KINOMEscan® RET(A883F)

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Panel:

Target/Description
ret proto-oncogene
Group
TK
Kinase Construct
Partial Length
Accession Number
NP_065681.1
Species
Human
Kinase Form
Mutation(A883F)
Expression System
Bacterial
Amino Acid Start/Stop
E713/D1014

Reference Inhibitor Information (all values in nM)

Compound
KD
CHIR-258
29
Ponatinib
5.6