KINOMEscan® KIT(V559D,V654A)

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Panel:

Target/Description
v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog
Group
TK
Kinase Construct
Partial Length
Accession Number
NP_000213.1
Species
Human
Kinase Form
Mutation (V559D,V654A)
Expression System
Bacterial
Amino Acid Start/Stop
Y545/D952

Assay Information

Average Z' Panel
0.71

Reference Inhibitor Information (all values in nM)

Compound
KD
Sunitinib
0.21
AMG-706
23
MLN-518
26
Imatinib
71
AST-487
100
PKC-412
1600