Target Gene ▲ | Common Name | Target Class | Family | Species |
ADCYAP1R1 | PAC1 | GPCR | VIP and PACAP | Human |
ADORA1 | A1 | GPCR | Adenosine | Human |
ADORA2A | A2A | GPCR | Adenosine | Human |
ADORA2B | A2B | GPCR | Adenosine | Human |
ADORA3 | A3 | GPCR | Adenosine | Human |
ADRA1A | α1A-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRA1B | α1B-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRA2A | α2A-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRA2B | α2B-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRA2C | α2C-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRB1 | β1-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRB2 | β2-adrenoreceptor | GPCR | Adrenoceptors | Human |
ADRB3 | β3-adrenoreceptor | GPCR | Adrenoceptors | Human |
AGTR1 | AT1 | GPCR | Angiotensin | Human |
AGTRL1 | APJ | GPCR | Apelin | Human |
AR | AR | NHR | NHR | Human |
AVPR1A | V1A | GPCR | Vasopressin and Oxytocin | Human |
AVPR1B | V1B | GPCR | Vasopressin and Oxytocin | Human |
AVPR2 | V2 | GPCR | Vasopressin and Oxytocin | Human |
AXL | EGFR | KINASE | RTK | Human |
BAI1 | BAI1 | GPCR | Class B Orphan | Human |
BAI2 | BAI2 | GPCR | Class B Orphan | Human |
BAI3 | BAI3 | GPCR | Class B Orphan | Human |
BDKRB1 | B1 | GPCR | Bradykinin | Human |
BDKRB2 | B2 | GPCR | Bradykinin | Human |
BLK | NULL | KINASE | CTK | Human |
BRS3 | BB3 | GPCR | Bombesin | Human |
C3AR1 | C3A | GPCR | Complement peptide | Human |
C5AR1 | C5A | GPCR | Complement peptide | Human |
C5L2 | C5L2 | GPCR | Complement peptide | Human |
CALCR | CT | GPCR | Calcitonin | Human |
CALCRL-RAMP1 | Calcitonin receptor-like receptor | GPCR | Calcitonin | Human |
CALCRL-RAMP2 | Calcitonin receptor-like receptor | GPCR | Calcitonin | Human |
CALCRL-RAMP3 | Calcitonin receptor-like receptor | GPCR | Calcitonin | Human |
CALCR-RAMP1 | CT | GPCR | Calcitonin | Human |
CALCR-RAMP2 | CT | GPCR | Calcitonin | Human |
CALCR-RAMP3 | CT | GPCR | Calcitonin | Human |
CASR | CaS | GPCR | Calcium sensing | Human |
CCKAR | CCK1 | GPCR | Cholecystokinin | Human |
CCKBR | CCK2 | GPCR | Cholecystokinin | Human |
CCR1 | CCR1 | GPCR | Chemokine | Human |
CCR10 | CCR10 | GPCR | Chemokine | Human |
CCR2 | CCR2 | GPCR | Chemokine | Human |
CCR3 | CCR3 | GPCR | Chemokine | Human |
CCR4 | CCR4 | GPCR | Chemokine | Human |
CCR5 | CCR5 | GPCR | Chemokine | Human |
CCR6 | CCR6 | GPCR | Chemokine | Human |
CCR7 | CCR7 | GPCR | Chemokine | Human |
CCR8 | CCR8 | GPCR | Chemokine | Human |
CCR9 | CCR9 | GPCR | Chemokine | Human |
CCRL2 | CCRL2 | GPCR | Class A Orphan | Human |
CDC25A | NULL | Pathway | Pathway | Human |
cEDG5 | cS1P2 | GPCR | Lysophospholipid (S1P) | Canine |
CHRM1 | M1 | GPCR | Acetylcholine | Human |
CHRM2 | M2 | GPCR | Acetylcholine | Human |
CHRM3 | M3 | GPCR | Acetylcholine | Human |
CHRM4 | M4 | GPCR | Acetylcholine | Human |
CHRM5 | M5 | GPCR | Acetylcholine | Human |
c-KIT | KIT | KINASE | RTK | Human |
c-MET | MET | KINASE | RTK | Human |
CMKLR1 | CMKLR1 | GPCR | Chemerin | Human |
CNR1 | CB1 | GPCR | Cannabinoid | Human |
CNR2 | CB2 | GPCR | Cannabinoid | Human |
c-Ret-GFRα2 | RET | KINASE | RTK | Human |
CRHR1 | CRF1 | GPCR | Corticotropin-releasing factor | Human |
CRHR2 | CRF2 | GPCR | Corticotropin-releasing factor | Human |
CRTH2 | PTGDR2 | GPCR | Prostanoid | Human |
CSF3R-JAK1 | NULL | KINASE | CTK | Human |
CX3CR1 | CX3CR1 | GPCR | Chemokine | Human |
CXCR1 | CXCR1 | GPCR | Chemokine | Human |
CXCR2 | CXCR2 | GPCR | Chemokine | Human |
CXCR3 | CXCR3 | GPCR | Chemokine | Human |
CXCR4 | CXCR4 | GPCR | Chemokine | Human |
CXCR5 | CXCR5 | GPCR | Chemokine | Human |
CXCR6 | CXCR6 | GPCR | Chemokine | Human |
CXCR7 | CXCR7 | GPCR | Chemokine | Human |
CYSLTR2 | CYSLT2 | GPCR | Leukotriene | Human |
DARC | FY | GPCR | Non-signalling 7TM chemokine-binding proteins | Human |
DDR1 | CD167a | KINASE | RTK | Human |
DRD1 | D1 | GPCR | Dopamine | Human |
DRD2L | D2L | GPCR | Dopamine | Human |
DRD2S | D2S | GPCR | Dopamine | Human |
DRD3 | D3 | GPCR | Dopamine | Human |
DRD4 | D4 | GPCR | Dopamine | Human |
DRD5 | D5 | GPCR | Dopamine | Human |
EBI2 | GPR183 | GPCR | Class A Orphan | Human |
EDG1 | S1P1 | GPCR | Lysophospholipid (S1P) | Human |
EDG2 | LPA1 | GPCR | Lysophospholipid (LPA) | Human |
EDG3 | S1P3 | GPCR | Lysophospholipid (S1P) | Human |
EDG4 | LPA2 | GPCR | Lysophospholipid (LPA) | Human |
EDG5 | S1P2 | GPCR | Lysophospholipid (S1P) | Human |
EDG6 | S1P4 | GPCR | Lysophospholipid (S1P) | Human |
EDG7 | LPA3 | GPCR | Lysophospholipid (LPA) | Human |
EDG8 | S1P5 | GPCR | Lysophospholipid (S1P) | Human |
EDNRA | ETA | GPCR | Endothelin | Human |
EDNRB | ETB | GPCR | Endothelin | Human |
EphA4 | EphA4 | KINASE | RTK | Human |
EphA5 | EphA5 | KINASE | RTK | Human |
EphA7 | EphA7 | KINASE | RTK | Human |
EphB1 | EphB1 | KINASE | RTK | Human |
EphB2 | EphB2 | KINASE | RTK | Human |
EphB3 | EphB3 | KINASE | RTK | Human |
EphB4 | EphB4 | KINASE | RTK | Human |
ErbB1 | EGFR | KINASE | RTK | Human |
ErbB2-ErbB3 | HER2 | KINASE | RTK | Human |
ErbB4 | HER4 | KINASE | RTK | Human |
ERRα | ESRRA | NHR | NHR | Human |
ERα | ESR1 | NHR | NHR | Human |
F2R | PAR1 | GPCR | Protease activated | Human |
F2RL1 | PAR2 | GPCR | Protease activated | Human |
F2RL3 | PAR4 | GPCR | Protease activated | Human |
FFAR1 | FFA1 | GPCR | Free Fatty Acid | Human |
FFAR2 | GPR43 | GPCR | Free Fatty Acid | Human |
FFAR3 | GPR41 | GPCR | Free Fatty Acid | Human |
FGFR1 | FGFR1 | KINASE | RTK | Human |
FGR | NULL | KINASE | CTK | Human |
FLT4 | EGFR | KINASE | RTK | Human |
FOXO3 | forkhead box O3 | Pathway | Pathway | Human |
FPR1 | FPR1 | GPCR | Formylpeptide | Human |
FPR3 | FPRL2 | GPCR | Formylpeptide | Human |
FPRL1 | FPR2/ALX | GPCR | Formylpeptide | Human |
FSHR | FSHR | GPCR | Glycoprotein hormone receptor | Human |
FXR | NR1H4 | NHR | NHR | Human |
GABBR1-GABBR2 | GABB1 | GPCR | GABAB | Human |
GALR1 | GALR1 | GPCR | Galanin | Human |
GALR2 | GALR2 | GPCR | Galanin | Human |
GCGR | glucagon | GPCR | Glucagon | Human |
GHRHR | GHRH | GPCR | Glucagon | Human |
GHR-JAK1 | NULL | KINASE | CTK | Human |
GHR-JAK2 | NULL | KINASE | CTK | Human |
GHSR | ghrelin | GPCR | Ghrelin | Human |
GHSR1b | GHSR1b | GPCR | Class A Orphan | Human |
GIPR | GIP | GPCR | Glucagon | Human |
GLP1R | GLP-1 | GPCR | Glucagon | Human |
GLP2R | GLP-2 | GPCR | Glucagon | Human |
GNRHR | GnRH | GPCR | Gonadotropin-releasing hormone | Human |
GPBAR1 | GPBA | GPCR | Bile acid | Human |
GPR1 | GPR1 | GPCR | Class A Orphan | Human |
GPR101 | GPR101 | GPCR | Class A Orphan | Human |
GPR103 | QRFPR | GPCR | Peptide P518 | Human |
GPR107 | GPR107 | GPCR | Other 7TM proteins | Human |
GPR109A | HCA2 | GPCR | Hydroxycarboxylic acid | Human |
GPR109B | HCA3 | GPCR | Hydroxycarboxylic acid | Human |
GPR119 | GPR119 | GPCR | Class A Orphan | Human |
GPR12 | GPR12 | GPCR | Class A Orphan | Human |
GPR120 | FFA4 | GPCR | Free fatty acid | Human |
GPR120S | FFA4 | GPCR | Free fatty acid | Human |
GPR123 | GPR123 | GPCR | Class B Orphan | Human |
GPR132 | GPR132 | GPCR | Class A Orphan | Human |
GPR135 | GPR135 | GPCR | Class A Orphan | Human |
GPR137 | TM7SF1 | GPCR | Class A Orphan | Human |
GPR139 | GPR139 | GPCR | Class A Orphan | Human |
GPR141 | GPR141 | GPCR | Class A Orphan | Human |
GPR142 | GPR142 | GPCR | Class A Orphan | Human |
GPR143 | GPR143 | GPCR | Other 7TM proteins | Human |
GPR146 | GPR146 | GPCR | Class A Orphan | Human |
GPR148 | GPR148 | GPCR | Class A Orphan | Human |
GPR149 | GPR149 | GPCR | Class A Orphan | Human |
GPR15 | GPR15 | GPCR | Class A Orphan | Human |
GPR150 | GPR150 | GPCR | Class A Orphan | Human |
GPR151 | GPR151 | GPCR | Class A Orphan | Human |
GPR152 | GPR152 | GPCR | Class A Orphan | Human |
GPR157 | GPR157 | GPCR | Class B Orphan | Human |
GPR161 | GPR161 | GPCR | Class A Orphan | Human |
GPR162 | GPR162 | GPCR | Class A Orphan | Human |
GPR17 | GPR17 | GPCR | Class A Orphan | Human |
GPR171 | GPR171 | GPCR | Class A Orphan | Human |
GPR173 | GPR173 | GPCR | Class A Orphan | Human |
GPR176 | GPR176 | GPCR | Class A Orphan | Human |
GPR18 | GPR18 | GPCR | Class A Orphan | Human |
GPR182 | GPR182 | GPCR | Class A Orphan | Human |
GPR20 | GPR20 | GPCR | Class A Orphan | Human |
GPR23 | LPA4 | GPCR | Class A Orphan | Human |
GPR25 | GPR25 | GPCR | Class A Orphan | Human |
GPR26 | GPR26 | GPCR | Class A Orphan | Human |
GPR27 | GPR27 | GPCR | Class A Orphan | Human |
GPR3 | GPR3 | GPCR | Class A Orphan | Human |
GPR30 | GPER | GPCR | Class A Orphan | Human |
GPR31 | GPR31 | GPCR | Class A Orphan | Human |
GPR32 | GPR32 | GPCR | Class A Orphan | Human |
GPR35 | GPR35 | GPCR | Class A Orphan | Human |
GPR37 | EDNRBL | GPCR | Class A Orphan | Human |
GPR37L1 | GPR37L1 | GPCR | Class A Orphan | Human |
GPR39 | GPR39 | GPCR | Class A Orphan | Human |
GPR4 | GPR4 | GPCR | Class A Orphan | Human |
GPR45 | GPR45 | GPCR | Class A Orphan | Human |
GPR50 | GPR50 | GPCR | Class A Orphan | Human |
GPR52 | GPR52 | GPCR | Class A Orphan | Human |
GPR55 | GPR55 | GPCR | Class A Orphan | Human |
GPR6 | GPR6 | GPCR | Class A Orphan | Human |
GPR61 | GPR61 | GPCR | Class A Orphan | Human |
GPR65 | GPR65 | GPCR | Class A Orphan | Human |
GPR75 | GPR75 | GPCR | Class A Orphan | Human |
GPR78 | GPR78 | GPCR | Class A Orphan | Human |
GPR79 | GPR79 | GPCR | Class A Orphan | Human |
GPR81 | HCA1 | GPCR | Hydroxycarboxylic acid | Human |
GPR83 | GPR83 | GPCR | Class A Orphan | Human |
GPR84 | GPR84 | GPCR | Class A Orphan | Human |
GPR85 | GPR85 | GPCR | Class A Orphan | Human |
GPR88 | GPR88 | GPCR | Class A Orphan | Human |
GPR91 | SUCNR1 | GPCR | Class A Orphan | Human |
GPR92 | GPR92 | GPCR | Lysophospholipid (LPA) | Human |
GPR97 | GPR97 | GPCR | Class B Orphan | Human |
GR | NR3C1 | NHR | NHR | Human |
GRM1 | mGlu1 | GPCR | Metabotropic glutamate | Human |
GRM2 | mGlu2 | GPCR | Metabotropic glutamate | Human |
GRM3 | MGlu3 | GPCR | Metabotropic glutamate | Human |
GRM4 | mGlu4 | GPCR | Metabotropic glutamate | Human |
GRM5 | mGlu5 | GPCR | Metabotropic glutamate | Human |
GRM6 | mGlu6 | GPCR | Metabotropic glutamate | Human |
GRPR | BB2 | GPCR | Bombesin | Human |
GSK3β | β-Catenin Translocation | Pathway | Pathway | Human |
HCRTR1 | OX1 | GPCR | Orexin | Human |
HCRTR2 | OX2 | GPCR | Orexin | Human |
HRH1 | H1 | GPCR | Histamine | Human |
HRH2 | H2 | GPCR | Histamine | Human |
HRH3 | H3 | GPCR | Histamine | Human |
HRH4 | H4 | GPCR | Histamine | Human |
HTR1A | 5HT1A | GPCR | 5-Hydroxytryptamine | Human |
HTR1B | 5HT1B | GPCR | 5-Hydroxytryptamine | Human |
HTR1E | 5HT1E | GPCR | 5-Hydroxytryptamine | Human |
HTR1F | 5HT1F | GPCR | 5-Hydroxytryptamine | Human |
HTR2A | 5HT2A | GPCR | 5-Hydroxytryptamine | Human |
HTR2B | 5HT2B | GPCR | 5-Hydroxytryptamine | Human |
HTR2C | 5HT2C | GPCR | 5-Hydroxytryptamine | Human |
HTR5A | 5HT5A | GPCR | 5-Hydroxytryptamine | Human |
HTR6 | 5HT6 | GPCR | 5-Hydroxytryptamine | Human |
HTR7D | 5HT7D | GPCR | 5-Hydroxytryptamine | Human |
IGF1R | IGF1R | KINASE | RTK | Human |
INSR | INSR | KINASE | RTK | Human |
IκB | NFKBIA | Pathway | Pathway | Human |
JAK3 | PRLR | KINASE | CTK | Human |
KDR | EGFR | KINASE | RTK | Human |
Keap1-NRF2 | NFE2L2 | Pathway | Pathway | Human |
KISS1R | kisspeptin | GPCR | Kisspeptin receptor | Human |
LGR4 | LGR4 | GPCR | Class A Orphan | Human |
LGR5 | LGR5 | GPCR | Class A Orphan | Human |
LGR6 | LGR6 | GPCR | Class A Orphan | Human |
LHCGR | LH | GPCR | Glycoprotein hormone receptor | Human |
LTB4R | BLT1 | GPCR | Leukotriene | Human |
LXRα | NR1H3 | NHR | NHR | Human |
LXRβ | NR1H2 | NHR | NHR | Human |
LXRβ-NCoR1 | NR1H2 | NHR | NHR | Human |
mADCYAP1R1 | mPAC1 | GPCR | VIP and PACAP | Mouse |
mADORA2B | mA2B | GPCR | Adenosine | Mouse |
mADORA3 | mA3 | GPCR | Adenosine | Mouse |
mAGTRL1 | mAPJ | GPCR | Apelin | Mouse |
MC1R | MC1 | GPCR | Melanocortin | Human |
MC3R | MC3 | GPCR | Melanocortin | Human |
MC4R | MC4 | GPCR | Melanocortin | Human |
mC5AR1 | mC5AR | GPCR | Complement peptide | Mouse |
MC5R | MC5 | GPCR | Melanocortin | Human |
mCCR1 | mCC1 | GPCR | Chemokine | Mouse |
mCCR2 | mCCR2 | GPCR | Chemokine | Mouse |
mCCR3 | mCCR3 | GPCR | Chemokine | Mouse |
mCCR4 | mCCR4 | GPCR | Chemokine | Mouse |
mCCR5 | mCCR5 | GPCR | Chemokine | Mouse |
mCCR6 | mCCR6 | GPCR | Chemokine | Mouse |
mCCR7 | mCCR7 | GPCR | Chemokine | Mouse |
mCCR8 | mCCR8 | GPCR | Chemokine | Mouse |
mCCR9 | mCCR9 | GPCR | Chemokine | Mouse |
MCHR1 | MCH1 | GPCR | Melanin-concentrating hormone | Human |
MCHR2 | MCH2 | GPCR | Melanin-concentrating hormone | Human |
mCMKLR1 | mCMKLR1 | GPCR | Chemokine | Mouse |
mCNR1 | mCB1 | GPCR | Cannabinoid | Mouse |
mCNR2 | mCB2 | GPCR | Cannabinoid | Mouse |
mCRHR1 | mCRF1 | GPCR | Corticotropin-releasing factor | Mouse |
mCRTH2 | mDP2 | GPCR | Prostanoid | Mouse |
mCX3CR1 | mCX3CR1 | GPCR | Chemokine | Mouse |
mCXCR2 | mCXCR2 | GPCR | Chemokine | Mouse |
mCXCR3 | mCXCR3 | GPCR | Chemokine | Mouse |
mCXCR4 | mCXCR4 | GPCR | Chemokine | Mouse |
mCXCR5 | mCXCR5 | GPCR | Chemokine | Mouse |
mCXCR6 | mCXCR6 | GPCR | Chemokine | Mouse |
mCXCR7 | mCXCR7 | GPCR | Chemokine | Mouse |
mDRD5 | mDRD5 | GPCR | Dopamine | Mouse |
mEDG1 | mS1P1 | GPCR | Lysophospholipid (S1P) | Mouse |
mEDG5 | mS1P2 | GPCR | Lysophospholipid (S1P) | Mouse |
mEDG6 | mS1P4 | GPCR | Lysophospholipid (S1P) | Mouse |
mEDNRA | mETA | GPCR | Endothelin | Mouse |
mEDNRB | mETB | GPCR | Endothelin | Mouse |
mFPR1 | mFPR1 | GPCR | Formylpeptide | Mouse |
mGALR2 | mGALR2 | GPCR | Galanin | Mouse |
mGCGR | glucagon | GPCR | Glucagon | Mouse |
mGHSR | ghrelin | GPCR | Ghrelin | Mouse |
mGIPR | mGIP | GPCR | Glucagon | Mouse |
mGLP1R | mGLP-1 | GPCR | Glucagon | Mouse |
mGPR1 | mGPR1 | GPCR | Class A Orphan | Mouse |
mGPR120 | mGPR120 | GPCR | Free fatty acid | Mouse |
mHTR2A | m5HT2A | GPCR | 5-Hydroxytryptamine | Mouse |
mHTR2C | m5HT2C | GPCR | 5-hydroxytryptamine | Mouse |
MLNR | motilin | GPCR | Motilin | Human |
mLTB4R | mBLT1 | GPCR | Leukotriene | Mouse |
mMCHR1 | MCH1 | GPCR | Melanin-concentrating hormone | Mouse |
mNPY1R | Y1 | GPCR | Neuropeptide Y | Mouse |
mNPY2R | NPY2R | GPCR | Neuropeptide Y | Mouse |
mOPRD1 | δ (murine) | GPCR | Opioid | Mouse |
mOPRK1 | κ (murine) | GPCR | Opioid | Mouse |
mOPRM1 | μ (murine) | GPCR | Opioid | Mouse |
mOXTR | OT | GPCR | Vasopressin and Oxytocin | Mouse |
mP2RY12 | mP2Y12 | GPCR | P2Y | Mouse |
mP2RY6 | P2Y6 | GPCR | P2Y | Mouse |
mPPYR1 | Y4 | GPCR | Neuropeptide Y | Mouse |
mPTAFR | mPAF | GPCR | Platelet-activating factor | Mouse |
MR | NR3C2 | NHR | NHR | Human |
MRGPRE | MRGPRE | GPCR | Class A Orphan | Human |
MRGPRF | MRGPRF | GPCR | Class A Orphan | Human |
MRGPRX1 | MRGPRX1 | GPCR | Class A Orphan | Human |
MRGPRX2 | MRGX2 | GPCR | Class A Orphan | Human |
MRGPRX4 | MRGPRX4 | GPCR | Class A Orphan | Human |
mSSTR2 | mSST2 | GPCR | Somatostatin | Mouse |
mSSTR5 | mSRIF1B | GPCR | Somatostatin | Mouse |
MTNR1A | MT1 | GPCR | Melatonin | Human |
MTNR1B | MT2 | GPCR | Melatonin | Human |
mUTR2 | mUT | GPCR | Urotensin | Mouse |
mVIPR1 | mVPAC1 | GPCR | VIP and PACAP | Mouse |
NMBR | NMB-R | GPCR | Bombesin | Human |
NMU1R | NMU1 | GPCR | Neuromedin U | Human |
NPBWR1 | NPBW1 | GPCR | Neuropeptide B & W | Human |
NPBWR2 | NPBW2 | GPCR | Neuropeptide B & W | Human |
NPFFR1 | NPFF1 | GPCR | Neuropeptide FF & AF | Human |
NPFFR2 | NPFF2 | GPCR | Neuropeptide FF & AF | Human |
NPR1 | NPR1 | Pathway | Pathway | Human |
NPSR1b | NPS receptor | GPCR | Neuropeptide S | Human |
NPY1R | Y1 | GPCR | Neuropeptide Y | Human |
NPY2R | Y2 | GPCR | Neuropeptide Y | Human |
NTSR1 | NTS1 | GPCR | Neurotensin | Human |
OPN5 | OPN5 | GPCR | Class A Orphan | Human |
OPRD1 | δ | GPCR | Opioid | Human |
OPRK1 | κ | GPCR | Opioid | Human |
OPRL1 | NOP | GPCR | Opioid | Human |
OPRM1 | μ | GPCR | Opioid | Human |
OXER1 | OXE | GPCR | Leukotriene | Human |
OXGR1 | OXGR1 | GPCR | Class A Orphan | Human |
OXTR | OT | GPCR | Vasopressin and Oxytocin | Human |
P2RY1 | P2RY1 | GPCR | P2Y | Human |
P2RY11 | P2Y11 | GPCR | P2Y | Human |
P2RY12 | P2Y12 | GPCR | P2Y | Human |
P2RY2 | P2Y2 | GPCR | P2Y | Human |
P2RY4 | P2Y4 | GPCR | P2Y | Human |
P2RY6 | P2Y6 | GPCR | P2Y | Human |
P2RY8 | P2RY8 | GPCR | Class A Orphan | Human |
P53 | NULL | Pathway | Pathway | Human |
PDGFRa | PDGFRa | KINASE | RTK | Human |
PDGFRb | PDGFRb | KINASE | RTK | Human |
PPARα | PPARA | NHR | NHR | Human |
PPARγ | PPARG | NHR | NHR | Human |
PPARδ | PPARD | NHR | NHR | Human |
PPYR1 | Y4 | GPCR | Neuropeptide Y | Human |
PRLHR | PRRP | GPCR | Prolactin releasing peptide receptor | Human |
PRLR-JAK1 | PRLR | KINASE | CTK | Human |
PRLR-JAK2 | PRLR | KINASE | CTK | Human |
PROKR1 | PKR1 | GPCR | Prokineticin | Human |
PROKR2 | PKR2 | GPCR | Prokineticin | Human |
PRα | PGR | NHR | NHR | Human |
PRβ | PGR | NHR | NHR | Human |
PTAFR | PAF | GPCR | Platelet-activating factor | Human |
PTGDR | DP1 | GPCR | Prostanoid | Human |
PTGER1 | EP1 | GPCR | Prostanoid | Human |
PTGER2 | EP2 | GPCR | Prostanoid | Human |
PTGER3 | EP3 | GPCR | Prostanoid | Human |
PTGER4 | EP4 | GPCR | Prostanoid | Human |
PTGFR | FP | GPCR | Prostanoid | Human |
PTGIR | IP1 | GPCR | Prostanoid | Human |
PTHR1 | PTH1 | GPCR | Parathyroid hormone | Human |
PTHR2 | PTH2 | GPCR | Parathyroid hormone | Human |
RARα | RARA | NHR | NHR | Human |
RARβ | RARB | NHR | NHR | Human |
rCHRM4 | rM4 | GPCR | Acetylcholine | Rat |
rCRTH2 | rGPR44 | GPCR | Prostanoid | Rat |
rDRD2L | rD2L | GPCR | Dopamine | Rat |
rDRD2S | rD2S | GPCR | Dopamine | Rat |
rEDG5 | rS1P2 | GPCR | Lysophospholipid (S1P) | Rat |
RELA-IκB | RELA | Pathway | Pathway | Human |
rGPR35 | rGPR35 | GPCR | Class A Orphan | Rat |
rHTR2C | HTR2C | GPCR | 5-Hydroxytryptamine | Rat |
rOPRM1 | μ | GPCR | Opioid | Rat |
RORγ | RORC | NHR | NHR | Human |
rPROKR1 | rPROKR1 | GPCR | Prokineticin | Rat |
rPROKR2 | rPKR2 | GPCR | Prokineticin | Rat |
rPTGER4 | rEP4 | GPCR | Prostanoid | Rat |
RXFP1 | RXFP1 | GPCR | Relaxin | Human |
RXFP3 | RXFP3 | GPCR | Relaxin | Human |
RXFP4 | RXFP4 | GPCR | Relaxin | Human |
RXRα | RXRA | NHR | NHR | Human |
RXRγ | RXRG | NHR | NHR | Human |
SCTR | secretin | GPCR | Glucagon | Human |
sEDG5 | sS1P2 | GPCR | Lysophospholipid (S1P) | Simian |
SREBP2 | SREBF2 | Pathway | Pathway | Human |
SSTR1 | SST1 | GPCR | Somatostatin | Human |
SSTR2 | SST2 | GPCR | Somatostatin | Human |
SSTR3 | SST3 | GPCR | Somatostatin | Human |
SSTR4 | SST4 | GPCR | Somatostatin | Human |
SSTR5 | SST5 | GPCR | Somatostatin | Human |
SYK | NULL | KINASE | CTK | Human |
TAAR1 | TA1 | GPCR | Trace amine | Human |
TAAR5 | TAAR5 | GPCR | Class A Orphan | Human |
TACR1 | NK1 | GPCR | Tachykinin | Human |
TACR2 | NK2 | GPCR | Tachykinin | Human |
TACR3 | NK3 | GPCR | Tachykinin | Human |
TBXA2R | TP | GPCR | Prostanoid | Human |
TGFBR1/TGFBR2 | TGFBR1 | Pathway | Pathway | Human |
THRα | THRA | NHR | NHR | Human |
THRβ | THRB | NHR | NHR | Human |
TORC1 | CRTC1 | Pathway | Pathway | Human |
TORC2 | CRTC2 | Pathway | Pathway | Human |
TRHR | TRH1 | GPCR | Thyrotropin releasing hormone | Human |
TrkA | NTRK1 | KINASE | RTK | Human |
TrkA-P75 | NTRK1 | KINASE | RTK | Human |
TrkB | NTRK2 | KINASE | RTK | Human |
TrkB-P75 | NTRK2 | KINASE | RTK | Human |
TrkC | NTRK3 | KINASE | RTK | Human |
TrkC-P75 | NTRK3 | KINASE | RTK | Human |
TSHR(L) | TSH | GPCR | Glycoprotein hormone receptor | Human |
TYK2 | NULL | KINASE | CTK | Human |
UTR2 | UT | GPCR | Urotensin | Human |
VIPR1 | VPAC1 | GPCR | VIP and PACAP | Human |
VIPR2 | VPAC2 | GPCR | VIP and PACAP | Human |
Wnt3 | β-Catenin Translocation | Pathway | Pathway | Human |
XBP1 | XBP1 | Pathway | Pathway | Human |
XCR1 | XCR1 | GPCR | Chemokine | Human |
YES1 | NULL | KINASE | CTK | Human |