JQ1 is a chemical compound which is under development as a non-hormonal male contraceptive drug. Its chemical structure is a triazolothienodiazepine, a series originally discovered by Mitsubishi Pharma [WO/2009/084693], related to benzodiazepinederivatives such as etizolam, however JQ1 does not produce sedative or anxiolytic effects and is instead a potent and selective inhibitor of the bromodomain testis-specific protein BRDT, which is essential for chromatin remodeling during spermatogenesis.

Catalog No. Size Price Quantity
92-1149 1 mg $87.00

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Compound Type
≤ -20◦C Please avoid multiple freeze/thaw cycles.
The above data is a representative example from a Eurofins DiscoverX cell-based assay that uses this ligand.