ChemiBrite™ FFA1/GPR40 Free Fatty Acid Receptor Stable Cell Line

FFA1/GPR40 is a Gi/Gq-coupled GPCR that is activated by free medium and long-chain fatty acids. FFA1 receptors are expressed in brain tissue and insulin-producing β Pancreatic islets (Briscoe et al., 2003). FFA1 receptors regulate insulin release from islets in response to long-chain fatty acids in the plasma (reviewed in Brown et al., 2005). Cloned human FFA1 receptor-expressing ChemiBrite cells were made by stable transfection of HEK293 cells with ChemiBrite clytin and the FFA1 receptor. These stability-tested cells are ready for luminescent and fluorescent analysis of agonists, antagonists and modulators at the FFA1 receptor.

Catalog No. Size Price Quantity
HTS038L 2 Vials $18,779.00

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Calcium Flux Assay, cAMP Accumulation
Free Fatty Acid
Accession Number
Host Cell Type
HEK 293
2 Vials of mycoplasma-free cells, 1 ml per vial
Cell vials are to be stored in the vapor phase of liquid N2.
  • [User Manual] ChemiSCREEN™ and ChemiBRITE™ Cell Lines

    The ChemiSCREEN and ChemiBRITE Cell Lines are designed to enable the measurement of intracellular calcium levels when a GPCR of interest has been activated by a ligand. These cell lines are suitable for studying small molecules as well as biologics. The assay protocol has been optimized for use in either a 384-well or 96-well format.

    ChemiSCREEN and ChemiBRITE cells stably expres...

    [User Manual] ChemiSCREEN™ and ChemiBRITE™ Cell Lines