TGR5 Receptor Agonist

TGR5 Receptor Agonist is a synthetic cell-permeable small molecule agonist for the G protein-coupled bile acid receptor TGR5 (pEC50=6.8-7.5nM). Improves glucagon like peptide-1 (GLP-1) secretion from intestinal cells, and mediates energy balance, inflammation, and digestion.

Catalog No. Size Price Quantity
92-1196 5 mg $534.00

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TGR5 Receptor Agonist
Compound Type
Cells were plated in a 384-well plate and incubated overnight at 37°C/5% CO₂ to allow the cells to attach and grow. Cells were then stimulated with a control agonist, using the assay conditions described below. Following stimulation, signal was detected using the PathHunter Detection Kit according to the recommended protocol.