Alphabetical Target List

AAK1 ABL1 ABL1(E255K)-phosphorylated ABL1(F317I)-nonphosphorylated ABL1(F317I)-phosphorylated
ABL1(F317L)-nonphosphorylated ABL1(F317L)-phosphorylated ABL1(H396P)-nonphosphorylated ABL1(H396P)-phosphorylated ABL1(M351T)-phosphorylated
ABL1(Q252H)-nonphosphorylated ABL1(Q252H)-phosphorylated ABL1(T315I)-nonphosphorylated ABL1(T315I)-phosphorylated ABL1(Y253F)-phosphorylated
ABL1-nonphosphorylated ABL1-phosphorylated ABL2 ACVR1 ACVR1B
ACVR1B/BMPR2 ACVR1C/ACVR2 ACVR1C/ACVR2B ACVR2/ACVR1 ACVR2A
ACVR2B ACVRL1 ACVRL1/ACVR2 ACVRL1/ACVR2B ACVRL1/BMPR2
ADCK3 ADCK4 ADCYAP1R1 ADORA1 ADORA2A
ADORA2B ADORA3 ADRA1A ADRA1B ADRA1D(82-572)
ADRA2A ADRA2B ADRA2C ADRB1 ADRB2
ADRB2(W158A) ADRB3 AGTR1 AGTRL1 AKT1
AKT2 AKT3 ALK ALK(1151Tins) ALK(C1156Y)
ALK(F1174L) ALK(L1196M) AMPK-alpha1 AMPK-alpha2 ANKK1
AR ARK5 ASK1 ASK2 ATAD2A
ATAD2B ATAD2B AURKA AURKB AURKC
AVPR1A AVPR1B AVPR2 AVPR2(S167T) AXL
BAI1 BAI2 BAI3 BAZ1A BAZ1B
BAZ2A BAZ2A BAZ2B BCL2-BAX BCL2-BIM
BCL2L1-BAX BCL2L1-BIM BDKRB1 BDKRB2 BIKE
BLK BMPR1A BMPR1A/ACVR2 BMPR1A/ACVR2B BMPR1A/BMPR2
BMPR1B BMPR1B/ACVR2 BMPR1B/ACVR2B BMPR1B/BMPR2 BMPR2
BMX BRAF BRAF(V600E) BRD1 Brd2(1)
BRD2(1,2) BRD2(2) BRD3(1) BRD3(1) BRD3(1,2)
BRD3(2) Brd4(1) BRD4(1,2) BRD4(2) BRD4(full-length,short-iso.)
Brd7 BRD8(1) BRD8(2) BRD9 BrdT(1)
BRDT(1,2) BRDT(2) BRK BRPF1 BRPF3
BRPF3 BRS3 BRSK1 BRSK2 BRWD3(2)
BTK BUB1 C3AR1 C5AR1 C5L2
CALCR CALCRL-RAMP1 CALCRL-RAMP2 CALCRL-RAMP3 CALCR-RAMP2
CALCR-RAMP3 CAMK1 CAMK1B CAMK1D CAMK1G
CAMK2A CAMK2B CAMK2D CAMK2G CAMK4
CAMKK1 CAMKK2 CASK CASR CCKAR
CCKBR CCR1 CCR10 CCR2 CCR3
CCR4 CCR5 CCR6 CCR7 CCR8
CCR9 CCRL1 CCRL2 CD137 CD86
CDC25A CDC2L1 CDC2L2 CDC2L5 CDK1
CDK10 CDK11 CDK12 CDK2 CDK20
CDK3 CDK4 CDK4-cyclinD1 CDK4-cyclinD1(F93L) CDK4-cyclinD3
CDK5 CDK6 CDK7 CDK8 CDK9
CDKL1 CDKL2 CDKL3 CDKL5 CECR2
cEDG5 CFTR-ΔF508 cGPR91 CHEK1 CHEK2
CHRM1 CHRM2 CHRM3 CHRM4 CHRM5
cINSRa cINSRb CIT c-KIT CLK1
CLK2 CLK3 CLK4 c-MET/c-MET CMKLR1
CNR1 CNR2 CREBBP c-Ret-GFRα1 c-Ret-GFRα2
CRHR1 CRHR2 CRTH2 CSF1R CSF1R/CSF1R
CSF1R-autoinhibited CSF2RB/CSF2RA CSF3R-JAK1 CSK CSNK1A1
CSNK1A1L CSNK1D CSNK1E CSNK1G1 CSNK1G2
CSNK1G3 CSNK2A1 CSNK2A2 CTK CTLA4
CX3CR1 CXCR1 CXCR2 CXCR3 CXCR4
CXCR5 CXCR6 CXCR7 cyno CXCR1 cyno CXCR2
cyno GPR120 cyno MRGPRX2 CYSLTR2 DAPK1 DAPK2
DAPK3 DARC DCAMKL1 DCAMKL2 DCAMKL3
DDR1 DDR2(T654M) DLK DMPK DMPK2
DRAK1 DRAK2 DRD1 DRD2L DRD2S
DRD3 DRD4 DRD5 DYRK1A DYRK1B
DYRK2 EBI2 EDG1 EDG2 EDG3
EDG4 EDG5 EDG6 EDG7 EDNRA
EDNRB EGFR EGFR(E746-A750del) EGFR(G719C) EGFR(G719S)
EGFR(L747-E749del, A750P) EGFR(L747-S752del, P753S) EGFR(L747-T751del,Sins) EGFR(L858R) EGFR(L858R,T790M)
EGFR(L861Q) EGFR(S752-I759del) EGFR(T790M) EGFR/EGFR EGFR/ErbB2
EGFR/ErbB3 EIF2AK1 EP300 EP300 EPHA1
EPHA2 EPHA3 EphA4 EphA5 EPHA6
EphA7 EPHA8 EphB1 EphB2 EphB3
EphB4 EPHB6 EpoR/EpoR EpoR-JAK2 ErbB1
ERBB2 ErbB2/ErbB3 ErbB2/ErbB4 ErbB2-ErbB3 ERBB3
ErbB4 ErbB4/ErbB4 ERK1 ERK1(Q122L) ERK2
ERK3 ERK4 ERK5 ERK8 ERN1
ERRα ERα F2R F2RL1 F2RL3
FAK FALZ FALZ FER FES
FFAR1 FFAR2 FFAR3 FGFR1 FGFR1-α-Klotho
FGFR1-β-Klotho FGFR2 FGFR2(N550K) FGFR3 FGFR3(G380R)/FGFR3(G380R)
FGFR3(G697C) FGFR3(K650E) FGFR3(V555M) FGFR3/FGFR3 FGFR4
FGFR4 FGFR4-α-Klotho FGFR4-β-Klotho FGR FLT1
FLT3 FLT3(D835H) FLT3(D835V) FLT3(D835Y) FLT3(ITD)
FLT3(ITD,D835V) FLT3(ITD,F691L) FLT3(K663Q) FLT3(N841I) FLT3(R834Q)
FLT3-autoinhibited FLT4 FOXO3 FPR1 FPR3
FPRL1 FRK FSHR FXR FYN
G9a GABBR1-GABBR2 GAK GALR1 GALR2
GCGR GCN2(Kin.Dom.2,S808G) GCN5L2 GHRHR GHR-JAK1
GHR-JAK2 GHSR GHSR1b GIPR GLP
GLP1R GLP2R GNRHR GPBAR1 GPR1
GPR101 GPR103 GPR107 GPR109A GPR109B
GPR119 GPR12 GPR120 GPR120S GPR123
GPR132 GPR135 GPR137 GPR139 GPR141
GPR142 GPR143 GPR146 GPR148 GPR149
GPR15 GPR150 GPR151 GPR152 GPR157
GPR161 GPR162 GPR17 GPR171 GPR173
GPR176 GPR18 GPR182 GPR20 GPR22
GPR23 GPR25 GPR26 GPR27 GPR3
GPR30 GPR31 GPR32 GPR35 GPR37
GPR37L1 GPR39 GPR4 GPR45 GPR50
GPR52 GPR55 GPR6 GPR61 GPR65
GPR75 GPR78 GPR79 GPR81 GPR83
GPR84 GPR85 GPR88 GPR92 GPR97
GR GRK1 GRK2 GRK3 GRK4
GRK7 GRM1 GRM2 GRM3 GRM4
GRM5 GRM6 GRPR GSK3A GSK3B
HASPIN HCK HCRTR1 HCRTR2 HIPK1
HIPK2 HIPK3 HIPK4 HPK1 HRH1
HRH2 HRH3 HRH4 HTR1A HTR1B
HTR1E HTR1F HTR2A HTR2B HTR2C
HTR2C(VGV) HTR2C(VNV) HTR2C(VSV) HTR5A HTR6
HTR7A HTR7B HTR7D HUNK ICK
IFNAR1/IFNAR2 IFNGR1/IFNGR2 IFNRL1/IL10RB IGF1R IKK-alpha
IKK-beta IKK-epsilon IL10RA/IL10RB IL11RA/IL6ST IL12RB1/IL12RB2
IL17RA/IL17RC IL17RD/TNFR2 IL18R1/IL18RAP IL1R1/IL1RAP IL1RL1/IL1RAP
IL20RA/IL10RB IL20RA/IL20RB IL21R/IL2RG IL22RA1/IL10RB IL23R/IL12RB1
IL27RA/IL6ST IL2RB/IL2RG IL2RB/IL2RG/IL2RA IL31RA/OSMRb IL3RA/CD131
IL4R/IL13RA1 IL4R/IL2RG IL5RA/CD131 IL6R/IL6ST IL7R/CRLF2
IL7R/IL2RG IL9R/IL2RG INSR INSRa INSRb
INSRR IRAK1 IRAK2 IRAK3 IRAK4
ITK IκB JAK1(JH1domain-catalytic) JAK1(JH2domain-pseudokinase) JAK2(JH1domain-catalytic)
JAK3 JAK3(JH1domain-catalytic) JNK1 JNK2 JNK3
KCNH2(G601S) KDR KDR/KDR Keap1-NRF2 KISS1R
KIT KIT(A829P) KIT(D816H) KIT(D816V) KIT(L576P)
KIT(V559D) KIT(V559D,T670I) KIT(V559D,V654A) KIT-autoinhibited LATS1
LATS2 LCK LGR4 LGR5 LGR6
LHCGR LIMK1 LIMK2 LKB1 LOK
LRRK2 LRRK2(G2019S) LTB4R LTK LXRα
LXRβ LXRβ-NCoR1 LYN LZK mADCYAP1R1
mADORA2B mADORA3 mADRA1B mAGTRL1 MAK
MAP3K1 MAP3K15 MAP3K2 MAP3K3 MAP3K4
MAP4K2 MAP4K3 MAP4K4 MAP4K5 MAPKAPK2
MAPKAPK5 MARK1 MARK2 MARK3 MARK4
MAST1 mAVPR2 mBRS3 MC1R MC3R
MC4R MC4R(T162I) mC5AR1 MC5R mCCKAR
mCCR1 mCCR2 mCCR3 mCCR4 mCCR5
mCCR6 mCCR7 mCCR8 mCCR9 MCHR1
MCHR2 MCL1-BIM mCMKLR1 mCNR1 mCNR2
mCRHR1 mCRTH2 mCX3CR1 mCXCR2 mCXCR3
mCXCR4 mCXCR5 mCXCR6 mCXCR7 mDRD5
mEBI2 mEDG1 mEDG3 mEDG5 mEDNRA
mEDNRB MEK1 MEK2 MEK3 MEK4
MEK5 MEK6 MELK MERTK MET
MET(M1250T) MET(Y1235D) mF2RL1 mFFAR1 mFPR1
mFPR2 mGALR1 mGALR2 mGCGR mGHSR
mGIPR mGLP1R mGLP1R-ADCY2 mGPR1 mGPR120
mGPR84 mHCRTR1 mHTR2A mHTR2C MINK
mINSRa mINSRb MKK7 MKNK1 MKNK2
MLCK MLK1 MLK2 MLK3 MLKL
MLKL(full-length) MLL MLNR mLTB4R mMC3R
mMC4R mMC5R mMCHR1 mNPY1R mNPY2R
mOPRD1 mOPRK1 mOPRM1 mOXTR mP2RY12
mP2RY6 mPPYR1 mPTAFR mPTGER4 mPTGIR
MR MRCKA MRCKB MRGPRD MRGPRE
MRGPRF MRGPRX1 MRGPRX2 MRGPRX4 mRHO(P23H)
mRXFP1 mRXFP3 mRXFP4 mSSTR2 mSSTR5
MST1 MST1R MST2 MST3 MST4
mTAAR1 mTACR1 MTH1 MTNR1A MTNR1B
MTOR MUSK mUTR2 mVIPR1 MYLK
MYLK2 MYLK4 MYO3A MYO3B NDR1
NDR2 NEK1 NEK10 NEK11 NEK2
NEK3 NEK4 NEK5 NEK6 NEK7
NEK9 NIK NIM1 NLK NMBR
NMU1R NPBWR1 NPBWR2 NPFFR1 NPR1
NPSR1b NPY1R NPY2R NTSR1 OPN5
OPRD1 OPRK1 OPRL1 OPRM1 OSMR/IL6ST
OSR1 OX40 OXER1 OXGR1 OXTR
P2RY1 P2RY11 P2RY12 P2RY2 P2RY4
P2RY6 P2RY8 p38-alpha p38-beta p38-delta
p38-gamma P53 PAK1 PAK2 PAK3
PAK4 PAK6 PAK7 PASK PB1(1)
PB1(2) PBRM1(2) PBRM1(5) PCAF PCTK1
PCTK2 PCTK3 PD-1 PDGFRa PDGFRb
PD-L1 PD-L1/PD-L1 PD-L2 PDPK1 PFCDPK1(P.falciparum)
PFPK5(P.falciparum) PFTAIRE2 PFTK1 PHIP(1) PHIP(2)
PHKG1 PHKG2 PI3Kδ PIK3C2B PIK3C2G
PIK3CA PIK3CA(C420R) PIK3CA(E542K) PIK3CA(E545A) PIK3CA(E545K)
PIK3CA(H1047L) PIK3CA(H1047Y) PIK3CA(I800L) PIK3CA(M1043I) PIK3CA(Q546K)
PIK3CB PIK3CD PIK3CG PIK4CB PIKFYVE
PIM1 PIM2 PIM3 PIP5K1A PIP5K1C
PIP5K2B PIP5K2C PKAC-alpha PKAC-alpha(L206R) PKAC-beta
PKMYT1 PKN1 PKN2 PKNB(M.tuberculosis) PLK1
PLK2 PLK3 PLK4 PPARα PPARγ
PPARδ PPYR1 PRKCBP1 PRKCD PRKCE
PRKCH PRKCI PRKCQ PRKD1 PRKD2
PRKD3 PRKG1 PRKG2 PRKR PRKX
PRLHR PRLR-JAK1 PRLR-JAK2 PRMT3 PROKR1
PROKR2 PRP4 PRα PRβ PTAFR
PTGDR PTGER1 PTGER2 PTGER3 PTGER4
PTGFR PTGIR PTHR1 PTHR2 PYK2
QSK RAF1 RANK-IκB RARα RARβ
rCHRM4 rCNR2 rCRTH2 rDRD1 rDRD2L
rDRD2S rEDG5 RELA-IκB RET RET(A883F)
RET(M918T) RET(V804E) RET(V804L) RET(V804M) rFFAR1
rGPR120 rGPR35 rHTR2C rhTrkA-rhP75 RIOK1
RIOK2 RIOK3 RIPK1 RIPK1 RIPK2
RIPK3 RIPK3 RIPK4 RIPK5 ROCK1
ROCK2 rOPRM1 ROS1 rPROKR1 rPROKR2
RPS6KA4(Kin.Dom.1-N-terminal) RPS6KA4(Kin.Dom.2-C-terminal) RPS6KA5(Kin.Dom.1-N-terminal) RPS6KA5(Kin.Dom.2-C-terminal) rPTGER4
RSK1(Kin.Dom.1-N-terminal) RSK1(Kin.Dom.2-C-terminal) RSK2(Kin.Dom.1-N-terminal) RSK2(Kin.Dom.2-C-terminal) RSK3(Kin.Dom.1-N-terminal)
RSK3(Kin.Dom.2-C-terminal) RSK4(Kin.Dom.1-N-terminal) RSK4(Kin.Dom.2-C-terminal) rTAAR1 rTrkA-rP75
rVIPR1 RXFP1 RXFP2 RXFP3 RXFP4
RXRα RXRγ S6K1 SBK1 SCTR
sEDG5 SGK SgK110 SGK2 SGK3
SIK SIK1 SIK2 SLK SMARCA2
SMARCA4 SMO(W535L) SNARK SNRK SP110
SP140 SRC SREBP2 SRMS SRPK1
SRPK2 SRPK3 SSTR1 SSTR2 SSTR3
SSTR4 SSTR5 STK16 STK33 STK35
STK36 STK39 SYK TAAR1 TAAR5
TACR1 TACR2 TACR3 TAF1(1,2) TAF1(2)
TAF1L(1) TAF1L(2) TAK1 TAOK1 TAOK2
TAOK3 TBK1 TBXA2R TEC TESK1
TGFBR1 TGFBR1/ACVR2 TGFBR1/ACVR2B TGFBR1/TGFBR2 TGFBR1/TGFBR2/ENG
TGFBR2 THRα THRβ TIE1 TIE2
Tie2 TIM3/TIM3 TLK1 TLK2 TNFα
TNIK TNK1 TNK2 TNNI3K TORC1
TORC2 TPOR/TPOR TRHR TRIM24(Bromo.) TRIM24(PHD,Bromo.)
TRIM33 TRIM33(PHD,Bromo.) TrkA TrkA-P75 TrkB
TrkB-P75 TrkC TrkC-P75 TRPM6 TSHR(L)
TSSK1B TSSK3 TTK TXK TYK2
TYK2(JH1domain-catalytic) TYK2(JH2domain-pseudokinase) TYRO3 ULK1 ULK2
ULK3 UTR2 VEGFR2 VIPR1 VIPR2
VISTA/VISTA VPS34 VRK2 WDR9(1) WDR9(2)
WEE1 WEE2 WNK1 WNK2 WNK3
WNK4 XBP1 XCR1 YANK1 YANK2
YANK3 YES YES1 YSK1 YSK4
ZAK ZAP70 β-Catenin