152GPR152GPCRClass A OrphanHuman
GPR157GPR157GPCRClass B OrphanHuman
GPR161GPR161GPCRClass A OrphanHuman
GPR162GPR162GPCRClass A OrphanHuman
GPR17GPR17GPCRClass A OrphanHuman
GPR171GPR171GPCRClass A OrphanHuman
GPR173GPR173GPCRClass A OrphanHuman
GPR176GPR176GPCRClass A OrphanHuman
GPR18GPR18GPCRClass A OrphanHuman
GPR182GPR182GPCRClass A OrphanHuman
GPR20GPR20GPCRClass A OrphanHuman
GPR23LPA4GPCRClass A OrphanHuman
GPR25GPR25GPCRClass A OrphanHuman
GPR26GPR26GPCRClass A OrphanHuman
GPR27GPR27GPCRClass A OrphanHuman
GPR3GPR3GPCRClass A OrphanHuman
GPR30GPERGPCRClass A OrphanHuman
GPR31GPR31GPCRClass A OrphanHuman
GPR32GPR32GPCRClass A OrphanHuman
GPR35GPR35GPCRClass A OrphanHuman
GPR37EDNRBLGPCRClass A OrphanHuman
GPR37L1GPR37L1GPCRClass A OrphanHuman
GPR39GPR39GPCRClass A OrphanHuman
GPR4GPR4GPCRClass A OrphanHuman
GPR45GPR45GPCRClass A OrphanHuman
GPR50GPR50GPCRClass A OrphanHuman
GPR52GPR52GPCRClass A OrphanHuman
GPR55GPR55GPCRClass A OrphanHuman
GPR6GPR6GPCRClass A OrphanHuman
GPR61GPR61GPCRClass A OrphanHuman
GPR65GPR65GPCRClass A OrphanHuman
GPR75GPR75GPCRClass A OrphanHuman
GPR78GPR78GPCRClass A OrphanHuman
GPR79GPR79GPCRClass A OrphanHuman
GPR81HCA1GPCRHydroxycarboxylic acidHuman
GPR83GPR83GPCRClass A OrphanHuman
GPR84GPR84GPCRClass A OrphanHuman
GPR85GPR85GPCRClass A OrphanHuman
GPR88GPR88GPCRClass A OrphanHuman
GPR91SUCNR1GPCRClass A OrphanHuman
GPR92GPR92GPCRLysophospholipid (LPA)Human
GPR97GPR97GPCRClass B OrphanHuman
GRNR3C1NHRNHRHuman
GRM1mGlu1GPCRMetabotropic glutamateHuman
GRM2mGlu2GPCRMetabotropic glutamateHuman
GRM3MGlu3GPCRMetabotropic glutamateHuman
GRM4mGlu4GPCRMetabotropic glutamateHuman
GRM5mGlu5GPCRMetabotropic glutamateHuman
GRM6mGlu6GPCRMetabotropic glutamateHuman
GRPRBB2GPCRBombesinHuman
GSK3ββ-Catenin TranslocationPathwayPathwayHuman
HCRTR1OX1GPCROrexinHuman
HCRTR2OX2GPCROrexinHuman
HRH1H1GPCRHistamineHuman
HRH2H2GPCRHistamineHuman
HRH3H3GPCRHistamineHuman
HRH4H4GPCRHistamineHuman
HTR1A5HT1AGPCR5-HydroxytryptamineHuman
HTR1B5HT1BGPCR5-HydroxytryptamineHuman
HTR1E5HT1EGPCR5-HydroxytryptamineHuman
HTR1F5HT1FGPCR5-HydroxytryptamineHuman
HTR2A5HT2AGPCR5-HydroxytryptamineHuman
HTR2B5HT2BGPCR5-HydroxytryptamineHuman
HTR2C5HT2CGPCR5-HydroxytryptamineHuman
HTR5A5HT5AGPCR5-HydroxytryptamineHuman
HTR65HT6GPCR5-HydroxytryptamineHuman
HTR7D5HT7DGPCR5-HydroxytryptamineHuman
IGF1RIGF1RKINASERTKHuman
INSRINSRKINASERTKHuman
IκBNFKBIAPathwayPathwayHuman
JAK3PRLRKINASECTKHuman
KDREGFRKINASERTKHuman
Keap1-NRF2NFE2L2PathwayPathwayHuman
KISS1RkisspeptinGPCRKisspeptin receptorHuman
LGR4LGR4GPCRClass A OrphanHuman
LGR5LGR5GPCRClass A OrphanHuman
LGR6LGR6GPCRClass A OrphanHuman
LHCGRLHGPCRGlycoprotein hormone receptorHuman
LTB4RBLT1GPCRLeukotrieneHuman
LXRαNR1H3NHRNHRHuman
LXRβNR1H2NHRNHRHuman
LXRβ-NCoR1NR1H2NHRNHRHuman
mADCYAP1R1mPAC1GPCRVIP and PACAPMouse
mADORA2BmA2BGPCRAdenosineMouse
mADORA3mA3GPCRAdenosineMouse
mAGTRL1mAPJGPCRApelinMouse
MC1RMC1GPCRMelanocortinHuman
MC3RMC3GPCRMelanocortinHuman
MC4RMC4GPCRMelanocortinHuman
mC5AR1mC5ARGPCRComplement peptideMouse
MC5RMC5GPCRMelanocortinHuman
mCCR1mCC1GPCRChemokineMouse
mCCR2mCCR2GPCRChemokineMouse
mCCR3mCCR3GPCRChemokineMouse
mCCR4mCCR4GPCRChemokineMouse
mCCR5mCCR5GPCRChemokineMouse
mCCR6mCCR6GPCRChemokineMouse
mCCR7mCCR7GPCRChemokineMouse
mCCR8mCCR8GPCRChemokineMouse
mCCR9mCCR9GPCRChemokine Mouse
MCHR1MCH1GPCRMelanin-concentrating hormone Human
MCHR2MCH2GPCRMelanin-concentrating hormone Human
mCMKLR1mCMKLR1GPCRChemokineMouse
mCNR1mCB1GPCRCannabinoidMouse
mCNR2mCB2GPCRCannabinoidMouse
mCRHR1mCRF1GPCRCorticotropin-releasing factorMouse
mCRTH2mDP2GPCRProstanoidMouse
mCX3CR1mCX3CR1GPCRChemokineMouse
mCXCR2mCXCR2GPCRChemokineMouse
mCXCR3mCXCR3GPCRChemokineMouse
mCXCR4mCXCR4GPCRChemokineMouse
mCXCR5mCXCR5GPCRChemokineMouse
mCXCR6mCXCR6GPCRChemokineMouse
mCXCR7mCXCR7GPCRChemokineMouse
mDRD5mDRD5GPCRDopamineMouse
mEDG1mS1P1GPCRLysophospholipid (S1P)Mouse
mEDG5mS1P2GPCRLysophospholipid (S1P)Mouse
mEDG6mS1P4GPCRLysophospholipid (S1P)Mouse
mEDNRAmETAGPCREndothelinMouse
mEDNRBmETBGPCREndothelinMouse
mFPR1mFPR1GPCRFormylpeptide Mouse
mGALR2mGALR2GPCRGalaninMouse
mGCGRglucagonGPCRGlucagonMouse
mGHSRghrelinGPCRGhrelinMouse
mGIPRmGIPGPCRGlucagonMouse
mGLP1RmGLP-1GPCRGlucagonMouse
mGPR1mGPR1GPCRClass A OrphanMouse
mGPR120mGPR120GPCRFree fatty acidMouse
mHTR2Am5HT2AGPCR5-HydroxytryptamineMouse
mHTR2Cm5HT2CGPCR5-hydroxytryptamineMouse
MLNRmotilinGPCRMotilinHuman
mLTB4RmBLT1GPCRLeukotrieneMouse
mMCHR1MCH1GPCRMelanin-concentrating hormoneMouse
mNPY1RY1GPCRNeuropeptide YMouse
mNPY2RNPY2RGPCRNeuropeptide YMouse
mOPRD1δ (murine)GPCROpioidMouse
mOPRK1κ (murine)GPCROpioidMouse
mOPRM1μ (murine)GPCROpioidMouse
mOXTROTGPCRVasopressin and OxytocinMouse
mP2RY12mP2Y12GPCRP2YMouse
mP2RY6P2Y6GPCRP2YMouse
mPPYR1Y4GPCRNeuropeptide YMouse
mPTAFRmPAFGPCRPlatelet-activating factor Mouse
MRNR3C2NHRNHRHuman
MRGPREMRGPREGPCRClass A OrphanHuman
MRGPRFMRGPRFGPCRClass A OrphanHuman
MRGPRX1MRGPRX1GPCRClass A OrphanHuman
MRGPRX2MRGX2GPCRClass A OrphanHuman
MRGPRX4MRGPRX4GPCRClass A OrphanHuman
mSSTR2mSST2GPCRSomatostatinMouse
mSSTR5mSRIF1BGPCRSomatostatinMouse
MTNR1AMT1GPCRMelatoninHuman
MTNR1BMT2GPCRMelatoninHuman
mUTR2mUTGPCRUrotensinMouse
mVIPR1mVPAC1GPCRVIP and PACAPMouse
NMBRNMB-RGPCRBombesinHuman
NMU1RNMU1GPCRNeuromedin UHuman
NPBWR1NPBW1GPCRNeuropeptide B & WHuman
NPBWR2NPBW2GPCRNeuropeptide B & WHuman
NPFFR1NPFF1GPCRNeuropeptide FF & AFHuman
NPFFR2NPFF2GPCRNeuropeptide FF & AFHuman
NPR1NPR1PathwayPathwayHuman
NPSR1bNPS receptorGPCRNeuropeptide SHuman
NPY1RY1GPCRNeuropeptide YHuman
NPY2RY2GPCRNeuropeptide YHuman
NTSR1NTS1GPCRNeurotensinHuman
OPN5OPN5GPCRClass A OrphanHuman
OPRD1δGPCROpioidHuman
OPRK1κGPCROpioidHuman
OPRL1NOPGPCROpioidHuman
OPRM1μGPCROpioidHuman
OXER1OXEGPCRLeukotrieneHuman
OXGR1OXGR1GPCRClass A OrphanHuman
OXTROTGPCRVasopressin and OxytocinHuman
P2RY1P2RY1GPCRP2YHuman
P2RY11P2Y11GPCRP2YHuman
P2RY12P2Y12GPCRP2YHuman
P2RY2P2Y2GPCRP2YHuman
P2RY4P2Y4GPCRP2YHuman
P2RY6P2Y6GPCRP2YHuman
P2RY8P2RY8GPCRClass A OrphanHuman
P53NULLPathwayPathwayHuman
PDGFRaPDGFRaKINASERTKHuman
PDGFRbPDGFRbKINASERTKHuman
PPARαPPARANHRNHRHuman
PPARγPPARGNHRNHRHuman
PPARδPPARDNHRNHRHuman
PPYR1Y4GPCRNeuropeptide YHuman
PRLHRPRRPGPCRProlactin releasing peptide receptorHuman
PRLR-JAK1PRLRKINASECTKHuman
PRLR-JAK2PRLRKINASECTKHuman
PROKR1PKR1GPCRProkineticinHuman
PROKR2PKR2GPCRProkineticinHuman
PRαPGRNHRNHRHuman
PRβPGRNHRNHRHuman
PTAFRPAFGPCRPlatelet-activating factorHuman
PTGDRDP1GPCRProstanoidHuman
PTGER1EP1GPCRProstanoidHuman
PTGER2EP2GPCRProstanoidHuman
PTGER3EP3GPCRProstanoidHuman
PTGER4EP4GPCRProstanoidHuman
PTGFRFPGPCRProstanoidHuman
PTGIRIP1GPCRProstanoidHuman
PTHR1PTH1GPCRParathyroid hormoneHuman
PTHR2PTH2GPCRParathyroid hormoneHuman
RARαRARANHRNHRHuman
RARβRARBNHRNHRHuman
rCHRM4rM4GPCRAcetylcholineRat
rCRTH2rGPR44GPCRProstanoidRat
rDRD2LrD2LGPCRDopamineRat
rDRD2SrD2SGPCRDopamineRat
rEDG5rS1P2GPCRLysophospholipid (S1P)Rat
RELA-IκBRELAPathwayPathwayHuman
rGPR35rGPR35GPCRClass A OrphanRat
rHTR2CHTR2CGPCR5-HydroxytryptamineRat
rOPRM1μGPCROpioidRat
RORγRORCNHRNHRHuman
rPROKR1rPROKR1GPCRProkineticinRat
rPROKR2rPKR2GPCRProkineticinRat
rPTGER4rEP4GPCRProstanoidRat
RXFP1RXFP1GPCRRelaxinHuman
RXFP3RXFP3GPCRRelaxinHuman
RXFP4RXFP4GPCRRelaxinHuman
RXRαRXRANHRNHRHuman
RXRγRXRGNHRNHRHuman
SCTRsecretinGPCRGlucagonHuman
sEDG5sS1P2GPCRLysophospholipid (S1P)Simian
SREBP2SREBF2PathwayPathwayHuman
SSTR1SST1GPCRSomatostatinHuman
SSTR2SST2GPCRSomatostatinHuman
SSTR3SST3GPCRSomatostatinHuman
SSTR4SST4GPCRSomatostatinHuman
SSTR5SST5GPCRSomatostatinHuman
SYKNULLKINASECTKHuman
TAAR1TA1GPCRTrace amineHuman
TAAR5TAAR5GPCRClass A OrphanHuman
TACR1NK1GPCRTachykininHuman
TACR2NK2GPCRTachykininHuman
TACR3NK3GPCRTachykininHuman
TBXA2RTPGPCRProstanoidHuman
TGFBR1/TGFBR2TGFBR1PathwayPathwayHuman
THRαTHRANHRNHRHuman
THRβTHRBNHRNHRHuman
TORC1CRTC1PathwayPathwayHuman
TORC2CRTC2PathwayPathwayHuman
TRHRTRH1GPCRThyrotropin releasing hormoneHuman
TrkANTRK1KINASERTKHuman
TrkA-P75NTRK1KINASERTKHuman
TrkBNTRK2KINASERTKHuman
TrkB-P75NTRK2KINASERTKHuman
TrkCNTRK3KINASERTKHuman
TrkC-P75NTRK3KINASERTKHuman
TSHR(L)TSHGPCRGlycoprotein hormone receptorHuman
TYK2NULLKINASECTKHuman
UTR2UTGPCRUrotensinHuman
VIPR1VPAC1GPCRVIP and PACAPHuman
VIPR2VPAC2GPCRVIP and PACAPHuman
Wnt3β-Catenin TranslocationPathwayPathwayHuman
XBP1XBP1PathwayPathwayHuman
XCR1XCR1GPCRChemokineHuman
YES1NULLKINASECTKHuman